SOMATOSTATIN RECEPTOR 1 AND/OR 4 SELECTIVE AGONISTS AND ANTAGONISTS
The invention relates to (hetero)arylsulfonylamino based peptidomimetics of formula (I), wherein R1, R2, R3, A, B, D, Q, k and n are defined as disclosed, or a pharmaceutically acceptable salt or ester thereof. Compounds of formula (I) possess high affinity and selectivity for the somatostatin recep...
Gespeichert in:
| Hauptverfasser: | , , , , , , |
|---|---|
| Format: | Patent |
| Sprache: | eng ; fre ; ger |
| Schlagworte: | |
| Online-Zugang: | Volltext bestellen |
| Tags: |
Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!
|
| container_end_page | |
|---|---|
| container_issue | |
| container_start_page | |
| container_title | |
| container_volume | |
| creator | TOMPERI, JUSSI ENGSTROEM, MIA WURSTER, SIEGFRIED SALO, HARRI TAUBER, ANDREI HAUTAMAEKI, PAEIVI HOFFREN, ANNA-MARJA |
| description | The invention relates to (hetero)arylsulfonylamino based peptidomimetics of formula (I), wherein R1, R2, R3, A, B, D, Q, k and n are defined as disclosed, or a pharmaceutically acceptable salt or ester thereof. Compounds of formula (I) possess high affinity and selectivity for the somatostatin receptor subtypes SSTR1 and/or SSTR4 and can be used for the treatment or diagnosis of diseases or conditions wherein an interaction with SSTR1 and/or SSTR4 is indicated to be useful. |
| format | Patent |
| fullrecord | <record><control><sourceid>epo_EVB</sourceid><recordid>TN_cdi_epo_espacenet_EP1675824A1</recordid><sourceformat>XML</sourceformat><sourcesystem>PC</sourcesystem><sourcerecordid>EP1675824A1</sourcerecordid><originalsourceid>FETCH-epo_espacenet_EP1675824A13</originalsourceid><addsrcrecordid>eNrjZHAO9vd1DPEPDnEM8fRTCHJ1dg0I8Q9SMFRw9HPRBzJMFIJdfVydQzzDXBUc3f39PINDgkFyQBwC4_MwsKYl5hSn8kJpbgYFN9cQZw_d1IL8-NTigsTk1LzUknjXAEMzc1MLIxNHQ2MilAAA0V0rEA</addsrcrecordid><sourcetype>Open Access Repository</sourcetype><iscdi>true</iscdi><recordtype>patent</recordtype></control><display><type>patent</type><title>SOMATOSTATIN RECEPTOR 1 AND/OR 4 SELECTIVE AGONISTS AND ANTAGONISTS</title><source>esp@cenet</source><creator>TOMPERI, JUSSI ; ENGSTROEM, MIA ; WURSTER, SIEGFRIED ; SALO, HARRI ; TAUBER, ANDREI ; HAUTAMAEKI, PAEIVI ; HOFFREN, ANNA-MARJA</creator><creatorcontrib>TOMPERI, JUSSI ; ENGSTROEM, MIA ; WURSTER, SIEGFRIED ; SALO, HARRI ; TAUBER, ANDREI ; HAUTAMAEKI, PAEIVI ; HOFFREN, ANNA-MARJA</creatorcontrib><description>The invention relates to (hetero)arylsulfonylamino based peptidomimetics of formula (I), wherein R1, R2, R3, A, B, D, Q, k and n are defined as disclosed, or a pharmaceutically acceptable salt or ester thereof. Compounds of formula (I) possess high affinity and selectivity for the somatostatin receptor subtypes SSTR1 and/or SSTR4 and can be used for the treatment or diagnosis of diseases or conditions wherein an interaction with SSTR1 and/or SSTR4 is indicated to be useful.</description><edition>7</edition><language>eng ; fre ; ger</language><subject>ACYCLIC OR CARBOCYCLIC COMPOUNDS ; CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><creationdate>2006</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20060705&DB=EPODOC&CC=EP&NR=1675824A1$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,776,881,25542,76289</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20060705&DB=EPODOC&CC=EP&NR=1675824A1$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>TOMPERI, JUSSI</creatorcontrib><creatorcontrib>ENGSTROEM, MIA</creatorcontrib><creatorcontrib>WURSTER, SIEGFRIED</creatorcontrib><creatorcontrib>SALO, HARRI</creatorcontrib><creatorcontrib>TAUBER, ANDREI</creatorcontrib><creatorcontrib>HAUTAMAEKI, PAEIVI</creatorcontrib><creatorcontrib>HOFFREN, ANNA-MARJA</creatorcontrib><title>SOMATOSTATIN RECEPTOR 1 AND/OR 4 SELECTIVE AGONISTS AND ANTAGONISTS</title><description>The invention relates to (hetero)arylsulfonylamino based peptidomimetics of formula (I), wherein R1, R2, R3, A, B, D, Q, k and n are defined as disclosed, or a pharmaceutically acceptable salt or ester thereof. Compounds of formula (I) possess high affinity and selectivity for the somatostatin receptor subtypes SSTR1 and/or SSTR4 and can be used for the treatment or diagnosis of diseases or conditions wherein an interaction with SSTR1 and/or SSTR4 is indicated to be useful.