Pyridine and pyrimidine derivatives as phosphodiesterase 10 inhibitors
Pyridine and pyrimidine compounds, and compositions containing them, and processes for preparing such compounds. Provided herein also are methods of treating disorders or diseases treatable by inhibition of PDE10, such as obesity, non-insulin dependent diabetes, schizophrenia, bipolar disorder, obse...
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| creator | RUMFELT, SHANNON SHAM, KELVIN CHEN, NING DEMORIN, FRENEL FILS ALLEN, JENNIFER R HARRINGTON, PAUL KALLER, MATTHEW R MONENSCHEIN, HOLGER RZASA, ROB BISWAS, KAUSTAV HORNE, DAN YAO, GUOMIN CHAVEZ JR., FRANK FROHN, MIKE KUNZ, ROXANNE REICHELT, ANDREAS FALSEY, JAMES R PICKRELL, ALEX HU, ESSA NGUYEN, TOM |
| description | Pyridine and pyrimidine compounds, and compositions containing them, and processes for preparing such compounds. Provided herein also are methods of treating disorders or diseases treatable by inhibition of PDE10, such as obesity, non-insulin dependent diabetes, schizophrenia, bipolar disorder, obsessive-compulsive disorder, and the like. |
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Provided herein also are methods of treating disorders or diseases treatable by inhibition of PDE10, such as obesity, non-insulin dependent diabetes, schizophrenia, bipolar disorder, obsessive-compulsive disorder, and the like.</abstract><oa>free_for_read</oa></addata></record> |
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| subjects | CHEMISTRY HETEROCYCLIC COMPOUNDS HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS |
| title | Pyridine and pyrimidine derivatives as phosphodiesterase 10 inhibitors |
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