PROCESS AND INTERMEDIATES FOR THE PREPARATION OF BENZO[B]THIOPHENE COMPOUNDS

A process for preparing compounds of formula (I), or a salt or solvate thereof, including Brexpiprazole, which process comprises cyclization of a compound of formula (II) or (III), or a salt or solvate thereof. The invention also refers to intermediates of said process.

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Hauptverfasser: PÉREZ ENCABO, Alfonso, LORENTE BONDE-LARSEN, Antonio, TURIEL HERNANDEZ, José Angel, FERNÁNDEZ SAINZ, Yolanda
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Sprache:eng ; fre ; ger
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creator PÉREZ ENCABO, Alfonso
LORENTE BONDE-LARSEN, Antonio
TURIEL HERNANDEZ, José Angel
FERNÁNDEZ SAINZ, Yolanda
description A process for preparing compounds of formula (I), or a salt or solvate thereof, including Brexpiprazole, which process comprises cyclization of a compound of formula (II) or (III), or a salt or solvate thereof. The invention also refers to intermediates of said process.
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subjects CHEMISTRY
HETEROCYCLIC COMPOUNDS
METALLURGY
ORGANIC CHEMISTRY
title PROCESS AND INTERMEDIATES FOR THE PREPARATION OF BENZO[B]THIOPHENE COMPOUNDS
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