2-aminothiazole-4-carboxylic amides as protein kinase inhibitors

The present invention relates to novel Anilinopiperazine Derivatives of formula (I), compositions comprising the Anilinopiperazine Derivatives, and methods for using the Anilinopiperazine Derivatives for treating or preventing a proliferative disorder, an anti-proliferative disorder, inflammation, a...

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Hauptverfasser: SIDDIQUI, M. ARSHAD, TADIKONDA, PRAVEEN K, RICHARDS, MATTHEW, SHIPPS JR., GERALD W, CHENG, CLIFF C, DWYER, MICHAEL P, ZENG, HONGBO, SUN, BINYUAN, WONG, TZU T, ZHAO, LIANYUN, GUZI, TIMOTHY J, REDDY, PANDURANGA A, HUANG, XIAOHUA, DUCA, JOSE S, FISCHMANN, THIERRY O, KEERTIKAR, KARTIK M, TORRES, LUIS E, TANG, SHUYI
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creator SIDDIQUI, M. ARSHAD
TADIKONDA, PRAVEEN K
RICHARDS, MATTHEW
SHIPPS JR., GERALD W
CHENG, CLIFF C
DWYER, MICHAEL P
ZENG, HONGBO
SUN, BINYUAN
WONG, TZU T
ZHAO, LIANYUN
GUZI, TIMOTHY J
REDDY, PANDURANGA A
HUANG, XIAOHUA
DUCA, JOSE S
FISCHMANN, THIERRY O
KEERTIKAR, KARTIK M
TORRES, LUIS E
TANG, SHUYI
description The present invention relates to novel Anilinopiperazine Derivatives of formula (I), compositions comprising the Anilinopiperazine Derivatives, and methods for using the Anilinopiperazine Derivatives for treating or preventing a proliferative disorder, an anti-proliferative disorder, inflammation, arthritis, a central nervous system disorder, a cardiovascular disease, alopecia, a neuronal disease, an ischemic injury, a viral disease, a fungal infection, or a disorder related to the activity of a protein kinase.
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subjects CHEMISTRY
HETEROCYCLIC COMPOUNDS
HUMAN NECESSITIES
HYGIENE
MEDICAL OR VETERINARY SCIENCE
METALLURGY
ORGANIC CHEMISTRY
PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES
SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS
title 2-aminothiazole-4-carboxylic amides as protein kinase inhibitors
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