HIV PROTEASE INHIBITORS, COMPOSITIONS CONTAINING THE SAME, THEIR PHARMACEUTICAL USES AND MATERIALS FOR THEIR SYNTHESIS
Compounds of formula (I) where the formula variables are as defined herein, are disclosed that advantageously inhibit or block the biological activity of the HIV protease. Theses compounds, as well as pharmaceutical compositions containing these compounds, are useful for treating patients or hosts i...
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| creator | CANAN KOCH, STACIE S BURKE, BENJAMIN J KUCERA, DAVID J VIRGIL, SCOTT C BOYER, FREDERICK E JEWELL, TANYA M REICH, SIEGFRIED H BARVIAN, MARK ALEXANDER, THERESE N MURPHY, SEAN T HOLLER, TOD MACHAK, JEFF MITCHELL, LENNERT J BOLTON, GARY TATLOCK, JOHN H WORLAND, STEPHEN T MELNICK, MICHAEL PRASAD JOSYULA, VARA SKALITZKY, DONALD J VARNEY, MICHAEL D |
| description | Compounds of formula (I) where the formula variables are as defined herein, are disclosed that advantageously inhibit or block the biological activity of the HIV protease. Theses compounds, as well as pharmaceutical compositions containing these compounds, are useful for treating patients or hosts infected with the HIV virus. Intermediates and synthetic methods for preparing such compounds are also described. |
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| subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PEPTIDES PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| title | HIV PROTEASE INHIBITORS, COMPOSITIONS CONTAINING THE SAME, THEIR PHARMACEUTICAL USES AND MATERIALS FOR THEIR SYNTHESIS |
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