Biarylcarbamoylindolines Are Novel and Selective 5-HT 2C Receptor Inverse Agonists:  Identification of 5-Methyl-1-[[2-[(2-methyl-3-pyridyl)oxy]- 5-pyridyl]carbamoyl]-6-trifluoromethylindoline (SB-243213) as a Potential Antidepressant/Anxiolytic Agent

Biarylcarbamoylindolines Are Novel and Selective 5-HT 2C Receptor Inverse Agonists:  Identification of 5-Methyl-1-[[2-[(2-methyl-3-pyridyl)oxy]- 5-pyridyl]carbamoyl]-6-trifluoromethylindoline (SB-243213) as a Potential Antidepressant/Anxiolytic Agent

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Veröffentlicht in:Journal of medicinal chemistry 2000-03, Vol.43 (6), p.1123-1134
Hauptverfasser: Bromidge, Steven M., Dabbs, Steven, Davies, David T., Davies, Susannah, Duckworth, D. Malcolm, Forbes, Ian T., Gaster, Laramie M., Ham, Peter, Jones, Graham E., King, Frank D., Mulholland, Keith R., Saunders, Damian V., Wyman, Paul A., Blaney, Frank E., Clarke, Stephen E., Blackburn, Thomas P., Holland, Vicky, Kennett, Guy A., Lightowler, Sean, Middlemiss, Derek N., Trail, Brenda, Riley, Graham J., Wood, Martyn D.
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container_end_page 1134
container_issue 6
container_start_page 1123
container_title Journal of medicinal chemistry
container_volume 43
creator Bromidge, Steven M.
Dabbs, Steven
Davies, David T.
Davies, Susannah
Duckworth, D. Malcolm
Forbes, Ian T.
Gaster, Laramie M.
Ham, Peter
Jones, Graham E.
King, Frank D.
Mulholland, Keith R.
Saunders, Damian V.
Wyman, Paul A.
Blaney, Frank E.
Clarke, Stephen E.
Blackburn, Thomas P.
Holland, Vicky
Kennett, Guy A.
Lightowler, Sean
Middlemiss, Derek N.
Trail, Brenda
Riley, Graham J.
Wood, Martyn D.
description
doi_str_mv 10.1021/jm990388c
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title Biarylcarbamoylindolines Are Novel and Selective 5-HT 2C Receptor Inverse Agonists:  Identification of 5-Methyl-1-[[2-[(2-methyl-3-pyridyl)oxy]- 5-pyridyl]carbamoyl]-6-trifluoromethylindoline (SB-243213) as a Potential Antidepressant/Anxiolytic Agent
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