ΠΑΡΑΓΩΓΑ ΥΠΟΚΑΤΕΣΤΗΜΕΝΩΝ ΟΞΑΖΟΛΙΔΙΝΟΝΩΝ ΚΑΙ Η ΧΡΗΣΗ ΤΟΥΣ ΩΣ ΑΝΑΣΤΟΛΕΙΣ ΠΑΡΑΓΟΝΤΑ ΧΑ
Η εφεύρεση αφορά το πεδίο της πήξης αίματος. Περιγράφονται νέα παράγωγα οξαζολιδινόνης του γενικού τύπου (Ι) μέθοδοι για την παραγωγή τους, καθώς και η χρήση τους ως φαρμακευτικές ουσίες για την πρόληψη και/ή αγωγή παθήσεων. N-oxazolidinylmethyl-substituted (benzo)thiophene carboxamides (I) and thei...
Gespeichert in:
| Hauptverfasser: | , , , , , , |
|---|---|
| Format: | Patent |
| Sprache: | Greek |
| Schlagworte: | |
| Online-Zugang: | Volltext bestellen |
| Tags: |
Tag hinzufügen
Keine Tags, Fügen Sie den ersten Tag hinzu!
|
| container_end_page | |
|---|---|
| container_issue | |
| container_start_page | |
| container_title | |
| container_volume | |
| creator | RÖHRIG Susanne Dr LAMPE Thomas Dr PERNERSTORFER Joseph Dr POHLMANN Jens Dr SCHLEMMER Karl-Heinz Dr STRAUB Alexander Dr PERZBORN Elisabeth Dr |
| description | Η εφεύρεση αφορά το πεδίο της πήξης αίματος. Περιγράφονται νέα παράγωγα οξαζολιδινόνης του γενικού τύπου (Ι) μέθοδοι για την παραγωγή τους, καθώς και η χρήση τους ως φαρμακευτικές ουσίες για την πρόληψη και/ή αγωγή παθήσεων.
N-oxazolidinylmethyl-substituted (benzo)thiophene carboxamides (I) and their salts, hydrates and prodrugs are new. N-oxazolidinylmethyl-substituted (benzo)thiophene carboxamides of formula (I) and their salts, hydrates and prodrugs are new. [Image] R 1> : optionally benzo-fused thiophene, optionally substituted one or more times; R 2> : any selected organic group; R 3>-R 8> : same or different hydrogen or 1-6C alkyl. Excluded are compounds where R 2> = phenyl (optionally substituted once or more) and all of R 3>-R 8> are hydrogen. Independent claims are also included for the following: (1) preparation of (I); and (2) pharmaceutical composition containing (I), optionally also auxiliaries and carriers. ACTIVITY : Anticoagulant; cardiant; anti-anginal; vasotropic; thrombolytic; cerebroprotective; antiarthritic; antiarteriosclerotic; cytostatic; nootropic; neuroprotective. Test details are described but no results given. MECHANISM OF ACTION : Coagulation factor Xa Inhibitor. |
| format | Patent |
| fullrecord | <record><control><sourceid>epo_EVB</sourceid><recordid>TN_cdi_epo_espacenet_CY1115117TT1</recordid><sourceformat>XML</sourceformat><sourcesystem>PC</sourcesystem><sourcerecordid>CY1115117TT1</sourcerecordid><originalsourceid>FETCH-epo_espacenet_CY1115117TT13</originalsourceid><addsrcrecordid>eNqNTksKwjAU7MaFqHeIB3ARRDxAUTxANq5KkbgSLdSLBK2h2vihKcXLzJmcSMGti_feMD9eP6rwhMGLc8KbYwQaUg9cSXkUqLktKiJHgxOU7pQuvDeUOHMccSeGVClgBVqWWqYJPfUGtaCFy9BrvrWhoWCe5O-JUOXDGy3MMOpt012uR90dROPlQsWric4Oic6zdKP3-pjEaynlTMq5UnL6j-cDMOSCZA</addsrcrecordid><sourcetype>Open Access Repository</sourcetype><iscdi>true</iscdi><recordtype>patent</recordtype></control><display><type>patent</type><title>ΠΑΡΑΓΩΓΑ ΥΠΟΚΑΤΕΣΤΗΜΕΝΩΝ ΟΞΑΖΟΛΙΔΙΝΟΝΩΝ ΚΑΙ Η ΧΡΗΣΗ ΤΟΥΣ ΩΣ ΑΝΑΣΤΟΛΕΙΣ ΠΑΡΑΓΟΝΤΑ ΧΑ</title><source>esp@cenet</source><creator>RÖHRIG Susanne Dr ; LAMPE Thomas Dr ; PERNERSTORFER Joseph Dr ; POHLMANN Jens Dr ; SCHLEMMER Karl-Heinz Dr ; STRAUB Alexander Dr ; PERZBORN Elisabeth Dr</creator><creatorcontrib>RÖHRIG Susanne Dr ; LAMPE Thomas Dr ; PERNERSTORFER Joseph Dr ; POHLMANN Jens Dr ; SCHLEMMER Karl-Heinz Dr ; STRAUB Alexander Dr ; PERZBORN Elisabeth Dr</creatorcontrib><description>Η εφεύρεση αφορά το πεδίο της πήξης αίματος. Περιγράφονται νέα παράγωγα οξαζολιδινόνης του γενικού τύπου (Ι) μέθοδοι για την παραγωγή τους, καθώς και η χρήση τους ως φαρμακευτικές ουσίες για την πρόληψη και/ή αγωγή παθήσεων.
N-oxazolidinylmethyl-substituted (benzo)thiophene carboxamides (I) and their salts, hydrates and prodrugs are new. N-oxazolidinylmethyl-substituted (benzo)thiophene carboxamides of formula (I) and their salts, hydrates and prodrugs are new. [Image] R 1> : optionally benzo-fused thiophene, optionally substituted one or more times; R 2> : any selected organic group; R 3>-R 8> : same or different hydrogen or 1-6C alkyl. Excluded are compounds where R 2> = phenyl (optionally substituted once or more) and all of R 3>-R 8> are hydrogen. Independent claims are also included for the following: (1) preparation of (I); and (2) pharmaceutical composition containing (I), optionally also auxiliaries and carriers. ACTIVITY : Anticoagulant; cardiant; anti-anginal; vasotropic; thrombolytic; cerebroprotective; antiarthritic; antiarteriosclerotic; cytostatic; nootropic; neuroprotective. Test details are described but no results given. MECHANISM OF ACTION : Coagulation factor Xa Inhibitor.</description><language>Greek</language><subject>CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>2016</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20161214&DB=EPODOC&CC=CY&NR=1115117T1$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,776,881,25543,76294</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20161214&DB=EPODOC&CC=CY&NR=1115117T1$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>RÖHRIG Susanne Dr</creatorcontrib><creatorcontrib>LAMPE Thomas Dr</creatorcontrib><creatorcontrib>PERNERSTORFER Joseph Dr</creatorcontrib><creatorcontrib>POHLMANN Jens Dr</creatorcontrib><creatorcontrib>SCHLEMMER Karl-Heinz Dr</creatorcontrib><creatorcontrib>STRAUB Alexander Dr</creatorcontrib><creatorcontrib>PERZBORN Elisabeth Dr</creatorcontrib><title>ΠΑΡΑΓΩΓΑ ΥΠΟΚΑΤΕΣΤΗΜΕΝΩΝ ΟΞΑΖΟΛΙΔΙΝΟΝΩΝ ΚΑΙ Η ΧΡΗΣΗ ΤΟΥΣ ΩΣ ΑΝΑΣΤΟΛΕΙΣ ΠΑΡΑΓΟΝΤΑ ΧΑ</title><description>Η εφεύρεση αφορά το πεδίο της πήξης αίματος. Περιγράφονται νέα παράγωγα οξαζολιδινόνης του γενικού τύπου (Ι) μέθοδοι για την παραγωγή τους, καθώς και η χρήση τους ως φαρμακευτικές ουσίες για την πρόληψη και/ή αγωγή παθήσεων.
