Azaindoles useful as inhibitors of jak and other protein kinases

The present invention relates to compounds of formula (I), which are inhibitors of protein kinases. The invention also provides pharmaceutical compositions comprising the compounds of the invention and methods of using the compositions in the treatment of various disorders.

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Hauptverfasser: EVERITT SIMON, BOYALL DEAN, BETHIEL RANDY, COME JON, LAUFFER DAVID, SALITURO FRANCESCO, WANG TIANSHEN, ROBINSON DANIEL, HARRINGTON EDMUND, BINCH HAYLEY, FARMER LUC, MORTIMORE MICHAEL, WANG JIAN, ARONOV ALEX, PIERARD FRANCOISE, PIERCE ALBERT, GREEN JEREMY, CHARRIER JEAN-DAMIEN, COURT JOHN, PINDER JOANNE, FRAYSSE DAMIEN
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creator EVERITT SIMON
BOYALL DEAN
BETHIEL RANDY
COME JON
LAUFFER DAVID
SALITURO FRANCESCO
WANG TIANSHEN
ROBINSON DANIEL
HARRINGTON EDMUND
BINCH HAYLEY
FARMER LUC
MORTIMORE MICHAEL
WANG JIAN
ARONOV ALEX
PIERARD FRANCOISE
PIERCE ALBERT
GREEN JEREMY
CHARRIER JEAN-DAMIEN
COURT JOHN
PINDER JOANNE
FRAYSSE DAMIEN
description The present invention relates to compounds of formula (I), which are inhibitors of protein kinases. The invention also provides pharmaceutical compositions comprising the compounds of the invention and methods of using the compositions in the treatment of various disorders.
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language chi ; eng
recordid cdi_epo_espacenet_CN103554104A
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subjects ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAININGELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN,SULFUR, SELENIUM OR TELLURIUM
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
title Azaindoles useful as inhibitors of jak and other protein kinases
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