Composiciones farmacéuticas que comprenden everolimus

Una formulación farmacéutica que comprende una primera parte y una segunda parte, en la que la primera parte comprende una capa con, en base al peso de la capa, más del 40% en peso de 40-O-(2-hidroxi)etil-rapamicina, y la segunda parte libera más de 85% en peso de 40-O-(2-hidroxi)etil-rapamicina de...

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Hauptverfasser: KUNZLER, Hans-Ulrich, DIEDERICH, Anke, GRANER, Oliver
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creator KUNZLER, Hans-Ulrich
DIEDERICH, Anke
GRANER, Oliver
description Una formulación farmacéutica que comprende una primera parte y una segunda parte, en la que la primera parte comprende una capa con, en base al peso de la capa, más del 40% en peso de 40-O-(2-hidroxi)etil-rapamicina, y la segunda parte libera más de 85% en peso de 40-O-(2-hidroxi)etil-rapamicina de la segunda parte en menos de 60 minutos. The invention relates to a pharmaceutical formulation comprising 40-O-(2-hydroxy)ethyl-rapamycin in a high drug load part and an immediate release part. In addition, the invention relates to a formulation comprising 40-O-(2-hydroxy)ethyl-rapamycin in a first layer and a surfactant in a layer beneath the first layer. The pharmaceutical composition is particularly suitable for use as a medicament.
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subjects HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
title Composiciones farmacéuticas que comprenden everolimus
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