Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof

The present invention provides a compound having an excellent inhibitory action on activation of STAT6 and a pharmaceutical composition thereof. In particular, it provides a compound represented by the following formula (I), a salt thereof or a hydrate of them. In the formula, the groups X,Y,Z,R 1 -...

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Hauptverfasser: OHASHI, YOSHIAKI, TAKASE, YASUTAKA, SAKUMA, YOSHINORI, YOSHIDA, ICHIRO, YONEDA, NAOKI, YOKOHAMA, HIROMITSU, MIYAZAKI, FUTOSHI, KAMATA, JUNICHI, SHIRATO, MANABU, SHIMOKUBO, DAIYA, SUZUKI, SHUICHI, SESHIMO, HIDENORI, MIYAMOTO, MITSUAKI
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creator OHASHI, YOSHIAKI
TAKASE, YASUTAKA
SAKUMA, YOSHINORI
YOSHIDA, ICHIRO
YONEDA, NAOKI
YOKOHAMA, HIROMITSU
MIYAZAKI, FUTOSHI
KAMATA, JUNICHI
SHIRATO, MANABU
SHIMOKUBO, DAIYA
SUZUKI, SHUICHI
SESHIMO, HIDENORI
MIYAMOTO, MITSUAKI
description The present invention provides a compound having an excellent inhibitory action on activation of STAT6 and a pharmaceutical composition thereof. In particular, it provides a compound represented by the following formula (I), a salt thereof or a hydrate of them. In the formula, the groups X,Y,Z,R 1 -R 4 and n are defined as in claim 1.
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In particular, it provides a compound represented by the following formula (I), a salt thereof or a hydrate of them. In the formula, the groups X,Y,Z,R 1 -R 4 and n are defined as in claim 1.</abstract><oa>free_for_read</oa></addata></record>
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subjects ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAININGELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN,SULFUR, SELENIUM OR TELLURIUM
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
title Nitrogen-containing condensed cyclic compound having a pyrazolyl group as a substituent group and pharmaceutical composition thereof
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