Acridin derivatives
Aminomethyl-acridine derivatives (I) are new. Aryl substituted aminomethyl-acridine derivatives of formula (I) and their salts are new. X = N and Y = C; or X = C and Y = N; R1 = A; R2 = H or OR12; R3 = H; or R2 and R3 together form a double bond; R4 = CH2NR14R15; R5 and R6 = H or 1-6C alkyl; and R7...
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| creator | WOLFGANG WERNER ALFRED STRASSBURGER OSWALD ZIMMER WERNER GUNTER ENGLBERGER CLAUDIA KATHARINA PUTZ |
| description | Aminomethyl-acridine derivatives (I) are new. Aryl substituted aminomethyl-acridine derivatives of formula (I) and their salts are new. X = N and Y = C; or X = C and Y = N; R1 = A; R2 = H or OR12; R3 = H; or R2 and R3 together form a double bond; R4 = CH2NR14R15; R5 and R6 = H or 1-6C alkyl; and R7 and R8 = H; or R3 = A; R1, R2, R4, R5, R7 and R8 = H; R4 = OR12; or R1 and R4 together or R4 and R5 together form a double bond; and R6 = CH2NR4R15; or R5 = A; R1-R4 and R7 = H; R6 = H or R12; or R3 and R6 together or R6 and R7 together form a double bond; and R8 = CH2NR14R15; A = group of formula (a); R9 and R10 = H, OH, 1-6C alkoxy, Cl, F, CF3, CN, COOH, CONR17R18, or COOR16; R11 = H, OH, 1-6C alkoxy, 3-7C cycloalkyloxy, aryloxy, or heterocyclyloxy; R12 = H, 1-6C alkyl, aryl, or COR13; R13 and R16 - R18 = 1-6C alkyl or aryl; and R14 and R15 = 1-6C alkyl, aryl or 3-7C cycloalkyl. An Independent claim is also included for the preparation of compounds (I) excluding those where R1 = A, R2 = H or OR12 and R3 = H or R2 and R3 together form a double bond, R4 = CH2NR14R15, R5 and R6 = 1-6C alkyl and R7 and R8 = H. |
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Aryl substituted aminomethyl-acridine derivatives of formula (I) and their salts are new. X = N and Y = C; or X = C and Y = N; R1 = A; R2 = H or OR12; R3 = H; or R2 and R3 together form a double bond; R4 = CH2NR14R15; R5 and R6 = H or 1-6C alkyl; and R7 and R8 = H; or R3 = A; R1, R2, R4, R5, R7 and R8 = H; R4 = OR12; or R1 and R4 together or R4 and R5 together form a double bond; and R6 = CH2NR4R15; or R5 = A; R1-R4 and R7 = H; R6 = H or R12; or R3 and R6 together or R6 and R7 together form a double bond; and R8 = CH2NR14R15; A = group of formula (a); R9 and R10 = H, OH, 1-6C alkoxy, Cl, F, CF3, CN, COOH, CONR17R18, or COOR16; R11 = H, OH, 1-6C alkoxy, 3-7C cycloalkyloxy, aryloxy, or heterocyclyloxy; R12 = H, 1-6C alkyl, aryl, or COR13; R13 and R16 - R18 = 1-6C alkyl or aryl; and R14 and R15 = 1-6C alkyl, aryl or 3-7C cycloalkyl. An Independent claim is also included for the preparation of compounds (I) excluding those where R1 = A, R2 = H or OR12 and R3 = H or R2 and R3 together form a double bond, R4 = CH2NR14R15, R5 and R6 = 1-6C alkyl and R7 and R8 = H.</description><edition>6</edition><language>eng</language><subject>CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>2000</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20000120&DB=EPODOC&CC=AU&NR=3798399A$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,776,881,25542,76290</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20000120&DB=EPODOC&CC=AU&NR=3798399A$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>WOLFGANG WERNER ALFRED STRASSBURGER</creatorcontrib><creatorcontrib>OSWALD ZIMMER</creatorcontrib><creatorcontrib>WERNER GUNTER ENGLBERGER</creatorcontrib><creatorcontrib>CLAUDIA KATHARINA PUTZ</creatorcontrib><title>Acridin derivatives</title><description>Aminomethyl-acridine derivatives (I) are new. Aryl substituted aminomethyl-acridine derivatives of formula (I) and their salts are new. X = N and Y = C; or X = C and Y = N; R1 = A; R2 = H or OR12; R3 = H; or R2 and R3 together form a double bond; R4 = CH2NR14R15; R5 and R6 = H or 1-6C alkyl; and R7 and R8 = H; or R3 = A; R1, R2, R4, R5, R7 and R8 = H; R4 = OR12; or R1 and R4 together or R4 and R5 together form a double bond; and R6 = CH2NR4R15; or R5 = A; R1-R4 and R7 = H; R6 = H or R12; or R3 and R6 together or R6 and R7 together form a double bond; and R8 = CH2NR14R15; A = group of formula (a); R9 and R10 = H, OH, 1-6C alkoxy, Cl, F, CF3, CN, COOH, CONR17R18, or COOR16; R11 = H, OH, 1-6C alkoxy, 3-7C cycloalkyloxy, aryloxy, or heterocyclyloxy; R12 = H, 1-6C alkyl, aryl, or COR13; R13 and R16 - R18 = 1-6C alkyl or aryl; and R14 and R15 = 1-6C alkyl, aryl or 3-7C cycloalkyl. An Independent claim is also included for the preparation of compounds (I) excluding those where R1 = A, R2 = H or OR12 and R3 = H or R2 and R3 together form a double bond, R4 = CH2NR14R15, R5 and R6 = 1-6C alkyl and R7 and R8 = H.