Novel heterocyclic compounds as CDK8/19 inhibitors
The present invention relates to novel compounds of formula (I), or a pharmaceutically acceptable salt or stereoisomer thereof, which exhibit the properties of a CDK 8/19 inhibitor. The invention also relates to a pharmaceutical composition containing said compounds and to the use thereof as pharmac...
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| creator | KASATKINA, Mariia Andreevna CHESTNOVA, Anna Jur'evna GORBUNOVA, Svetlana Leonidovna ZAVIALOV, Kirill Vadimovich KOZHEMYAKINA, Natalia Vladimirovna POPKOVA, Aleksandra Vladimirovna ALAFINOV, Andrei Ivanovich IAKOVLEV, Pavel Andreevich KUSHAKOVA, Anna Sergeevna MOROZOV, Dmitry Valentinovich MINDICH, Aleksei Leonidovich SHEKHAUTSOU, Artsiom Evgenievich ALESHUNIN, Pavel Aleksandrovich REKHARSKY, Mikhail Vladimirovich EVDOKIMOV, Anton Aleksandrovich MAKSIMENKO, Elena Aleksandrovna MISHINA, Mariia Sergeevna |
| description | The present invention relates to novel compounds of formula (I), or a pharmaceutically acceptable salt or stereoisomer thereof, which exhibit the properties of a CDK 8/19 inhibitor. The invention also relates to a pharmaceutical composition containing said compounds and to the use thereof as pharmaceutical drugs for treating diseases or disorders. |
| format | Patent |
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| subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| title | Novel heterocyclic compounds as CDK8/19 inhibitors |
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