PHENYL-PYRAZOLE DERIVATIVES AS NON-STEROIDAL GLUCOCORICOID RECEPTOR LIGANDS

The present invention provides compounds of formula (I): a process for their preparation, to pharmaceutical compositions comprising the compounds and the preparation of said compositions, to intermediates and to use of the compounds for the manufacture of a medicament for therapeutic treatment, part...

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Hauptverfasser: COOPER, ANTHONY WILLIAM JAMES, WOOLVEN, JAMES MICHAEL, BARNETT, HEATHER ANNE, INGLIS, GRAHAM GEORGE ADAM, MCLAY, IAIN MCFARLANE, KEELING, STEVEN PHILIP, MACDONALD, SIMON JOHN FAWCETT, CAMPBELL, IAN BAXTER, COE, DIANE MARY, JONES, HAYDN TERENCE, SKONE, PHILIP ALAN, WEINGARTEN, GORDON GAD
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creator COOPER, ANTHONY WILLIAM JAMES
WOOLVEN, JAMES MICHAEL
BARNETT, HEATHER ANNE
INGLIS, GRAHAM GEORGE ADAM
MCLAY, IAIN MCFARLANE
KEELING, STEVEN PHILIP
MACDONALD, SIMON JOHN FAWCETT
CAMPBELL, IAN BAXTER
COE, DIANE MARY
JONES, HAYDN TERENCE
SKONE, PHILIP ALAN
WEINGARTEN, GORDON GAD
description The present invention provides compounds of formula (I): a process for their preparation, to pharmaceutical compositions comprising the compounds and the preparation of said compositions, to intermediates and to use of the compounds for the manufacture of a medicament for therapeutic treatment, particularly for the treatment of inflammation, allergy and/or auto-immune conditions. La présente invention concerne des composés de formule (I), un procédé pour leur préparation, des compositions pharmaceutiques comprenant les composés et la préparation desdites compositions, des intermédiaires et l'utilisation des composés pour la fabrication d'un médicament pour un traitement thérapeutique, en particulier pour le traitement de l'inflammation, de l'allergie et/ou de pathologies auto-immunes.
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subjects CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
title PHENYL-PYRAZOLE DERIVATIVES AS NON-STEROIDAL GLUCOCORICOID RECEPTOR LIGANDS
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