THIAZOLOPYRIDINONE DERIVATES AS MCH RECEPTOR ANTAGONISTS

The present invention relates to a melanin concentrating hormone antagonist compound of formula (I); wherein w, R1, q, p, R2, t, Ar1, L1, R3 and R4 are as defined, or a pharmaceutically acceptable salt, solvate, or enantiomer thereof useful in the treatment, prevention or amelioration of symptoms as...

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Hauptverfasser: GARDINIER, KEVIN MATTHEW, SAVIN, KENNETH ALLEN, AMEGADZIE, ALBERT KUDZOVI, HEMBRE, ERIK JAMES, WAKEFIELD, BRIAN DAVID, BECK, JAMES PETER, RUBLE, JAMES CRAIG
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creator GARDINIER, KEVIN MATTHEW
SAVIN, KENNETH ALLEN
AMEGADZIE, ALBERT KUDZOVI
HEMBRE, ERIK JAMES
WAKEFIELD, BRIAN DAVID
BECK, JAMES PETER
RUBLE, JAMES CRAIG
description The present invention relates to a melanin concentrating hormone antagonist compound of formula (I); wherein w, R1, q, p, R2, t, Ar1, L1, R3 and R4 are as defined, or a pharmaceutically acceptable salt, solvate, or enantiomer thereof useful in the treatment, prevention or amelioration of symptoms associated with obesity and related diseases.
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wherein w, R1, q, p, R2, t, Ar1, L1, R3 and R4 are as defined, or a pharmaceutically acceptable salt, solvate, or enantiomer thereof useful in the treatment, prevention or amelioration of symptoms associated with obesity and related diseases.</abstract><oa>free_for_read</oa></addata></record>
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subjects CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
title THIAZOLOPYRIDINONE DERIVATES AS MCH RECEPTOR ANTAGONISTS
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