</description><subject>CHEMISTRY</subject><subject>HETEROCYCLIC COMPOUNDS</subject><subject>HUMAN NECESSITIES</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>METALLURGY</subject><subject>ORGANIC CHEMISTRY</subject><subject>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><subject>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>2000</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNrjZBB2TC7KTMnMU0hJLcosSyzJLEst5mFgTUvMKU7lhdLcDPJuriHOHrqpBfnxqcUFicmpeakl8Y6hxuaWFsaWlo7GhFUAALW8H-A</recordid><startdate>20000120</startdate><enddate>20000120</enddate><creator>WOLFGANG WERNER ALFRED STRASSBURGER</creator><creator>OSWALD ZIMMER</creator><creator>WERNER GUNTER ENGLBERGER</creator><creator>CLAUDIA KATHARINA PUTZ</creator><scope>EVB</scope></search><sort><creationdate>20000120</creationdate><title>Acridin derivatives</title><author>WOLFGANG WERNER ALFRED STRASSBURGER ; OSWALD ZIMMER ; WERNER GUNTER ENGLBERGER ; CLAUDIA KATHARINA PUTZ</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_AU3798399A3</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>eng</language><creationdate>2000</creationdate><topic>CHEMISTRY</topic><topic>HETEROCYCLIC COMPOUNDS</topic><topic>HUMAN NECESSITIES</topic><topic>HYGIENE</topic><topic>MEDICAL OR VETERINARY SCIENCE</topic><topic>METALLURGY</topic><topic>ORGANIC CHEMISTRY</topic><topic>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</topic><topic>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</topic><toplevel>online_resources</toplevel><creatorcontrib>WOLFGANG WERNER ALFRED STRASSBURGER</creatorcontrib><creatorcontrib>OSWALD ZIMMER</creatorcontrib><creatorcontrib>WERNER GUNTER ENGLBERGER</creatorcontrib><creatorcontrib>CLAUDIA KATHARINA PUTZ</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>WOLFGANG WERNER ALFRED STRASSBURGER</au><au>OSWALD ZIMMER</au><au>WERNER GUNTER ENGLBERGER</au><au>CLAUDIA KATHARINA PUTZ</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>Acridin derivatives</title><date>2000-01-20</date><risdate>2000</risdate><abstract>Aminomethyl-acridine derivatives (I) are new. Aryl substituted aminomethyl-acridine derivatives of formula (I) and their salts are new. X = N and Y = C; or X = C and Y = N; R1 = A; R2 = H or OR12; R3 = H; or R2 and R3 together form a double bond; R4 = CH2NR14R15; R5 and R6 = H or 1-6C alkyl; and R7 and R8 = H; or R3 = A; R1, R2, R4, R5, R7 and R8 = H; R4 = OR12; or R1 and R4 together or R4 and R5 together form a double bond; and R6 = CH2NR4R15; or R5 = A; R1-R4 and R7 = H; R6 = H or R12; or R3 and R6 together or R6 and R7 together form a double bond; and R8 = CH2NR14R15; A = group of formula (a); R9 and R10 = H, OH, 1-6C alkoxy, Cl, F, CF3, CN, COOH, CONR17R18, or COOR16; R11 = H, OH, 1-6C alkoxy, 3-7C cycloalkyloxy, aryloxy, or heterocyclyloxy; R12 = H, 1-6C alkyl, aryl, or COR13; R13 and R16 - R18 = 1-6C alkyl or aryl; and R14 and R15 = 1-6C alkyl, aryl or 3-7C cycloalkyl. An Independent claim is also included for the preparation of compounds (I) excluding those where R1 = A, R2 = H or OR12 and R3 = H or R2 and R3 together form a double bond, R4 = CH2NR14R15, R5 and R6 = 1-6C alkyl and R7 and R8 = H.</abstract><edition>6</edition><oa>free_for_read</oa></addata></record> |
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| subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| title | Acridin derivatives |
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