2-carboxamide-7-piperazinyl-benzofuran derivatives 774

The present invention relates to compounds of formula (I), wherein R is heteroaryl or heterocyclyl, optionally substituted R is Calkyl, heterocyclyl, Calkylaryl, Calkylheteroaryl, carbocyclyl, C alkylheterocyclyl, heterocyclylheteroaryl, arylheterocyclyl, carbocyclylheteroaryl, heterocyclylaryl, opt...

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Hauptverfasser: LINDE, CHRISTIAN ERIK, MALMSTROM, JONAS, NORDVALL, GUNNAR, ANDERSSON, JOHAN, WEIGELT, TATJANA, JOHANSSON, ANH, GYBACK, HELENA, TERP, GITTE
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creator LINDE, CHRISTIAN ERIK
MALMSTROM, JONAS
NORDVALL, GUNNAR
ANDERSSON, JOHAN
WEIGELT, TATJANA
JOHANSSON, ANH
GYBACK, HELENA
TERP, GITTE
description The present invention relates to compounds of formula (I), wherein R is heteroaryl or heterocyclyl, optionally substituted R is Calkyl, heterocyclyl, Calkylaryl, Calkylheteroaryl, carbocyclyl, C alkylheterocyclyl, heterocyclylheteroaryl, arylheterocyclyl, carbocyclylheteroaryl, heterocyclylaryl, optionally substituted Ris hydrogen or Calkyl, or R and R may together with the nitrogen atom, form a saturated ring system containing 4, 5 or 6 ring forming atoms, and optionally substituted R is hydrogen, halogen, methyl or methoxy to pharmaceutical composition containing said compounds and to the use of said compounds in therapy, for instance in treating cognitive disorders. The present invention further relates to new intermediates useful in the preparation thereof.
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subjects CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
title 2-carboxamide-7-piperazinyl-benzofuran derivatives 774
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