VERFAHREN ZUR HERSTELLUNG VON NEUEN AMINOACRIDIN-ALPHA- UND/ODER -BETA-(D)-N-GLYKOSID-UND/ODER AMINOACRIDIN-ALPHA- UND/ODER -BETA-(L)-N-GLYKOSIDDERIVATEN
The invention relates to novel aminoacridine- alpha , beta -(D)- and -(L)-N-glycoside derivatives, the salts thereof and to a novel process for the preparation of such compounds and salts. The novel compounds have the formula I I wherein R is hydrogen or a group of the formula II II wherein n=0 or 1...
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| creator | JANOSSY LORANT LIPTAK ANDRAS DR NANASI PAL DR POLYA KALMAN DR NESZMELYI ANDRAS. DR ERDEI JANOS DR CSERNUS ISTVAN KOVACS ANTAL DR |
| description | The invention relates to novel aminoacridine- alpha , beta -(D)- and -(L)-N-glycoside derivatives, the salts thereof and to a novel process for the preparation of such compounds and salts. The novel compounds have the formula I I wherein R is hydrogen or a group of the formula II II wherein n=0 or 1, p=1 or 2, A-p is an anion, preferably halogenide, R1 is hydrogen or a methyl group and R2 is hydrogen or a sugar residue, or R is dimethylamine, and the two substituents X and X1 are identical or different and stand for hydrogen, a group of the formula II, dimethylamine, halogen, a C1-4 alkyl group, a C1-4 alkoxy group, for a nitro-, cyano-, carbomethoxy-, carbamoyl-, phenyl- or a C1-4 alkylphenyl group, with the restriction that at least one of the substituents R, X and X1 represents a group of formula II with R2=sugar residue, and R3 is hydrogen or a C1-5 alkyl group. |
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DR ; ERDEI JANOS DR ; CSERNUS ISTVAN ; KOVACS ANTAL DR</creator><creatorcontrib>JANOSSY LORANT ; LIPTAK ANDRAS DR ; NANASI PAL DR ; POLYA KALMAN DR ; NESZMELYI ANDRAS. DR ; ERDEI JANOS DR ; CSERNUS ISTVAN ; KOVACS ANTAL DR</creatorcontrib><description>The invention relates to novel aminoacridine- alpha , beta -(D)- and -(L)-N-glycoside derivatives, the salts thereof and to a novel process for the preparation of such compounds and salts. The novel compounds have the formula I I wherein R is hydrogen or a group of the formula II II wherein n=0 or 1, p=1 or 2, A-p is an anion, preferably halogenide, R1 is hydrogen or a methyl group and R2 is hydrogen or a sugar residue, or R is dimethylamine, and the two substituents X and X1 are identical or different and stand for hydrogen, a group of the formula II, dimethylamine, halogen, a C1-4 alkyl group, a C1-4 alkoxy group, for a nitro-, cyano-, carbomethoxy-, carbamoyl-, phenyl- or a C1-4 alkylphenyl group, with the restriction that at least one of the substituents R, X and X1 represents a group of formula II with R2=sugar residue, and R3 is hydrogen or a C1-5 alkyl group.</description><edition>4</edition><language>ger</language><subject>CHEMISTRY ; DERIVATIVES THEREOF ; HUMAN NECESSITIES ; HYGIENE ; MEDICAL OR VETERINARY SCIENCE ; METALLURGY ; NUCLEIC ACIDS ; NUCLEOSIDES ; NUCLEOTIDES ; ORGANIC CHEMISTRY ; PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES ; SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS ; SUGARS</subject><creationdate>1985</creationdate><oa>free_for_read</oa><woscitedreferencessubscribed>false</woscitedreferencessubscribed></display><links><openurl>$$Topenurl_article</openurl><openurlfulltext>$$Topenurlfull_article</openurlfulltext><thumbnail>$$Tsyndetics_thumb_exl</thumbnail><linktohtml>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=19851015&DB=EPODOC&CC=AT&NR=A73382A$$EHTML$$P50$$Gepo$$Hfree_for_read</linktohtml><link.rule.ids>230,308,776,881,25543,76293</link.rule.ids><linktorsrc>$$Uhttps://worldwide.espacenet.com/publicationDetails/biblio?FT=D&date=19851015&DB=EPODOC&CC=AT&NR=A73382A$$EView_record_in_European_Patent_Office$$FView_record_in_$$GEuropean_Patent_Office$$Hfree_for_read</linktorsrc></links><search><creatorcontrib>JANOSSY LORANT</creatorcontrib><creatorcontrib>LIPTAK ANDRAS DR</creatorcontrib><creatorcontrib>NANASI PAL DR</creatorcontrib><creatorcontrib>POLYA KALMAN DR</creatorcontrib><creatorcontrib>NESZMELYI ANDRAS. DR</creatorcontrib><creatorcontrib>ERDEI JANOS DR</creatorcontrib><creatorcontrib>CSERNUS ISTVAN</creatorcontrib><creatorcontrib>KOVACS ANTAL DR</creatorcontrib><title>VERFAHREN ZUR HERSTELLUNG VON NEUEN AMINOACRIDIN-ALPHA- UND/ODER -BETA-(D)-N-GLYKOSID-UND/ODER AMINOACRIDIN-ALPHA- UND/ODER -BETA-(L)-N-GLYKOSIDDERIVATEN</title><description>The invention relates to novel aminoacridine- alpha , beta -(D)- and -(L)-N-glycoside derivatives, the salts thereof and to a novel process for the preparation of such compounds and salts. The novel compounds have the formula I I wherein R is hydrogen or a group of the formula II II wherein n=0 or 1, p=1 or 2, A-p is an anion, preferably halogenide, R1 is hydrogen or a methyl group and R2 is hydrogen or a sugar residue, or R is dimethylamine, and the two substituents X and X1 are identical or different and stand for hydrogen, a group of the formula II, dimethylamine, halogen, a C1-4 alkyl group, a C1-4 alkoxy group, for a nitro-, cyano-, carbomethoxy-, carbamoyl-, phenyl- or a C1-4 alkylphenyl group, with the restriction that at least one of the substituents R, X and X1 represents a group of formula II with R2=sugar residue, and R3 is hydrogen or a C1-5 alkyl group.</description><subject>CHEMISTRY</subject><subject>DERIVATIVES THEREOF</subject><subject>HUMAN NECESSITIES</subject><subject>HYGIENE</subject><subject>MEDICAL OR VETERINARY SCIENCE</subject><subject>METALLURGY</subject><subject>NUCLEIC ACIDS</subject><subject>NUCLEOSIDES</subject><subject>NUCLEOTIDES</subject><subject>ORGANIC CHEMISTRY</subject><subject>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</subject><subject>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</subject><subject>SUGARS</subject><fulltext>true</fulltext><rsrctype>patent</rsrctype><creationdate>1985</creationdate><recordtype>patent</recordtype><sourceid>EVB</sourceid><recordid>eNqNi7EKwjAURbs4iPoLklGHh2AHuz6b1yYYXyRNCrqUInESLdSf8W_tIOKm04V7zhknz5pcgcoRi1NwQpGrPBkTuBS1ZcEUBoJ7zRZzp6VmQHNQCCKwXFlJTsCWPMJCLoGhNMedrbSED_0nNd_p8OsaPfE0GV3aax9n750k84J8riB29yb2XXuOt_ho0OMmTbM1pj-FF76YQTQ</recordid><startdate>19851015</startdate><enddate>19851015</enddate><creator>JANOSSY LORANT</creator><creator>LIPTAK ANDRAS DR</creator><creator>NANASI PAL DR</creator><creator>POLYA KALMAN DR</creator><creator>NESZMELYI ANDRAS. 