Design, Synthesis, and Biological Evaluation of New 8-Heterocyclic Xanthine Derivatives as Highly Potent and Selective Human A 2B Adenosine Receptor Antagonists

Design, Synthesis, and Biological Evaluation of New 8-Heterocyclic Xanthine Derivatives as Highly Potent and Selective Human A 2B Adenosine Receptor Antagonists

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Veröffentlicht in:Journal of medicinal chemistry 2004-03, Vol.47 (6), p.1434-1447
Hauptverfasser: Baraldi, Pier Giovanni, Tabrizi, Mojgan Aghazadeh, Preti, Delia, Bovero, Andrea, Romagnoli, Romeo, Fruttarolo, Francesca, Zaid, Naser Abdel, Moorman, Allan R., Varani, Katia, Gessi, Stefania, Merighi, Stefania, Borea, Pier Andrea
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container_end_page 1447
container_issue 6
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container_title Journal of medicinal chemistry
container_volume 47
creator Baraldi, Pier Giovanni
Tabrizi, Mojgan Aghazadeh
Preti, Delia
Bovero, Andrea
Romagnoli, Romeo
Fruttarolo, Francesca
Zaid, Naser Abdel
Moorman, Allan R.
Varani, Katia
Gessi, Stefania
Merighi, Stefania
Borea, Pier Andrea
description
doi_str_mv 10.1021/jm0309654
format Article
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title Design, Synthesis, and Biological Evaluation of New 8-Heterocyclic Xanthine Derivatives as Highly Potent and Selective Human A 2B Adenosine Receptor Antagonists
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