Novel Selective PDE4 Inhibitors. 1. Synthesis, Structure−Activity Relationships, and Molecular Modeling of 4-(3,4-Dimethoxyphenyl)-2 H -phthalazin-1-ones and Analogues

Novel Selective PDE4 Inhibitors. 1. Synthesis, Structure−Activity Relationships, and Molecular Modeling of 4-(3,4-Dimethoxyphenyl)-2 H -phthalazin-1-ones and Analogues

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Veröffentlicht in:Journal of medicinal chemistry 2001-08, Vol.44 (16), p.2511-2522
Hauptverfasser: Van der Mey, Margaretha, Hatzelmann, Armin, Van der Laan, Ivonne J., Sterk, Geert J., Thibaut, Ulrich, Timmerman, Hendrik
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container_end_page 2522
container_issue 16
container_start_page 2511
container_title Journal of medicinal chemistry
container_volume 44
creator Van der Mey, Margaretha
Hatzelmann, Armin
Van der Laan, Ivonne J.
Sterk, Geert J.
Thibaut, Ulrich
Timmerman, Hendrik
description
doi_str_mv 10.1021/jm010837k
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title Novel Selective PDE4 Inhibitors. 1. Synthesis, Structure−Activity Relationships, and Molecular Modeling of 4-(3,4-Dimethoxyphenyl)-2 H -phthalazin-1-ones and Analogues
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