PYRAZOLE DERIVATIVES ASR ET KINASE INHIBITORS
Disclosed herein are compounds of formula I: or a pharmaceutically acceptable salt thereof, where the variables are as defined herein. These compounds are useful in treating RET associated cancers. Formulations containing the compounds of formula I and methods of making the compounds of formula I ar...
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| creator | PANCALDI, Thomas KOLAKOWSKI, Gabrielle BOLDRON, Christopher MCKENNEY, Megan CONDROSKI, Kevin MUNCHHOF, Michael ANDERSON, Erin ANDREWS, Steven IRVIN, Thomas KUMAR, Manoj MCFADDIN, Elizabeth MCLEAN, Johnathan PILKINGTON-MIKSA, Michael Alexander PINTO, Marta MOURET, Tiphaine |
| description | Disclosed herein are compounds of formula I: or a pharmaceutically acceptable salt thereof, where the variables are as defined herein. These compounds are useful in treating RET associated cancers. Formulations containing the compounds of formula I and methods of making the compounds of formula I are also disclosed. |
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These compounds are useful in treating RET associated cancers. Formulations containing the compounds of formula I and methods of making the compounds of formula I are also disclosed.</description><language>eng</language><subject>CHEMISTRY ; HETEROCYCLIC COMPOUNDS ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><creationdate>2024</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20240801&DB=EPODOC&CC=AU&NR=2021376367B2$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,780,885,25564,76547</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=20240801&DB=EPODOC&CC=AU&NR=2021376367B2$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>PANCALDI, Thomas</creatorcontrib><creatorcontrib>KOLAKOWSKI, Gabrielle</creatorcontrib><creatorcontrib>BOLDRON, Christopher</creatorcontrib><creatorcontrib>MCKENNEY, Megan</creatorcontrib><creatorcontrib>CONDROSKI, Kevin</creatorcontrib><creatorcontrib>MUNCHHOF, Michael</creatorcontrib><creatorcontrib>ANDERSON, Erin</creatorcontrib><creatorcontrib>ANDREWS, Steven</creatorcontrib><creatorcontrib>IRVIN, Thomas</creatorcontrib><creatorcontrib>KUMAR, Manoj</creatorcontrib><creatorcontrib>MCFADDIN, Elizabeth</creatorcontrib><creatorcontrib>MCLEAN, Johnathan</creatorcontrib><creatorcontrib>PILKINGTON-MIKSA, Michael Alexander</creatorcontrib><creatorcontrib>PINTO, Marta</creatorcontrib><creatorcontrib>MOURET, Tiphaine</creatorcontrib><title>PYRAZOLE DERIVATIVES ASR ET KINASE INHIBITORS</title><description>Disclosed herein are compounds of formula I: or a pharmaceutically acceptable salt thereof, where the variables are as defined herein. These compounds are useful in treating RET associated cancers. 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These compounds are useful in treating RET associated cancers. Formulations containing the compounds of formula I and methods of making the compounds of formula I are also disclosed.</abstract><oa>free_for_read</oa></addata></record> |
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| subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| title | PYRAZOLE DERIVATIVES ASR ET KINASE INHIBITORS |
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