Bruton's Tyrosine Kinase (BTK) Degrader Nx-2127 Exhibits Lethal Activity and Synergy with Venetoclax and BET Protein Inhibitor Against MCL Cells Sensitive or Resistant to Covalent BTK Inhibitors

Bruton's Tyrosine Kinase (BTK) Degrader Nx-2127 Exhibits Lethal Activity and Synergy with Venetoclax and BET Protein Inhibitor Against MCL Cells Sensitive or Resistant to Covalent BTK Inhibitors

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Veröffentlicht in:Blood 2022-11, Vol.140 (Supplement 1), p.5980-5981
Hauptverfasser: Fiskus, Warren C., Das, Kaberi, Mill, Christopher Peter, Birdwell, Christine E, Davis, John A., Alhamadani, Noor, Philip, Kevin, Tan, May, Brown, Robert A, Green, Michael R, Bhalla, Kapil N.
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container_end_page 5981
container_issue Supplement 1
container_start_page 5980
container_title Blood
container_volume 140
creator Fiskus, Warren C.
Das, Kaberi
Mill, Christopher Peter
Birdwell, Christine E
Davis, John A.
Alhamadani, Noor
Philip, Kevin
Tan, May
Brown, Robert A
Green, Michael R
Bhalla, Kapil N.
description
doi_str_mv 10.1182/blood-2022-168483
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title Bruton's Tyrosine Kinase (BTK) Degrader Nx-2127 Exhibits Lethal Activity and Synergy with Venetoclax and BET Protein Inhibitor Against MCL Cells Sensitive or Resistant to Covalent BTK Inhibitors
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