Compuestos derivados de amida; composición farmacéutica que comprende a dicho compuesto; combinación farmacéutica; y uso del compuesto en el tratamiento del vih
COMPUESTO DE LA FORMULA LAS SALES Y FORMAS ESTEREOISOMÉRICAS DEL MISMO, DONDE R, RL, R2, R3, R4, R5 YX SON COMO SE DEFINEN EN LA MEMORIA DESCRIPTIVA; USO DE DICHO COMPUESTO QUE SIRVE PARA PREPARAR UN MEDICAMENTO ÚTIL PARA REFORZAR ANTIVIRALES DE VIH; COMBINACIÓN FARMACÉUTICA QUE COMPRENDE DICHO COMP...
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| creator | HACHE, GEERWIN YVONNE PAUL JONCKERS, TIM HUGO MARIA SCHEPENS, WIM BERT GRIET HALLENBERGER, BEATE SABINE SASAKI, JENNIFER CHIYOMI BAUMEISTER, JUDITH EVA VAN T. KLOOSTER, GERBEN ALBERT E |
| description | COMPUESTO DE LA FORMULA
LAS SALES Y FORMAS ESTEREOISOMÉRICAS DEL MISMO, DONDE R, RL, R2, R3, R4, R5 YX SON COMO SE DEFINEN EN LA
MEMORIA DESCRIPTIVA;
USO DE DICHO COMPUESTO QUE SIRVE PARA PREPARAR UN MEDICAMENTO ÚTIL PARA REFORZAR ANTIVIRALES DE VIH;
COMBINACIÓN FARMACÉUTICA QUE COMPRENDE DICHO COMPUESTO; Y
USO DE DICHA COMBINACIÓN QUE SIRVE PARA PREPARAR UN MEDICAMENTO.
The present invention relates to compounds that have CYP450 inhibiting properties and are therefore useful as boosters of certain drugs, i.e. they are able to increase at least one of the pharmacokinetic variables of certain drugs when co-administered. The invention further provides the use of said compounds as improvers of the bioavailability of certain drugs. Methods for the preparation of the compounds of the invention and pharmaceutical compositions are also provided. |
| format | Patent |
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LAS SALES Y FORMAS ESTEREOISOMÉRICAS DEL MISMO, DONDE R, RL, R2, R3, R4, R5 YX SON COMO SE DEFINEN EN LA
MEMORIA DESCRIPTIVA;
USO DE DICHO COMPUESTO QUE SIRVE PARA PREPARAR UN MEDICAMENTO ÚTIL PARA REFORZAR ANTIVIRALES DE VIH;
COMBINACIÓN FARMACÉUTICA QUE COMPRENDE DICHO COMPUESTO; Y
USO DE DICHA COMBINACIÓN QUE SIRVE PARA PREPARAR UN MEDICAMENTO.
The present invention relates to compounds that have CYP450 inhibiting properties and are therefore useful as boosters of certain drugs, i.e. they are able to increase at least one of the pharmacokinetic variables of certain drugs when co-administered. The invention further provides the use of said compounds as improvers of the bioavailability of certain drugs. Methods for the preparation of the compounds of the invention and pharmaceutical compositions are also provided.</description><language>spa</language><subject>CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>2010</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20100115&DB=EPODOC&CC=CL&NR=2008003639A1$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,776,881,25543,76293</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20100115&DB=EPODOC&CC=CL&NR=2008003639A1$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>HACHE, GEERWIN YVONNE PAUL; JONCKERS, TIM HUGO MARIA; SCHEPENS, WIM BERT GRIET; HALLENBERGER, BEATE SABINE; SASAKI, JENNIFER CHIYOMI; BAUMEISTER, JUDITH EVA; VAN T. KLOOSTER, GERBEN ALBERT E</creatorcontrib><title>Compuestos derivados de amida; composición farmacéutica que comprende a dicho compuesto; combinación farmacéutica; y uso del compuesto en el tratamiento del vih</title><description>COMPUESTO DE LA FORMULA
LAS SALES Y FORMAS ESTEREOISOMÉRICAS DEL MISMO, DONDE R, RL, R2, R3, R4, R5 YX SON COMO SE DEFINEN EN LA
MEMORIA DESCRIPTIVA;
USO DE DICHO COMPUESTO QUE SIRVE PARA PREPARAR UN MEDICAMENTO ÚTIL PARA REFORZAR ANTIVIRALES DE VIH;
COMBINACIÓN FARMACÉUTICA QUE COMPRENDE DICHO COMPUESTO; Y
USO DE DICHA COMBINACIÓN QUE SIRVE PARA PREPARAR UN MEDICAMENTO.
