Quinazoline antifolate thymidylate synthase inhibitors: 2'-Fluoro-N10-propargyl-5,8,-dideazafolic acid and derivatives with modifications in the C-2 position

Quinazoline antifolate thymidylate synthase inhibitors: 2'-Fluoro-N10-propargyl-5,8,-dideazafolic acid and derivatives with modifications in the C-2 position

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Veröffentlicht in:Journal of medicinal chemistry 1990-11, Vol.33 (11), p.3067-3071
Hauptverfasser: Jackman, Ann L, Marsham, Peter R, Thornton, Timothy J, Bishop, Joel A. M, O'Connor, Brigid M, Hughes, Leslie R, Calvert, A. Hilary, Jones, Terence R
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container_end_page 3071
container_issue 11
container_start_page 3067
container_title Journal of medicinal chemistry
container_volume 33
creator Jackman, Ann L
Marsham, Peter R
Thornton, Timothy J
Bishop, Joel A. M
O'Connor, Brigid M
Hughes, Leslie R
Calvert, A. Hilary
Jones, Terence R
description
doi_str_mv 10.1021/jm00173a025
format Article
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title Quinazoline antifolate thymidylate synthase inhibitors: 2'-Fluoro-N10-propargyl-5,8,-dideazafolic acid and derivatives with modifications in the C-2 position
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