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DR ; ERDEI JANOS DR ; CSERNUS ISTVAN ; KOVACS ANTAL DR</author></sort><facets><frbrtype>5</frbrtype><frbrgroupid>cdi_FETCH-epo_espacenet_ATA73382A3</frbrgroupid><rsrctype>patents</rsrctype><prefilter>patents</prefilter><language>ger</language><creationdate>1985</creationdate><topic>CHEMISTRY</topic><topic>DERIVATIVES THEREOF</topic><topic>HUMAN NECESSITIES</topic><topic>HYGIENE</topic><topic>MEDICAL OR VETERINARY SCIENCE</topic><topic>METALLURGY</topic><topic>NUCLEIC ACIDS</topic><topic>NUCLEOSIDES</topic><topic>NUCLEOTIDES</topic><topic>ORGANIC CHEMISTRY</topic><topic>PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES</topic><topic>SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS</topic><topic>SUGARS</topic><toplevel>online_resources</toplevel><creatorcontrib>JANOSSY LORANT</creatorcontrib><creatorcontrib>LIPTAK ANDRAS DR</creatorcontrib><creatorcontrib>NANASI PAL DR</creatorcontrib><creatorcontrib>POLYA KALMAN DR</creatorcontrib><creatorcontrib>NESZMELYI ANDRAS. DR</creatorcontrib><creatorcontrib>ERDEI JANOS DR</creatorcontrib><creatorcontrib>CSERNUS ISTVAN</creatorcontrib><creatorcontrib>KOVACS ANTAL DR</creatorcontrib><collection>esp@cenet</collection></facets><delivery><delcategory>Remote Search Resource</delcategory><fulltext>fulltext_linktorsrc</fulltext></delivery><addata><au>JANOSSY LORANT</au><au>LIPTAK ANDRAS DR</au><au>NANASI PAL DR</au><au>POLYA KALMAN DR</au><au>NESZMELYI ANDRAS. DR</au><au>ERDEI JANOS DR</au><au>CSERNUS ISTVAN</au><au>KOVACS ANTAL DR</au><format>patent</format><genre>patent</genre><ristype>GEN</ristype><title>VERFAHREN ZUR HERSTELLUNG VON NEUEN AMINOACRIDIN-ALPHA- UND/ODER -BETA-(D)-N-GLYKOSID-UND/ODER AMINOACRIDIN-ALPHA- UND/ODER -BETA-(L)-N-GLYKOSIDDERIVATEN</title><date>1985-10-15</date><risdate>1985</risdate><abstract>The invention relates to novel aminoacridine- alpha , beta -(D)- and -(L)-N-glycoside derivatives, the salts thereof and to a novel process for the preparation of such compounds and salts. The novel compounds have the formula I I wherein R is hydrogen or a group of the formula II II wherein n=0 or 1, p=1 or 2, A-p is an anion, preferably halogenide, R1 is hydrogen or a methyl group and R2 is hydrogen or a sugar residue, or R is dimethylamine, and the two substituents X and X1 are identical or different and stand for hydrogen, a group of the formula II, dimethylamine, halogen, a C1-4 alkyl group, a C1-4 alkoxy group, for a nitro-, cyano-, carbomethoxy-, carbamoyl-, phenyl- or a C1-4 alkylphenyl group, with the restriction that at least one of the substituents R, X and X1 represents a group of formula II with R2=sugar residue, and R3 is hydrogen or a C1-5 alkyl group.</abstract><edition>4</edition><oa>free_for_read</oa></addata></record> |
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| subjects | CHEMISTRY DERIVATIVES THEREOF HUMAN NECESSITIES HYGIENE MEDICAL OR VETERINARY SCIENCE METALLURGY NUCLEIC ACIDS NUCLEOSIDES NUCLEOTIDES ORGANIC CHEMISTRY PREPARATIONS FOR MEDICAL, DENTAL, OR TOILET PURPOSES SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS ORMEDICINAL PREPARATIONS SUGARS |
| title | VERFAHREN ZUR HERSTELLUNG VON NEUEN AMINOACRIDIN-ALPHA- UND/ODER -BETA-(D)-N-GLYKOSID-UND/ODER AMINOACRIDIN-ALPHA- UND/ODER -BETA-(L)-N-GLYKOSIDDERIVATEN |
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