Purine inhibitors of human phosphatidylinositol 3-kinase delta

The instant invention provides compounds of formula I which are PI3K-delta inhibitors, and as such are useful for the treatment of PI3K-delta-mediated diseases such as inflamation, asthma, COPD and cancer.

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Hauptverfasser: GARCIA, YUDITH, KATTAR, SOLOMON, ZHAO, XIAOLI, METHOT, JOEY L, ANTHONY, NEVILLE JOHN, SHI, FENG, ACHAB, ABDELGHANI ABE, CHRISTOPHER, MATTHEW P, FONG, KIN CHIU, ALTMAN, MICHAEL D, KATZ, JASON D, LENG, XIANSHENG, YANG, LIPING, MCGOWAN, MEREDETH, FRADERA LLINAS, FRANCESC XAVIER, DENG, YONGQI, MU, CHANGWEI, YE, BAIJUN, ZHOU, HUA, ZHANG, SIXING, WANG, XIAONA, ZHANG, RONG
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creator GARCIA, YUDITH
KATTAR, SOLOMON
ZHAO, XIAOLI
METHOT, JOEY L
ANTHONY, NEVILLE JOHN
SHI, FENG
ACHAB, ABDELGHANI ABE
CHRISTOPHER, MATTHEW P
FONG, KIN CHIU
ALTMAN, MICHAEL D
KATZ, JASON D
LENG, XIANSHENG
YANG, LIPING
MCGOWAN, MEREDETH
FRADERA LLINAS, FRANCESC XAVIER
DENG, YONGQI
MU, CHANGWEI
YE, BAIJUN
ZHOU, HUA
ZHANG, SIXING
WANG, XIAONA
ZHANG, RONG
description The instant invention provides compounds of formula I which are PI3K-delta inhibitors, and as such are useful for the treatment of PI3K-delta-mediated diseases such as inflamation, asthma, COPD and cancer.
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subjects CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
title Purine inhibitors of human phosphatidylinositol 3-kinase delta
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