DERIVADOS DE 1H-INDOL-3-ACETAMIDAS COMO INHIBIDORES DE SPLA2
SE DESCRIBE UNA CLASE DE DERIVADOS DE ACIDO 1H 3 ACETOAMIDAS, REPRESENTADO POR LA FORMULA (I), Y SALES FARMACEUTICAMENTE ACEPTABLES DE ELLOS; JUNTO CON EL USO DE TALES COMPUESTOS INDOLO PARA INHIBIR SPLA2 MEDIADO POR LIBERACION DE ACIDOS GRASOS PARA TRATAMIENTO DE CONDICIONES TALES COMO CHOQUE SEPTI...
Gespeichert in:
Hauptverfasser: | , , , , |
---|---|
Format: | Patent |
Sprache: | spa |
Schlagworte: | |
Online-Zugang: | Volltext bestellen |
Tags: |
Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!
|
container_end_page | |
---|---|
container_issue | |
container_start_page | |
container_title | |
container_volume | |
creator | DILLARD, ROBERT DELANE BACH, NICHOLAS JAMES DRAHEIM, SUSAN ELIZABETH SCHEVITZ, RICHARD WALTER HERMANN, ROBERT BELL |
description | SE DESCRIBE UNA CLASE DE DERIVADOS DE ACIDO 1H 3 ACETOAMIDAS, REPRESENTADO POR LA FORMULA (I), Y SALES FARMACEUTICAMENTE ACEPTABLES DE ELLOS; JUNTO CON EL USO DE TALES COMPUESTOS INDOLO PARA INHIBIR SPLA2 MEDIADO POR LIBERACION DE ACIDOS GRASOS PARA TRATAMIENTO DE CONDICIONES TALES COMO CHOQUE SEPTICO.
A class of 1H-indole-3-acetamides, represented by the formula (I), and pharmaceutically acceptable salts thereof; is disclosed together with the use of such indole compounds for inhibiting sPLA2 mediated release of fatty acids for treatment of conditions such as septic shock. |
format | Patent |
fullrecord | <record><control><sourceid>epo_EVB</sourceid><recordid>TN_cdi_epo_espacenet_ES2138648TT3</recordid><sourceformat>XML</sourceformat><sourcesystem>PC</sourcesystem><sourcerecordid>ES2138648TT3</sourcerecordid><originalsourceid>FETCH-epo_espacenet_ES2138648TT33</originalsourceid><addsrcrecordid>eNrjZLBxcQ3yDHN08Q9WcHFVMPTQ9fRz8ffRNdZ1dHYNcfT1dHEMVnD29_VX8PTz8HTydPEPcgWrDA7wcTTiYWBNS8wpTuWF0twMim6uIc4euqkF-fGpxQWJyal5qSXxrsFGhsYWZiYWISHGxsSoAQC3FilN</addsrcrecordid><sourcetype>Open Access Repository</sourcetype><iscdi>true</iscdi><recordtype>patent</recordtype></control><display><type>patent</type><title>DERIVADOS DE 1H-INDOL-3-ACETAMIDAS COMO INHIBIDORES DE SPLA2</title><source>esp@cenet</source><creator>DILLARD, ROBERT DELANE ; BACH, NICHOLAS JAMES ; DRAHEIM, SUSAN ELIZABETH ; SCHEVITZ, RICHARD WALTER ; HERMANN, ROBERT BELL</creator><creatorcontrib>DILLARD, ROBERT DELANE ; BACH, NICHOLAS JAMES ; DRAHEIM, SUSAN ELIZABETH ; SCHEVITZ, RICHARD WALTER ; HERMANN, ROBERT BELL</creatorcontrib><description>SE DESCRIBE UNA CLASE DE DERIVADOS DE ACIDO 1H 3 ACETOAMIDAS, REPRESENTADO POR LA FORMULA (I), Y SALES FARMACEUTICAMENTE ACEPTABLES DE ELLOS; JUNTO CON EL USO DE TALES COMPUESTOS INDOLO PARA INHIBIR SPLA2 MEDIADO POR LIBERACION DE ACIDOS GRASOS PARA TRATAMIENTO DE CONDICIONES TALES COMO CHOQUE SEPTICO.
A class of 1H-indole-3-acetamides, represented by the formula (I), and pharmaceutically acceptable salts thereof; is disclosed together with the use of such indole compounds for inhibiting sPLA2 mediated release of fatty acids for treatment of conditions such as septic shock.</description><edition>7</edition><language>spa</language><subject>ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAININGELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN,SULFUR, SELENIUM OR TELLURIUM ; CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>2000</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20000116&DB=EPODOC&CC=ES&NR=2138648T3$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,776,881,25542,76290</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20000116&DB=EPODOC&CC=ES&NR=2138648T3$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>DILLARD, ROBERT DELANE</creatorcontrib><creatorcontrib>BACH, NICHOLAS JAMES</creatorcontrib><creatorcontrib>DRAHEIM, SUSAN ELIZABETH</creatorcontrib><creatorcontrib>SCHEVITZ, RICHARD WALTER</creatorcontrib><creatorcontrib>HERMANN, ROBERT BELL</creatorcontrib><title>DERIVADOS DE 1H-INDOL-3-ACETAMIDAS COMO INHIBIDORES DE SPLA2</title><description>SE DESCRIBE UNA CLASE DE DERIVADOS DE ACIDO 1H 3 ACETOAMIDAS, REPRESENTADO POR LA FORMULA (I), Y SALES FARMACEUTICAMENTE ACEPTABLES DE ELLOS; JUNTO CON EL USO DE TALES COMPUESTOS INDOLO PARA INHIBIR SPLA2 MEDIADO POR LIBERACION DE ACIDOS GRASOS PARA TRATAMIENTO DE CONDICIONES TALES COMO CHOQUE SEPTICO.
