5′-Substituted Amiloride Derivatives as Allosteric Modulators Binding in the Sodium Ion Pocket of the Adenosine A 2A Receptor

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Veröffentlicht in:Journal of medicinal chemistry 2016-05, Vol.59 (10), p.4769-4777
Hauptverfasser: Massink, Arnault, Louvel, Julien, Adlere, Ilze, van Veen, Corine, Huisman, Berend J. H., Dijksteel, Gabrielle S., Guo, Dong, Lenselink, Eelke B., Buckley, Benjamin J., Matthews, Hayden, Ranson, Marie, Kelso, Michael, IJzerman, Adriaan P.
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container_end_page 4777
container_issue 10
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container_title Journal of medicinal chemistry
container_volume 59
creator Massink, Arnault
Louvel, Julien
Adlere, Ilze
van Veen, Corine
Huisman, Berend J. H.
Dijksteel, Gabrielle S.
Guo, Dong
Lenselink, Eelke B.
Buckley, Benjamin J.
Matthews, Hayden
Ranson, Marie
Kelso, Michael
IJzerman, Adriaan P.
description
doi_str_mv 10.1021/acs.jmedchem.6b00142
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title 5′-Substituted Amiloride Derivatives as Allosteric Modulators Binding in the Sodium Ion Pocket of the Adenosine A 2A Receptor
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