HETEROARILAMINOSULFONAMIDAS DE 5 MIEMBROS PARA TRATAR AFECCIONES MEDIADAS POR UNA ACTIVIDAD DEFICIENTE DE CFTR

La invenci?n est? relacionada con compuestos de heteroarilo, sales farmac?uticamente aceptables de estos, y preparaciones farmac?uticas de estos. En la presente tambi?n se describen composiciones y el uso de esos compuestos en m?todos de tratamiento de enfermedades y afecciones mediadas por la defic...

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Hauptverfasser: BALTZER, Sylvie, NESTLER, Hans, WIRE, William, MA, Nina, HARTUNG, Ryan, GAO, Zhongli, YEOMAN, Helen, LIAO, Junkai, HURLBUT, Gregory, MECHIN, Ingrid, THURAIRATNAM, Sukanthini, VIVET, Bertrand, FREED, Brian, MUNSON, Mark, SMRCINA, Martin, LEBRETON, Sylvain
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creator BALTZER, Sylvie
NESTLER, Hans
WIRE, William
MA, Nina
HARTUNG, Ryan
GAO, Zhongli
YEOMAN, Helen
LIAO, Junkai
HURLBUT, Gregory
MECHIN, Ingrid
THURAIRATNAM, Sukanthini
VIVET, Bertrand
FREED, Brian
MUNSON, Mark
SMRCINA, Martin
LEBRETON, Sylvain
description La invenci?n est? relacionada con compuestos de heteroarilo, sales farmac?uticamente aceptables de estos, y preparaciones farmac?uticas de estos. En la presente tambi?n se describen composiciones y el uso de esos compuestos en m?todos de tratamiento de enfermedades y afecciones mediadas por la deficiencia de la actividad del CFTR, en particular la fibrosis qu?stica. The invention relates to heteroaryl compounds, pharmaceutically acceptable salts thereof, and pharmaceutical preparations thereof. Also described herein are compositions and the use of such compounds in methods of treating diseases and conditions mediated by deficient CFTR activity, in particular cystic fibrosis.
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subjects CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
title HETEROARILAMINOSULFONAMIDAS DE 5 MIEMBROS PARA TRATAR AFECCIONES MEDIADAS POR UNA ACTIVIDAD DEFICIENTE DE CFTR
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