Terazosinmonohydrochlorid und Verfahren und Zwischenprodukte für seine Herstellung

The present invention provides a non-solvated crystalline polymorph of terazosin monohydrochloride designated Form III and methods for its preparation. Also disclosed is terazosin monohydrochloride methanolate and processes for its production as well as processes for its conversion to other crystall...

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Hauptverfasser: HENRY, RODGER F., WAUKEGAN, ILLINOIS 60085, US, SPANTON, STEPHEN G., GRAYSLAKE, ILLINOIS 60030, US, MORLEY, JAMES A., GURNEE, ILLINOIS 60031, US, BAUER, JOHN F., LAKE BLUFF, ILLINOIS 60044, US, PATEL, RAMESH R., CHICAGO, ILLINOIS 60659, US
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creator HENRY, RODGER F., WAUKEGAN, ILLINOIS 60085, US
SPANTON, STEPHEN G., GRAYSLAKE, ILLINOIS 60030, US
MORLEY, JAMES A., GURNEE, ILLINOIS 60031, US
BAUER, JOHN F., LAKE BLUFF, ILLINOIS 60044, US
PATEL, RAMESH R., CHICAGO, ILLINOIS 60659, US
description The present invention provides a non-solvated crystalline polymorph of terazosin monohydrochloride designated Form III and methods for its preparation. Also disclosed is terazosin monohydrochloride methanolate and processes for its production as well as processes for its conversion to other crystalline forms of terazosin monohydrochloride.
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subjects APPARATUS THEREFOR
CHEMISTRY
GENERAL METHODS OF ORGANIC CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
title Terazosinmonohydrochlorid und Verfahren und Zwischenprodukte für seine Herstellung
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