PYRAZOLE DERIVATIVE AND USE THEREOF FOR MEDICAL PURPOSES

PYRAZOLE DERIVATIVE AND USE THEREOF FOR MEDICAL PURPOSES

The present invention provides pyrazole derivatives, uses thereof for for medical purposes and so on. More particularly, the present invention relates to pharmaceuticals useful for the prevention or treatment of constipation, which comprise as an active ingredient 3-(3-{4-[3-(²-D-glucopyranosyloxy)-...

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Hauptverfasser: TAKEMURA, MASAAKI, MIYASHITA, ITARU, HOTEI, YUKIHIKO, ISAJI, MASAYUKI, ISAWA, HIDETOSHI
Format: Patent
Sprache:eng ; fre ; ger
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HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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creator TAKEMURA, MASAAKI
MIYASHITA, ITARU
HOTEI, YUKIHIKO
ISAJI, MASAYUKI
ISAWA, HIDETOSHI
description The present invention provides pyrazole derivatives, uses thereof for for medical purposes and so on. More particularly, the present invention relates to pharmaceuticals useful for the prevention or treatment of constipation, which comprise as an active ingredient 3-(3-{4-[3-(²-D-glucopyranosyloxy)-5-isopropyl-1H-pyrazol-4-ylmethyl]-3-methylphenoxy}propylamino)-2,2-dimethylpropionamide, or a pharmaceutically acceptable salt thereof. The pharmaceuticals of the present invention exert an effect of increasing the frequency of bowel movement or the like, and are useful for the prevention or treatment of constipation.
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subjects HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
title PYRAZOLE DERIVATIVE AND USE THEREOF FOR MEDICAL PURPOSES
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