HISTONE ACETYLASE P300 INHIBITOR AND USE THEREOF
Provided are a histone acetylase p300 inhibitor and a use thereof, belonging to the filed of medicinal chemistry technology. A compound represented by formula (I), or a stereochemical isomer thereof, or a solvate thereof, or a pharmaceutically acceptable salt thereof, can inhibit the activity of his...
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| creator | ZHANG, Shaohua DU, Wu HUO, Yongxu WU, Xiaoquan FAN, Lei ZHANG, Chengzhi CHEN, Ke LI, Xinghai XU, Kexin WANG, Fei LUO, Tongchuan CHEN, Yuanwei TU, Zhilin |
| description | Provided are a histone acetylase p300 inhibitor and a use thereof, belonging to the filed of medicinal chemistry technology. A compound represented by formula (I), or a stereochemical isomer thereof, or a solvate thereof, or a pharmaceutically acceptable salt thereof, can inhibit the activity of histone acetylase p300 and inhibit the proliferation activity of a variety of tumor cells. |
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| subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| title | HISTONE ACETYLASE P300 INHIBITOR AND USE THEREOF |
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