AROMATIC DERIVATIVES AS HIV ASPARTYL PROTEASE INHIBITORS

AROMATIC DERIVATIVES AS HIV ASPARTYL PROTEASE INHIBITORS

The present invention provides HIV aspartyl protease inhibitors of the formula; (see formula I) and when the compound of formula I comprises an amino group, pharmaceutically acceptable ammonium salts thereof, wherein n is 3 or 4, wherein R1 may be, for example, iso-butyl, wherein X and Y, same or di...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Hauptverfasser: LAVALLEE, JEAN-FRANCOIS, PERRON, VALERIE, LEBERRE, NICOLAS, STRANIX, BRENT RICHARD
Format: Patent
Sprache:eng ; fre
Schlagworte:
ACYCLIC OR CARBOCYCLIC COMPOUNDS
CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
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Beschreibung
Zusammenfassung:The present invention provides HIV aspartyl protease inhibitors of the formula; (see formula I) and when the compound of formula I comprises an amino group, pharmaceutically acceptable ammonium salts thereof, wherein n is 3 or 4, wherein R1 may be, for example, iso-butyl, wherein X and Y, same or different, may be, for example, NH2 and F, and wherein R2 and R3 are as defined herein.