NOVEL HETEROCYCLES
Described are novel heterocyclic compounds of the general formula (1), their derivatives, analogs, tautomeric forms, stereoisomers, polymorphs, hydrates, solvates, pharmaceutically acceptable salts, pharmaceutical compositions, metabolites and prodrugs thereof. These compounds are useful in the trea...
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creator | NARAYANAN, SUKUNATH JANARTHANAM, VENKATESAN SRINIVAS, VISWESWARA AKELLA SATYA SURYA SURENDRAN, NARAYANAN TADIPARTHI, RAVIKUMAR BHAKIARAJ, DURAIRAJ PETER NARASIMHAN, KILAMBI BALASUBRAMANIAN, GOPALAN GADDE, SATHYANARAYANA NARAYANAM, MARUTHIKUMAR VISHWAKARMA, LOLAKNATH SANTOSH PARAMESWARAN, VENKATESAN SAPPANIMUTHU, THIRUNAVUKKARASU SHARMA, GANAPAVARAPU VEERA RAGHAVA RAMACHANDRAN, UMA NARAYANAN, SHRIDHAR THARA, SATHYA NARAYANA RAJAGOPAL, SRIRAM SAXENA, SANJEEV REDDY, GADDAM OM KACHHADIA, VIRENDRA |
description | Described are novel heterocyclic compounds of the general formula (1), their derivatives, analogs, tautomeric forms, stereoisomers, polymorphs, hydrates, solvates, pharmaceutically acceptable salts, pharmaceutical compositions, metabolites and prodrugs thereof. These compounds are useful in the treatment of immunological diseases, inflammation, pain disorder, rheumatoid arthritis; osteoporosis; multiple myeloma; uveititis; acute and chronic myelogenous leukemia; atherosclerosis; cancer; cachexia; ischemic-induced cell damage; pancreatic beta cell destruction; osteoarthritis; rheumatoid spondylitis; gouty arthritis; inflammatory bowel disease; ARDS; psoriasis; Crohn's disease; allergic rhinitis; ulcerative colitis; anaphylaxis; contact dermatitis; muscle degeneration; asthma; COPD; bone resorption diseases; multiple sclerosis; sepsis; septic shock; toxic shock syndrome and fever. More particularly these compounds are useful as PDE4 inhibitors and are useful for treating PDE4 mediated diseases. |
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These compounds are useful in the treatment of immunological diseases, inflammation, pain disorder, rheumatoid arthritis; osteoporosis; multiple myeloma; uveititis; acute and chronic myelogenous leukemia; atherosclerosis; cancer; cachexia; ischemic-induced cell damage; pancreatic beta cell destruction; osteoarthritis; rheumatoid spondylitis; gouty arthritis; inflammatory bowel disease; ARDS; psoriasis; Crohn's disease; allergic rhinitis; ulcerative colitis; anaphylaxis; contact dermatitis; muscle degeneration; asthma; COPD; bone resorption diseases; multiple sclerosis; sepsis; septic shock; toxic shock syndrome and fever. More particularly these compounds are useful as PDE4 inhibitors and are useful for treating PDE4 mediated diseases.</description><language>eng ; fre</language><subject>CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><creationdate>2016</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20160607&DB=EPODOC&CC=CA&NR=2715069C$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,776,881,25542,76289</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20160607&DB=EPODOC&CC=CA&NR=2715069C$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>NARAYANAN, SUKUNATH</creatorcontrib><creatorcontrib>JANARTHANAM, VENKATESAN</creatorcontrib><creatorcontrib>SRINIVAS, VISWESWARA AKELLA SATYA SURYA</creatorcontrib><creatorcontrib>SURENDRAN, NARAYANAN</creatorcontrib><creatorcontrib>TADIPARTHI, RAVIKUMAR</creatorcontrib><creatorcontrib>BHAKIARAJ, DURAIRAJ PETER</creatorcontrib><creatorcontrib>NARASIMHAN, KILAMBI</creatorcontrib><creatorcontrib>BALASUBRAMANIAN, GOPALAN</creatorcontrib><creatorcontrib>GADDE, SATHYANARAYANA</creatorcontrib><creatorcontrib>NARAYANAM, MARUTHIKUMAR</creatorcontrib><creatorcontrib>VISHWAKARMA, LOLAKNATH