N-oxazolidinylmethyl-substituted (benzo)thiophene carboxamides (I) and their salts, hydrates and prodrugs are new. N-oxazolidinylmethyl-substituted (benzo)thiophene carboxamides of formula (I) and their salts, hydrates and prodrugs are new. [Image] R 1> : optionally benzo-fused thiophene, optionally substituted one or more times; R 2> : any selected organic group; R 3>-R 8> : same or different hydrogen or 1-6C alkyl. Excluded are compounds where R 2> = phenyl (optionally substituted once or more) and all of R 3>-R 8> are hydrogen. Independent claims are also included for the following: (1) preparation of (I); and (2) pharmaceutical composition containing (I), optionally also auxiliaries and carriers. ACTIVITY : Anticoagulant; cardiant; anti-anginal; vasotropic; thrombolytic; cerebroprotective; antiarthritic; antiarteriosclerotic; cytostatic; nootropic; neuroprotective. Test details are described but no results given. MECHANISM OF ACTION : Coagulation factor Xa Inhibitor.</description><subject>CHEMISTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>HUMAN NECESSITIES</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><subject>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><subject>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2016</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNqNTksKwjAU7MaFqHeIB3ARRDxAUTxANq5KkbgSLdSLBK2h2vihKcXLzJmcSMGti_feMD9eP6rwhMGLc8KbYwQaUg9cSXkUqLktKiJHgxOU7pQuvDeUOHMccSeGVClgBVqWWqYJPfUGtaCFy9BrvrWhoWCe5O-JUOXDGy3MMOpt012uR90dROPlQsWric4Oic6zdKP3-pjEaynlTMq5UnL6j-cDMOSCZA</recordid><startdate>20161214</startdate><enddate>20161214</enddate><creator>RÖHRIG Susanne Dr</creator><creator>LAMPE Thomas Dr</creator><creator>PERNERSTORFER Joseph Dr</creator><creator>POHLMANN Jens Dr</creator><creator>SCHLEMMER Karl-Heinz Dr</creator><creator>STRAUB Alexander Dr</creator><creator>PERZBORN Elisabeth Dr</creator><scope>EVB</scope></search><sort><creationdate>20161214</creationdate><title>ΠΑΡΑΓΩΓΑ ΥΠΟΚΑΤΕΣΤΗΜΕΝΩΝ ΟΞΑΖΟΛΙΔΙΝΟΝΩΝ ΚΑΙ Η ΧΡΗΣΗ ΤΟΥΣ ΩΣ ΑΝΑΣΤΟΛΕΙΣ ΠΑΡΑΓΟΝΤΑ ΧΑ</title><author>RÖHRIG Susanne Dr ; LAMPE Thomas Dr ; PERNERSTORFER Joseph Dr ; POHLMANN Jens Dr ; SCHLEMMER Karl-Heinz Dr ; STRAUB Alexander Dr ; PERZBORN Elisabeth Dr</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_CY1115117TT13</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>Greek</language><creationdate>2016</creationdate><topic>CHEMISTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>HUMAN NECESSITIES</topic><topic>HYGIENE</topic><topic>MEDICAL OR VETERINARY SCIENCE</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><topic>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</topic><topic>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</topic><toplevel>online_resources</toplevel><creatorcontrib>RÖHRIG Susanne Dr</creatorcontrib><creatorcontrib>LAMPE Thomas