PHENYL-HETEROARYL DERIVATIVES AND METHODS OF USE THEREOF
The present invention provides phenyl-heteroaryl derivatives of Formula (I) and pharmaceutically acceptable salts thereof These compounds are useful in the treatment of RAGE-mediated diseases such as Alzheimer's Disease. The present invention further relates to methods for the preparation of co...
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| creator | SUNDERMANN, KURT RAO, MOHAN GUPTA, SUPARNA JONES, DAVID BANNER, WILLIAM, KENNETH BONDLELA, MURALIDHAR WANG, PINGZHEN HARI, ANITHA QABAJA, GHASSAN GOHIMUKKULA, DEVI, REDDY GOWDA, RAJU, BORE ZHU, JEFF, JIQUN ANDREWS, ROBERT, C COOPER, JEREMY, T |
| description | The present invention provides phenyl-heteroaryl derivatives of Formula (I) and pharmaceutically acceptable salts thereof These compounds are useful in the treatment of RAGE-mediated diseases such as Alzheimer's Disease. The present invention further relates to methods for the preparation of compounds of Formula (I) and pharmaceutically acceptable salts thereof, pharmaceutical compositions comprising such compounds, and the use of such compounds and/or pharmaceutical compositions in treating RAGE-mediated diseases. |
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The present invention further relates to methods for the preparation of compounds of Formula (I) and pharmaceutically acceptable salts thereof, pharmaceutical compositions comprising such compounds, and the use of such compounds and/or pharmaceutical compositions in treating RAGE-mediated diseases.</description><language>eng ; fre ; ger</language><subject>CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>2015</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20150729&DB=EPODOC&CC=EP&NR=2536283B1$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,776,881,25542,76290</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20150729&DB=EPODOC&CC=EP&NR=2536283B1$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>SUNDERMANN, KURT</creatorcontrib><creatorcontrib>RAO, MOHAN</creatorcontrib><creatorcontrib>GUPTA, SUPARNA</creatorcontrib><creatorcontrib>JONES, DAVID</creatorcontrib><creatorcontrib>BANNER, WILLIAM, KENNETH</creatorcontrib><creatorcontrib>BONDLELA, MURALIDHAR</creatorcontrib><creatorcontrib>WANG, PINGZHEN</creatorcontrib><creatorcontrib>HARI, ANITHA</creatorcontrib><creatorcontrib>QABAJA, GHASSAN</creatorcontrib><creatorcontrib>GOHIMUKKULA, DEVI, REDDY</creatorcontrib><creatorcontrib>GOWDA, RAJU, BORE</creatorcontrib><creatorcontrib>ZHU, JEFF, JIQUN</creatorcontrib><creatorcontrib>ANDREWS, ROBERT, C</creatorcontrib><creatorcontrib>COOPER, JEREMY, T</creatorcontrib><title>PHENYL-HETEROARYL DERIVATIVES AND METHODS OF USE THEREOF</title><description>The present invention provides phenyl-heteroaryl derivatives of Formula (I) and pharmaceutically acceptable salts thereof These compounds are useful in the treatment of RAGE-mediated diseases such as Alzheimer's Disease. 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The present invention further relates to methods for the preparation of compounds of Formula (I) and pharmaceutically acceptable salts thereof, pharmaceutical compositions comprising such compounds, and the use of such compounds and/or pharmaceutical compositions in treating RAGE-mediated diseases.</abstract><oa>free_for_read</oa></addata></record> |
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| subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| title | PHENYL-HETEROARYL DERIVATIVES AND METHODS OF USE THEREOF |
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