SANTOSH</creatorcontrib><creatorcontrib>PARAMESWARAN, VENKATESAN</creatorcontrib><creatorcontrib>SAPPANIMUTHU, THIRUNAVUKKARASU</creatorcontrib><creatorcontrib>SHARMA, GANAPAVARAPU VEERA RAGHAVA</creatorcontrib><creatorcontrib>RAMACHANDRAN, UMA</creatorcontrib><creatorcontrib>NARAYANAN, SHRIDHAR</creatorcontrib><creatorcontrib>THARA, SATHYA NARAYANA</creatorcontrib><creatorcontrib>RAJAGOPAL, SRIRAM</creatorcontrib><creatorcontrib>SAXENA, SANJEEV</creatorcontrib><creatorcontrib>REDDY, GADDAM OM</creatorcontrib><creatorcontrib>KACHHADIA, VIRENDRA</creatorcontrib><title>NOVEL HETEROCYCLES</title><description>Described are novel heterocyclic compounds of the general formula (1), their derivatives, analogs, tautomeric forms, stereoisomers, polymorphs, hydrates, solvates, pharmaceutically acceptable salts, pharmaceutical compositions, metabolites and prodrugs thereof. These compounds are useful in the treatment of immunological diseases, inflammation, pain disorder, rheumatoid arthritis; osteoporosis; multiple myeloma; uveititis; acute and chronic myelogenous leukemia; atherosclerosis; cancer; cachexia; ischemic-induced cell damage; pancreatic beta cell destruction; osteoarthritis; rheumatoid spondylitis; gouty arthritis; inflammatory bowel disease; ARDS; psoriasis; Crohn's disease; allergic rhinitis; ulcerative colitis; anaphylaxis; contact dermatitis; muscle degeneration; asthma; COPD; bone resorption diseases; multiple sclerosis; sepsis; septic shock; toxic shock syndrome and fever. More particularly these compounds are useful as PDE4 inhibitors and are useful for treating PDE4 mediated diseases.</description><subject>CHEMISTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>HUMAN NECESSITIES</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><subject>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2016</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNrjZBDy8w9z9VHwcA1xDfJ3jnT2cQ3mYWBNS8wpTuWF0twM8m6uIc4euqkF-fGpxQWJyal5qSXxzo5G5oamBmaWzsaEVQAA1CodSQ</recordid><startdate>20160607</startdate><enddate>20160607</enddate><creator>NARAYANAN, SUKUNATH</creator><creator>JANARTHANAM, VENKATESAN</creator><creator>SRINIVAS, VISWESWARA AKELLA SATYA SURYA</creator><creator>SURENDRAN, NARAYANAN</creator><creator>TADIPARTHI, RAVIKUMAR</creator><creator>BHAKIARAJ, DURAIRAJ PETER</creator><creator>NARASIMHAN, KILAMBI</creator><creator>BALASUBRAMANIAN, GOPALAN</creator><creator>GADDE, SATHYANARAYANA</creator><creator>NARAYANAM, MARUTHIKUMAR</creator><creator>VISHWAKARMA, LOLAKNATH SANTOSH</creator><creator>PARAMESWARAN, VENKATESAN</creator><creator>SAPPANIMUTHU, THIRUNAVUKKARASU</creator><creator>SHARMA, GANAPAVARAPU VEERA RAGHAVA</creator><creator>RAMACHANDRAN, UMA</creator><creator>NARAYANAN, SHRIDHAR</creator><creator>THARA, SATHYA NARAYANA</creator><creator>RAJAGOPAL, SRIRAM</creator><creator>SAXENA, SANJEEV</creator><creator>REDDY, GADDAM OM</creator><creator>KACHHADIA, VIRENDRA</creator><scope>EVB</scope></search><sort><creationdate>20160607</creationdate><title>NOVEL HETEROCYCLES</title><author>NARAYANAN, SUKUNATH ; JANARTHANAM, VENKATESAN ; SRINIVAS, VISWESWARA AKELLA SATYA SURYA ; SURENDRAN, NARAYANAN ; TADIPARTHI, RAVIKUMAR ; BHAKIARAJ, DURAIRAJ PETER ; NARASIMHAN, KILAMBI ; BALASUBRAMANIAN, GOPALAN ; GADDE, SATHYANARAYANA ; NARAYANAM, MARUTHIKUMAR ; VISHWAKARMA, LOLAKNATH SANTOSH ; PARAMESWARAN, VENKATESAN ; SAPPANIMUTHU, THIRUNAVUKKARASU ; SHARMA, GANAPAVARAPU VEERA RAGHAVA ; RAMACHANDRAN, UMA ; NARAYANAN, SHRIDHAR ; THARA, SATHYA NARAYANA ; RAJAGOPAL, SRIRAM ; SAXENA, SANJEEV ; REDDY, GADDAM OM ; KACHHADIA, VIRENDRA</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_CA2715069C3</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>eng ; fre</language><creationdate>2016</creationdate><topic>CHEMISTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>HUMAN NECESSITIES</topic><topic>HYGIENE</topic><topic>MEDICAL OR VETERINARY SCIENCE</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><topic>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</topic><toplevel>online_resources</toplevel><creatorcontrib>NARAYANAN, SUKUNATH</creatorcontrib><creatorcontrib>JANARTHANAM, VENKATESAN</creatorcontrib><creatorcontrib>SRINIVAS, VISWESWARA AKELLA SATYA SURYA</creatorcontrib><creatorcontrib>SURENDRAN, NARAYANAN</creatorcontrib><creatorcontrib>TADIPARTHI, RAVIKUMAR</creatorcontrib><creatorcontrib>BHAKIARAJ, DURAIRAJ PETER</creatorcontrib><creatorcontrib>NARASIMHAN, KILAMBI</creatorcontrib><creatorcontrib>BALASUBRAMANIAN, GOPALAN</creatorcontrib><creatorcontrib>GADDE, SATHYANARAYANA</creatorcontrib><creatorcontrib>NARAYANAM, MARUTHIKUMAR</creatorcontrib><creatorcontrib>VISHWAKARMA, LOLAKNATH SANTOSH</creatorcontrib><creatorcontrib>PARAMESWARAN, VENKATESAN</creatorcontrib><creatorcontrib>SAPPANIMUTHU, THIRUNAVUKKARASU</creatorcontrib><creatorcontrib>SHARMA, GANAPAVARAPU VEERA RAGHAVA</creatorcontrib><creatorcontrib>RAMACHANDRAN, UMA</creatorcontrib><creatorcontrib>NARAYANAN, SHRIDHAR</creatorcontrib><creatorcontrib>THARA, SATHYA NARAYANA</creatorcontrib><creatorcontrib>RAJAGOPAL, SRIRAM</creatorcontrib><creatorcontrib>SAXENA, SANJEEV</creatorcontrib><creatorcontrib>REDDY, GADDAM OM</creatorcontrib><creatorcontrib>KACHHADIA, VIRENDRA</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>NARAYANAN, SUKUNATH</au><au>JANARTHANAM, VENKATESAN</au><au>SRINIVAS, VISWESWARA AKELLA SATYA SURYA</au><au>SURENDRAN, NARAYANAN</au><au>TADIPARTHI, RAVIKUMAR</au><au>BHAKIARAJ, DURAIRAJ PETER</au><au>NARASIMHAN, KILAMBI</au><au>BALASUBRAMANIAN, GOPALAN</au><au>GADDE, SATHYANARAYANA</au><au>NARAYANAM, MARUTHIKUMAR</au><au>VISHWAKARMA, LOLAKNATH SANTOSH</au><au>PARAMESWARAN, VENKATESAN</au><au>SAPPANIMUTHU, THIRUNAVUKKARASU</au><au>SHARMA, GANAPAVARAPU VEERA RAGHAVA</au><au>RAMACHANDRAN, UMA</au><au>NARAYANAN, SHRIDHAR</au><au>THARA, SATHYA NARAYANA</au><au>RAJAGOPAL, SRIRAM</au><au>SAXENA, SANJEEV</au><au>REDDY, GADDAM OM</au><au>KACHHADIA, VIRENDRA</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>NOVEL HETEROCYCLES</title><date>2016-06-07</date><risdate>2016</risdate><abstract>Described are novel heterocyclic compounds of the general formula (1), their derivatives, analogs, tautomeric forms, stereoisomers, polymorphs, hydrates, solvates, pharmaceutically acceptable salts, pharmaceutical compositions, metabolites and prodrugs thereof. These compounds are useful in the treatment of immunological diseases, inflammation, pain disorder, rheumatoid arthritis; osteoporosis; multiple myeloma; uveititis; acute and chronic myelogenous leukemia; atherosclerosis; cancer; cachexia; ischemic-induced cell damage; pancreatic beta cell destruction; osteoarthritis; rheumatoid spondylitis; gouty arthritis; inflammatory bowel disease; ARDS; psoriasis; Crohn's disease; allergic rhinitis; ulcerative colitis; anaphylaxis; contact dermatitis; muscle degeneration; asthma; COPD; bone resorption diseases; multiple sclerosis; sepsis; septic shock; toxic shock syndrome and fever. More particularly these compounds are useful as PDE4 inhibitors and are useful for treating PDE4 mediated diseases.</abstract><oa>free_for_read</oa></addata></record> |
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subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES |
title | NOVEL HETEROCYCLES |
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