Dr</creatorcontrib><creatorcontrib>PERNERSTORFER Joseph Dr</creatorcontrib><creatorcontrib>POHLMANN Jens Dr</creatorcontrib><creatorcontrib>SCHLEMMER Karl-Heinz Dr</creatorcontrib><creatorcontrib>STRAUB Alexander Dr</creatorcontrib><creatorcontrib>PERZBORN Elisabeth Dr</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>RÖHRIG Susanne Dr</au><au>LAMPE Thomas Dr</au><au>PERNERSTORFER Joseph Dr</au><au>POHLMANN Jens Dr</au><au>SCHLEMMER Karl-Heinz Dr</au><au>STRAUB Alexander Dr</au><au>PERZBORN Elisabeth Dr</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>ΠΑΡΑΓΩΓΑ ΥΠΟΚΑΤΕΣΤΗΜΕΝΩΝ ΟΞΑΖΟΛΙΔΙΝΟΝΩΝ ΚΑΙ Η ΧΡΗΣΗ ΤΟΥΣ ΩΣ ΑΝΑΣΤΟΛΕΙΣ ΠΑΡΑΓΟΝΤΑ ΧΑ</title><date>2016-12-14</date><risdate>2016</risdate><abstract>Η εφεύρεση αφορά το πεδίο της πήξης αίματος. Περιγράφονται νέα παράγωγα οξαζολιδινόνης του γενικού τύπου (Ι) μέθοδοι για την παραγωγή τους, καθώς και η χρήση τους ως φαρμακευτικές ουσίες για την πρόληψη και/ή αγωγή παθήσεων.
N-oxazolidinylmethyl-substituted (benzo)thiophene carboxamides (I) and their salts, hydrates and prodrugs are new. N-oxazolidinylmethyl-substituted (benzo)thiophene carboxamides of formula (I) and their salts, hydrates and prodrugs are new. [Image] R 1> : optionally benzo-fused thiophene, optionally substituted one or more times; R 2> : any selected organic group; R 3>-R 8> : same or different hydrogen or 1-6C alkyl. Excluded are compounds where R 2> = phenyl (optionally substituted once or more) and all of R 3>-R 8> are hydrogen. Independent claims are also included for the following: (1) preparation of (I); and (2) pharmaceutical composition containing (I), optionally also auxiliaries and carriers. ACTIVITY : Anticoagulant; cardiant; anti-anginal; vasotropic; thrombolytic; cerebroprotective; antiarthritic; antiarteriosclerotic; cytostatic; nootropic; neuroprotective. Test details are described but no results given. MECHANISM OF ACTION : Coagulation factor Xa Inhibitor.</abstract><oa>free_for_read</oa></addata></record> |
| fulltext | fulltext_linktorsrc |
| identifier | |
| ispartof | |
| issn | |
| language | Greek |
| recordid | cdi_epo_espacenet_CY1115117TT1 |
| source | esp@cenet |
| subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| title | ΠΑΡΑΓΩΓΑ ΥΠΟΚΑΤΕΣΤΗΜΕΝΩΝ ΟΞΑΖΟΛΙΔΙΝΟΝΩΝ ΚΑΙ Η ΧΡΗΣΗ ΤΟΥΣ ΩΣ ΑΝΑΣΤΟΛΕΙΣ ΠΑΡΑΓΟΝΤΑ ΧΑ |
| url | https://sfx.bib-bvb.de/sfx_tum?ctx_ver=Z39.88-2004&ctx_enc=info:ofi/enc:UTF-8&ctx_tim=2025-01-22T00%3A49%3A41IST&url_ver=Z39.88-2004&url_ctx_fmt=infofi/fmt:kev:mtx:ctx&rfr_id=info:sid/primo.exlibrisgroup.com:primo3-Article-epo_EVB&rft_val_fmt=info:ofi/fmt:kev:mtx:patent&rft.genre=patent&rft.au=R%C3%96HRIG%20Susanne%20Dr&rft.date=2016-12-14&rft_id=info:doi/&rft_dat=%3Cepo_EVB%3ECY1115117TT1%3C/epo_EVB%3E%3Curl%3E%3C/url%3E&disable_directlink=true&sfx.directlink=off&sfx.report_link=0&rft_id=info:oai/&rft_id=info:pmid/&rfr_iscdi=true |