A class of 1H-indole-3-acetamides, represented by the formula (I), and pharmaceutically acceptable salts thereof; is disclosed together with the use of such indole compounds for inhibiting sPLA2 mediated release of fatty acids for treatment of conditions such as septic shock.</description><subject>ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAININGELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN,SULFUR, SELENIUM OR TELLURIUM</subject><subject>CHEMISTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>HUMAN NECESSITIES</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><subject>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><subject>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2000</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNrjZLBxcQ3yDHN08Q9WcHFVMPTQ9fRz8ffRNdZ1dHYNcfT1dHEMVnD29_VX8PTz8HTydPEPcgWrDA7wcTTiYWBNS8wpTuWF0twMim6uIc4euqkF-fGpxQWJyal5qSXxrsFGhsYWZiYWISHGxsSoAQC3FilN</recordid><startdate>20000116</startdate><enddate>20000116</enddate><creator>DILLARD, ROBERT DELANE</creator><creator>BACH, NICHOLAS JAMES</creator><creator>DRAHEIM, SUSAN ELIZABETH</creator><creator>SCHEVITZ, RICHARD WALTER</creator><creator>HERMANN, ROBERT BELL</creator><scope>EVB</scope></search><sort><creationdate>20000116</creationdate><title>DERIVADOS DE 1H-INDOL-3-ACETAMIDAS COMO INHIBIDORES DE SPLA2</title><author>DILLARD, ROBERT DELANE ; BACH, NICHOLAS JAMES ; DRAHEIM, SUSAN ELIZABETH ; SCHEVITZ, RICHARD WALTER ; HERMANN, ROBERT BELL</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_ES2138648TT33</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>spa</language><creationdate>2000</creationdate><topic>ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAININGELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN,SULFUR, SELENIUM OR TELLURIUM</topic><topic>CHEMISTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>HUMAN NECESSITIES</topic><topic>HYGIENE</topic><topic>MEDICAL OR VETERINARY SCIENCE</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><topic>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</topic><topic>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</topic><toplevel>online_resources</toplevel><creatorcontrib>DILLARD, ROBERT DELANE</creatorcontrib><creatorcontrib>BACH, NICHOLAS JAMES</creatorcontrib><creatorcontrib>DRAHEIM, SUSAN ELIZABETH</creatorcontrib><creatorcontrib>SCHEVITZ, RICHARD WALTER</creatorcontrib><creatorcontrib>HERMANN, ROBERT BELL</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>DILLARD, ROBERT DELANE</au><au>BACH, NICHOLAS JAMES</au><au>DRAHEIM, SUSAN ELIZABETH</au><au>SCHEVITZ, RICHARD WALTER</au><au>HERMANN, ROBERT BELL</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>DERIVADOS DE 1H-INDOL-3-ACETAMIDAS COMO INHIBIDORES DE SPLA2</title><date>2000-01-16</date><risdate>2000</risdate><abstract>SE DESCRIBE UNA CLASE DE DERIVADOS DE ACIDO 1H 3 ACETOAMIDAS, REPRESENTADO POR LA FORMULA (I), Y SALES FARMACEUTICAMENTE ACEPTABLES DE ELLOS; JUNTO CON EL USO DE TALES COMPUESTOS INDOLO PARA INHIBIR SPLA2 MEDIADO POR LIBERACION DE ACIDOS GRASOS PARA TRATAMIENTO DE CONDICIONES TALES COMO CHOQUE SEPTICO.
A class of 1H-indole-3-acetamides, represented by the formula (I), and pharmaceutically acceptable salts thereof; is disclosed together with the use of such indole compounds for inhibiting sPLA2 mediated release of fatty acids for treatment of conditions such as septic shock.</abstract><edition>7</edition><oa>free_for_read</oa></addata></record> |
fulltext | fulltext_linktorsrc |
identifier | |
ispartof | |
issn | |
language | spa |
recordid | cdi_epo_espacenet_ES2138648TT3 |
source | esp@cenet |
subjects | ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAININGELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN,SULFUR, SELENIUM OR TELLURIUM CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
title | DERIVADOS DE 1H-INDOL-3-ACETAMIDAS COMO INHIBIDORES DE SPLA2 |
url | https://sfx.bib-bvb.de/sfx_tum?ctx_ver=Z39.88-2004&ctx_enc=info:ofi/enc:UTF-8&ctx_tim=2025-02-01T23%3A40%3A36IST&url_ver=Z39.88-2004&url_ctx_fmt=infofi/fmt:kev:mtx:ctx&rfr_id=info:sid/primo.exlibrisgroup.com:primo3-Article-epo_EVB&rft_val_fmt=info:ofi/fmt:kev:mtx:patent&rft.genre=patent&rft.au=DILLARD,%20ROBERT%20DELANE&rft.date=2000-01-16&rft_id=info:doi/&rft_dat=%3Cepo_EVB%3EES2138648TT3%3C/epo_EVB%3E%3Curl%3E%3C/url%3E&disable_directlink=true&sfx.directlink=off&sfx.report_link=0&rft_id=info:oai/&rft_id=info:pmid/&rfr_iscdi=true |