The present invention relates to compounds that have CYP450 inhibiting properties and are therefore useful as boosters of certain drugs, i.e. they are able to increase at least one of the pharmacokinetic variables of certain drugs when co-administered. The invention further provides the use of said compounds as improvers of the bioavailability of certain drugs. Methods for the preparation of the compounds of the invention and pharmaceutical compositions are also provided.</description><subject>CHEMISTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>HUMAN NECESSITIES</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><subject>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><subject>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2010</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNqNjTsKwkAQhtNYiHqHAWthNSBKKgmKhaV9GDcjGUh24z4C3sfG2iPkYq6rYGNhNY_vfwyTW66b1pN12kJJhjss4wbYcIkZyIC1Zcn9Q8EZTYOyv3vHEuHiKWJD6qWHkmWl4yfmRe-JFf7wZnAFb3Xoqb8GIAXhdgZdKCfl3rzjapwMzlhbmnzmKJnutsd8P6NWF2RblKTIFflhIcRKiHSZrjfz9D_VEyxSWlo</recordid><startdate>20100115</startdate><enddate>20100115</enddate><creator>HACHE, GEERWIN YVONNE PAUL; JONCKERS, TIM HUGO MARIA; SCHEPENS, WIM BERT GRIET; HALLENBERGER, BEATE SABINE; SASAKI, JENNIFER CHIYOMI; BAUMEISTER, JUDITH EVA; VAN T. KLOOSTER, GERBEN ALBERT E</creator><scope>EVB</scope></search><sort><creationdate>20100115</creationdate><title>Compuestos derivados de amida; composición farmacéutica que comprende a dicho compuesto; combinación farmacéutica; y uso del compuesto en el tratamiento del vih</title><author>HACHE, GEERWIN YVONNE PAUL; JONCKERS, TIM HUGO MARIA; SCHEPENS, WIM BERT GRIET; HALLENBERGER, BEATE SABINE; SASAKI, JENNIFER CHIYOMI; BAUMEISTER, JUDITH EVA; VAN T. KLOOSTER, GERBEN ALBERT E</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_CL2008003639A13</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>spa</language><creationdate>2010</creationdate><topic>CHEMISTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>HUMAN NECESSITIES</topic><topic>HYGIENE</topic><topic>MEDICAL OR VETERINARY SCIENCE</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><topic>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</topic><topic>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</topic><toplevel>online_resources</toplevel><creatorcontrib>HACHE, GEERWIN YVONNE PAUL; JONCKERS, TIM HUGO MARIA; SCHEPENS, WIM BERT GRIET; HALLENBERGER, BEATE SABINE; SASAKI, JENNIFER CHIYOMI; BAUMEISTER, JUDITH EVA; VAN T. KLOOSTER, GERBEN ALBERT E</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>HACHE, GEERWIN YVONNE PAUL; JONCKERS, TIM HUGO MARIA; SCHEPENS, WIM BERT GRIET; HALLENBERGER, BEATE SABINE; SASAKI, JENNIFER CHIYOMI; BAUMEISTER, JUDITH EVA; VAN T. KLOOSTER, GERBEN ALBERT E</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>Compuestos derivados de amida; composición farmacéutica que comprende a dicho compuesto; combinación farmacéutica; y uso del compuesto en el tratamiento del vih</title><date>2010-01-15</date><risdate>2010</risdate><abstract>COMPUESTO DE LA FORMULA
LAS SALES Y FORMAS ESTEREOISOMÉRICAS DEL MISMO, DONDE R, RL, R2, R3, R4, R5 YX SON COMO SE DEFINEN EN LA
MEMORIA DESCRIPTIVA;
USO DE DICHO COMPUESTO QUE SIRVE PARA PREPARAR UN MEDICAMENTO ÚTIL PARA REFORZAR ANTIVIRALES DE VIH;
COMBINACIÓN FARMACÉUTICA QUE COMPRENDE DICHO COMPUESTO; Y
USO DE DICHA COMBINACIÓN QUE SIRVE PARA PREPARAR UN MEDICAMENTO.
The present invention relates to compounds that have CYP450 inhibiting properties and are therefore useful as boosters of certain drugs, i.e. they are able to increase at least one of the pharmacokinetic variables of certain drugs when co-administered. The invention further provides the use of said compounds as improvers of the bioavailability of certain drugs. Methods for the preparation of the compounds of the invention and pharmaceutical compositions are also provided.</abstract><oa>free_for_read</oa></addata></record> |
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| subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| title | Compuestos derivados de amida; composición farmacéutica que comprende a dicho compuesto; combinación farmacéutica; y uso del compuesto en el tratamiento del vih |
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