HETERO RING-FUSED IMIDAZOLE DERIVATIVE HAVING AMPK ACTIVATING EFFECT
Disclosed is a compound which is useful as an AMPK activator. A compound represented by the formula: its pharmaceutically acceptable salt, or a solvate thereof, wherein a group represented by the formula: is a group represented by the formula: R 1 is each independently halogen, hydroxy, cyano, nitro...
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| creator | IWATSU, MASAFUMI INO, AKIRA TONOGAKI, KEISUKE KOJIMA, EIICHI FUJIOKA, MASAHIKO KATOU, MANABU TANAKA, NOBUYUKI |
| description | Disclosed is a compound which is useful as an AMPK activator. A compound represented by the formula:
its pharmaceutically acceptable salt, or a solvate thereof,
wherein
a group represented by the formula:
is a group represented by the formula:
R 1 is each independently halogen, hydroxy, cyano, nitro, carboxy, substituted or unsubstituted alkyl, substituted or unsubstituted alkenyl or the like;
m is an integer of 0 to 3;
R 2 is hydrogen, or substituted or unsubstituted alkyl;
X is -O-; and
Y is substituted or unsubstituted aryl, or substituted or unsubstituted heteroaryl. |
| format | Patent |
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its pharmaceutically acceptable salt, or a solvate thereof,
wherein
a group represented by the formula:
is a group represented by the formula:
R 1 is each independently halogen, hydroxy, cyano, nitro, carboxy, substituted or unsubstituted alkyl, substituted or unsubstituted alkenyl or the like;
m is an integer of 0 to 3;
R 2 is hydrogen, or substituted or unsubstituted alkyl;
X is -O-; and
Y is substituted or unsubstituted aryl, or substituted or unsubstituted heteroaryl.</description><language>eng ; fre ; ger</language><subject>CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>2016</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20160323&DB=EPODOC&CC=EP&NR=2617722B1$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,776,881,25542,76289</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20160323&DB=EPODOC&CC=EP&NR=2617722B1$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>IWATSU, MASAFUMI</creatorcontrib><creatorcontrib>INO, AKIRA</creatorcontrib><creatorcontrib>TONOGAKI, KEISUKE</creatorcontrib><creatorcontrib>KOJIMA, EIICHI</creatorcontrib><creatorcontrib>FUJIOKA, MASAHIKO</creatorcontrib><creatorcontrib>KATOU, MANABU</creatorcontrib><creatorcontrib>TANAKA, NOBUYUKI</creatorcontrib><title>HETERO RING-FUSED IMIDAZOLE DERIVATIVE HAVING AMPK ACTIVATING EFFECT</title><description>Disclosed is a compound which is useful as an AMPK activator. A compound represented by the formula:
its pharmaceutically acceptable salt, or a solvate thereof,
wherein
a group represented by the formula:
is a group represented by the formula:
R 1 is each independently halogen, hydroxy, cyano, nitro, carboxy, substituted or unsubstituted alkyl, substituted or unsubstituted alkenyl or the like;
m is an integer of 0 to 3;
R 2 is hydrogen, or substituted or unsubstituted alkyl;
X is -O-; and
Y is substituted or unsubstituted aryl, or substituted or unsubstituted heteroaryl.</description><subject>CHEMISTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>HUMAN NECESSITIES</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><subject>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><subject>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2016</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNrjZHDxcA1xDfJXCPL0c9d1Cw12dVHw9PV0cYzy93FVcHEN8gxzDPEMc1XwcAwDqlBw9A3wVnB0DgELA_mubm6uziE8DKxpiTnFqbxQmptBwc01xNlDN7UgPz61uCAxOTUvtSTeNcDIzNDc3MjIydCYCCUAAUsrVA</recordid><startdate>20160323</startdate><enddate>20160323</enddate><creator>IWATSU, MASAFUMI</creator><creator>INO, AKIRA</creator><creator>TONOGAKI, KEISUKE</creator><creator>KOJIMA, EIICHI</creator><creator>FUJIOKA, MASAHIKO</creator><creator>KATOU, MANABU</creator><creator>TANAKA, NOBUYUKI</creator><scope>EVB</scope></search><sort><creationdate>20160323</creationdate><title>HETERO RING-FUSED IMIDAZOLE DERIVATIVE HAVING AMPK ACTIVATING EFFECT</title><author>IWATSU, MASAFUMI ; INO, AKIRA ; TONOGAKI, KEISUKE ; KOJIMA, EIICHI ; FUJIOKA, MASAHIKO ; KATOU, MANABU ; TANAKA, NOBUYUKI</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_EP2617722B13</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>eng ; fre ; ger</language><creationdate>2016</creationdate><topic>CHEMISTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>HUMAN NECESSITIES</topic><topic>HYGIENE</topic><topic>MEDICAL OR VETERINARY SCIENCE</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><topic>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</topic><topic>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</topic><toplevel>online_resources</toplevel><creatorcontrib>IWATSU, MASAFUMI</creatorcontrib><creatorcontrib>INO, AKIRA</creatorcontrib><creatorcontrib>TONOGAKI, KEISUKE</creatorcontrib><creatorcontrib>KOJIMA, EIICHI</creatorcontrib><creatorcontrib>FUJIOKA, MASAHIKO</creatorcontrib><creatorcontrib>KATOU, MANABU</creatorcontrib><creatorcontrib>TANAKA, NOBUYUKI</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>IWATSU, MASAFUMI</au><au>INO, AKIRA</au><au>TONOGAKI, KEISUKE</au><au>KOJIMA, EIICHI</au><au>FUJIOKA, MASAHIKO</au><au>KATOU, MANABU</au><au>TANAKA, NOBUYUKI</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>HETERO RING-FUSED IMIDAZOLE DERIVATIVE HAVING AMPK ACTIVATING EFFECT</title><date>2016-03-23</date><risdate>2016</risdate><abstract>Disclosed is a compound which is useful as an AMPK activator. A compound represented by the formula:
its pharmaceutically acceptable salt, or a solvate thereof,
wherein
a group represented by the formula:
is a group represented by the formula:
R 1 is each independently halogen, hydroxy, cyano, nitro, carboxy, substituted or unsubstituted alkyl, substituted or unsubstituted alkenyl or the like;
m is an integer of 0 to 3;
R 2 is hydrogen, or substituted or unsubstituted alkyl;
X is -O-; and
Y is substituted or unsubstituted aryl, or substituted or unsubstituted heteroaryl.</abstract><oa>free_for_read</oa></addata></record> |
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| language | eng ; fre ; ger |
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| subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| title | HETERO RING-FUSED IMIDAZOLE DERIVATIVE HAVING AMPK ACTIVATING EFFECT |
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