NOVEL HETEROCYCLES

Described are novel heterocyclic compounds of the general formula (1), their derivatives, analogs, tautomeric forms, stereoisomers, polymorphs, hydrates, solvates, pharmaceutically acceptable salts, pharmaceutical compositions, metabolites and prodrugs thereof. These compounds are useful in the trea...

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Hauptverfasser: NARAYANAN, SUKUNATH, JANARTHANAM, VENKATESAN, SRINIVAS, VISWESWARA AKELLA SATYA SURYA, SURENDRAN, NARAYANAN, TADIPARTHI, RAVIKUMAR, BHAKIARAJ, DURAIRAJ PETER, NARASIMHAN, KILAMBI, BALASUBRAMANIAN, GOPALAN, GADDE, SATHYANARAYANA, NARAYANAM, MARUTHIKUMAR, VISHWAKARMA, LOLAKNATH SANTOSH, PARAMESWARAN, VENKATESAN, SAPPANIMUTHU, THIRUNAVUKKARASU, SHARMA, GANAPAVARAPU VEERA RAGHAVA, RAMACHANDRAN, UMA, NARAYANAN, SHRIDHAR, THARA, SATHYA NARAYANA, RAJAGOPAL, SRIRAM, SAXENA, SANJEEV, REDDY, GADDAM OM, KACHHADIA, VIRENDRA
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creator NARAYANAN, SUKUNATH
JANARTHANAM, VENKATESAN
SRINIVAS, VISWESWARA AKELLA SATYA SURYA
SURENDRAN, NARAYANAN
TADIPARTHI, RAVIKUMAR
BHAKIARAJ, DURAIRAJ PETER
NARASIMHAN, KILAMBI
BALASUBRAMANIAN, GOPALAN
GADDE, SATHYANARAYANA
NARAYANAM, MARUTHIKUMAR
VISHWAKARMA, LOLAKNATH SANTOSH
PARAMESWARAN, VENKATESAN
SAPPANIMUTHU, THIRUNAVUKKARASU
SHARMA, GANAPAVARAPU VEERA RAGHAVA
RAMACHANDRAN, UMA
NARAYANAN, SHRIDHAR
THARA, SATHYA NARAYANA
RAJAGOPAL, SRIRAM
SAXENA, SANJEEV
REDDY, GADDAM OM
KACHHADIA, VIRENDRA
description Described are novel heterocyclic compounds of the general formula (1), their derivatives, analogs, tautomeric forms, stereoisomers, polymorphs, hydrates, solvates, pharmaceutically acceptable salts, pharmaceutical compositions, metabolites and prodrugs thereof. These compounds are useful in the treatment of immunological diseases, inflammation, pain disorder, rheumatoid arthritis; osteoporosis; multiple myeloma; uveititis; acute and chronic myelogenous leukemia; atherosclerosis; cancer; cachexia; ischemic-induced cell damage; pancreatic beta cell destruction; osteoarthritis; rheumatoid spondylitis; gouty arthritis; inflammatory bowel disease; ARDS; psoriasis; Crohn's disease; allergic rhinitis; ulcerative colitis; anaphylaxis; contact dermatitis; muscle degeneration; asthma; COPD; bone resorption diseases; multiple sclerosis; sepsis; septic shock; toxic shock syndrome and fever. More particularly these compounds are useful as PDE4 inhibitors and are useful for treating PDE4 mediated diseases.
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subjects CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
title NOVEL HETEROCYCLES
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