PROCESS FOR MAKING PIPERIDINONE CARBOXAMIDE INDANE AND AZAINANE CGRP RECEPTOR ANTAGONISTS
The invention encompasses a novel process for making piperidinone carboxamide indane and azainane derivatives, which are CGRP receptor antagonists useful for the treatment of migraine, utilizing a highly effective spiroacid synthesis (see formula I) La présente invention porte sur un nouveau procédé...
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| creator | CLEATOR, EDWARD KUO, SHENUN YASUDA, NOBUYOSHI YIN, JIANGUO XIANG, BANGPING MALIGRES, PETER EMMANUEL BELYK, KEVIN M |
| description | The invention encompasses a novel process for making piperidinone carboxamide indane and azainane derivatives, which are CGRP receptor antagonists useful for the treatment of migraine, utilizing a highly effective spiroacid synthesis (see formula I)
La présente invention porte sur un nouveau procédé de production de dérivés pipéridinone carboxamide indane et azainane, qui sont des antagonistes du récepteur CGRP utiles dans le traitement de la migraine, ledit procédé faisant appel à une synthèse hautement efficace de spiroacides. |
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La présente invention porte sur un nouveau procédé de production de dérivés pipéridinone carboxamide indane et azainane, qui sont des antagonistes du récepteur CGRP utiles dans le traitement de la migraine, ledit procédé faisant appel à une synthèse hautement efficace de spiroacides.</description><subject>ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAININGELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN,SULFUR, SELENIUM OR TELLURIUM</subject><subject>CHEMISTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2020</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNqFjDEKwkAQRdNYiHoG5wI2GsWU4-xkHSSzy-4WahOCrJVoIN4fI9hbfd7j8afFxQdHHCPULkCDJ1ELXjwHMaJOGQjDwZ2xEcMganBUqAbwiqJfIBs8BCb2aXxATWidSkxxXkzu3WPIi9_OimXNiY6r3L_aPPTdLT_zuyVc73fbqixp87_4AGFxMLg</recordid><startdate>20201208</startdate><enddate>20201208</enddate><creator>CLEATOR, EDWARD</creator><creator>KUO, SHENUN</creator><creator>YASUDA, NOBUYOSHI</creator><creator>YIN, JIANGUO</creator><creator>XIANG, BANGPING</creator><creator>MALIGRES, PETER EMMANUEL</creator><creator>BELYK, KEVIN M</creator><scope>EVB</scope></search><sort><creationdate>20201208</creationdate><title>PROCESS FOR MAKING PIPERIDINONE CARBOXAMIDE INDANE AND AZAINANE CGRP RECEPTOR ANTAGONISTS</title><author>CLEATOR, EDWARD ; KUO, SHENUN ; YASUDA, NOBUYOSHI ; YIN, JIANGUO ; XIANG, BANGPING ; MALIGRES, PETER EMMANUEL ; BELYK, KEVIN M</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_CA2865944C3</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>eng ; fre</language><creationdate>2020</creationdate><topic>ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAININGELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN,SULFUR, SELENIUM OR TELLURIUM</topic><topic>CHEMISTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><toplevel>online_resources</toplevel><creatorcontrib>CLEATOR, EDWARD</creatorcontrib><creatorcontrib>KUO, SHENUN</creatorcontrib><creatorcontrib>YASUDA, NOBUYOSHI</creatorcontrib><creatorcontrib>YIN, JIANGUO</creatorcontrib><creatorcontrib>XIANG, BANGPING</creatorcontrib><creatorcontrib>MALIGRES, PETER EMMANUEL</creatorcontrib><creatorcontrib>BELYK, KEVIN M</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>CLEATOR, EDWARD</au><au>KUO, SHENUN</au><au>YASUDA, NOBUYOSHI</au><au>YIN, JIANGUO</au><au>XIANG, BANGPING</au><au>MALIGRES, PETER EMMANUEL</au><au>BELYK, KEVIN M</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>PROCESS FOR MAKING PIPERIDINONE CARBOXAMIDE INDANE AND AZAINANE CGRP RECEPTOR ANTAGONISTS</title><date>2020-12-08</date><risdate>2020</risdate><abstract>The invention encompasses a novel process for making piperidinone carboxamide indane and azainane derivatives, which are CGRP receptor antagonists useful for the treatment of migraine, utilizing a highly effective spiroacid synthesis (see formula I)
La présente invention porte sur un nouveau procédé de production de dérivés pipéridinone carboxamide indane et azainane, qui sont des antagonistes du récepteur CGRP utiles dans le traitement de la migraine, ledit procédé faisant appel à une synthèse hautement efficace de spiroacides.</abstract><oa>free_for_read</oa></addata></record> |
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| subjects | ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAININGELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN,SULFUR, SELENIUM OR TELLURIUM CHEMISTRY HETEROCYCLIC COMPOUNDS METALLURGY ORGANIC CHEMISTRY |
| title | PROCESS FOR MAKING PIPERIDINONE CARBOXAMIDE INDANE AND AZAINANE CGRP RECEPTOR ANTAGONISTS |
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