</description><subject>ACYCLIC OR CARBOCYCLIC COMPOUNDS</subject><subject>CHEMISTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>HUMAN NECESSITIES</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><subject>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2006</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNrjZHAO9vd1DPEPDnEM8fRTCHJ1dg0I8Q9SMFRw9HPRBzJMFIJdfVydQzzDXBUc3f39PINDgkFyQBwC4_MwsKYl5hSn8kJpbgYFN9cQZw_d1IL8-NTigsTk1LzUknjXAEMzc1MLIxNHQ2MilAAA0V0rEA</recordid><startdate>20060705</startdate><enddate>20060705</enddate><creator>TOMPERI, JUSSI</creator><creator>ENGSTROEM, MIA</creator><creator>WURSTER, SIEGFRIED</creator><creator>SALO, HARRI</creator><creator>TAUBER, ANDREI</creator><creator>HAUTAMAEKI, PAEIVI</creator><creator>HOFFREN, ANNA-MARJA</creator><scope>EVB</scope></search><sort><creationdate>20060705</creationdate><title>SOMATOSTATIN RECEPTOR 1 AND/OR 4 SELECTIVE AGONISTS AND ANTAGONISTS</title><author>TOMPERI, JUSSI ; ENGSTROEM, MIA ; WURSTER, SIEGFRIED ; SALO, HARRI ; TAUBER, ANDREI ; HAUTAMAEKI, PAEIVI ; HOFFREN, ANNA-MARJA</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_EP1675824A13</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>eng ; fre ; ger</language><creationdate>2006</creationdate><topic>ACYCLIC OR CARBOCYCLIC COMPOUNDS</topic><topic>CHEMISTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>HUMAN NECESSITIES</topic><topic>HYGIENE</topic><topic>MEDICAL OR VETERINARY SCIENCE</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><topic>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</topic><toplevel>online_resources</toplevel><creatorcontrib>TOMPERI, JUSSI</creatorcontrib><creatorcontrib>ENGSTROEM, MIA</creatorcontrib><creatorcontrib>WURSTER, SIEGFRIED</creatorcontrib><creatorcontrib>SALO, HARRI</creatorcontrib><creatorcontrib>TAUBER, ANDREI</creatorcontrib><creatorcontrib>HAUTAMAEKI, PAEIVI</creatorcontrib><creatorcontrib>HOFFREN, ANNA-MARJA</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>TOMPERI, JUSSI</au><au>ENGSTROEM, MIA</au><au>WURSTER, SIEGFRIED</au><au>SALO, HARRI</au><au>TAUBER, ANDREI</au><au>HAUTAMAEKI, PAEIVI</au><au>HOFFREN, ANNA-MARJA</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>SOMATOSTATIN RECEPTOR 1 AND/OR 4 SELECTIVE AGONISTS AND ANTAGONISTS</title><date>2006-07-05</date><risdate>2006</risdate><abstract>The invention relates to (hetero)arylsulfonylamino based peptidomimetics of formula (I), wherein R1, R2, R3, A, B, D, Q, k and n are defined as disclosed, or a pharmaceutically acceptable salt or ester thereof. Compounds of formula (I) possess high affinity and selectivity for the somatostatin receptor subtypes SSTR1 and/or SSTR4 and can be used for the treatment or diagnosis of diseases or conditions wherein an interaction with SSTR1 and/or SSTR4 is indicated to be useful.</abstract><edition>7</edition><oa>free_for_read</oa></addata></record> |
| fulltext | fulltext_linktorsrc |
| identifier | |
| ispartof | |
| issn | |
| language | eng ; fre ; ger |
| recordid | cdi_epo_espacenet_EP1675824A1 |
| source | esp@cenet |
| subjects | ACYCLIC OR CARBOCYCLIC COMPOUNDS CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES |
| title | SOMATOSTATIN RECEPTOR 1 AND/OR 4 SELECTIVE AGONISTS AND ANTAGONISTS |
| url | https://sfx.bib-bvb.de/sfx_tum?ctx_ver=Z39.88-2004&ctx_enc=info:ofi/enc:UTF-8&ctx_tim=2025-02-05T21%3A14%3A03IST&url_ver=Z39.88-2004&url_ctx_fmt=infofi/fmt:kev:mtx:ctx&rfr_id=info:sid/primo.exlibrisgroup.com:primo3-Article-epo_EVB&rft_val_fmt=info:ofi/fmt:kev:mtx:patent&rft.genre=patent&rft.au=TOMPERI,%20JUSSI&rft.date=2006-07-05&rft_id=info:doi/&rft_dat=%3Cepo_EVB%3EEP1675824A1%3C/epo_EVB%3E%3Curl%3E%3C/url%3E&disable_directlink=true&sfx.directlink=off&sfx.report_link=0&rft_id=info:oai/&rft_id=info:pmid/&rfr_iscdi=true |