Isomerization of Allylbenzenes von Hassam, Mohammad, Taher, Abu, Arnott, Gareth E, Green, Ivan R, van Otterlo, Willem A. L

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Metathesis in the Synthesis of Aromatic Compounds von van Otterlo, Willem A. L, de Koning, Charles B

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Covalent-Allosteric Kinase Inhibitors von Weisner, Jörn, Gontla, Rajesh, van der Westhuizen, Leandi, Oeck, Sebastian, Ketzer, Julia, Janning, Petra, Richters, André, Mühlenberg, Thomas, Fang, Zhizhou, Taher, Abu, Jendrossek, Verena, Pelly, Stephen C., Bauer, Sebastian, van Otterlo, Willem A. L., Rauh, Daniel

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The role of silicon in drug discovery: a review von Panayides, Jenny-Lee, Riley, Darren Lyall, Hasenmaile, Felix, van Otterlo, Willem A. L

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The Phylum Bryozoa: From Biology to Biomedical Potential von Ciavatta, Maria Letizia, Lefranc, Florence, Vieira, Leandro M, Kiss, Robert, Carbone, Marianna, van Otterlo, Willem A L, Lopanik, Nicole B, Waeschenbach, Andrea

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Inhibition of osimertinib-resistant epidermal growth factor receptor EGFR-T790M/C797S von Lategahn, Jonas, Keul, Marina, Klvekorn, Philip, Tumbrink, Hannah L, Niggenaber, Janina, Mller, Matthias P, Hodson, Luke, Flahoff, Maren, Hardick, Julia, Grabe, Tobias, Engel, Julian, Schultz-Fademrecht, Carsten, Baumann, Matthias, Ketzer, Julia, Mhlenberg, Thomas, Hiller, Wolf, Gnther, Georgia, Unger, Anke, Mller, Heiko, Heimsoeth, Alena, Golz, Christopher, Blank-Landeshammer, Bernhard, Kollipara, Laxmikanth, Zahedi, Ren P, Strohmann, Carsten, Hengstler, Jan G, van Otterlo, Willem A. L, Bauer, Sebastian, Rauh, Daniel

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New hemisynthetic derivatives of sphaeropsidin phytotoxins triggering severe endoplasmic reticulum swelling in cancer cells von Ingels, Aude, Scott, Robert, Hooper, Annie R., van der Westhuyzen, Aletta E., Wagh, Sachin B., de Meester, Joséphine, Maddau, Lucia, Marko, Doris, Aichinger, Georg, Berger, Walter, Vermeersch, Marjorie, Pérez-Morga, David, Maslivetc, Vladimir A., Evidente, Antonio, van Otterlo, Willem A. L., Kornienko, Alexander, Mathieu, Véronique

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In search of a treatment for HIV - current therapies and the role of non-nucleoside reverse transcriptase inhibitors (NNRTIs) von Reynolds, Chevonne, de Koning, Charles B, Pelly, Stephen C, van Otterlo, Willem A. L, Bode, Moira L

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Unprecedented Direct Asymmetric Total Syntheses of 5,8’‐Naphthylisoquinoline Alkaloids from their Fully Substituted Precursors Employing a Novel Nickel/N,N‐ligand‐Catalyzed Atropos... von Berthold, Dino, van Otterlo, Willem A. L.

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Deciphering the chemical instability of sphaeropsidin A under physiological conditions - degradation studies and structural elucidation of the major metabolite von van der Westhuyzen, Alet E, Ingels, Aude, Rosière, Rémi, Amighi, Karim, Oberer, Lukas, Gustafson, Kirk R, Wang, Dongdong, Evidente, Antonio, Maddau, Lucia, Masi, Marco, de Villiers, André, Green, Ivan R, Berger, Walter, Kornienko, Alexander, Mathieu, Veronique, van Otterlo, Willem A. L

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Atroposelective NiII‐Catalyzed Cross‐Coupling Reactions Enable a Deeper Understanding of Negishi Couplings: Isolation and Application of Solid Aryl Higher‐Order Zincates von Groß, Damian, Otterlo, Willem A. L., Trapp, Oliver, Berthold, Dino

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The synthesis of 2- and 3-aryl indoles and 1,3,4,5-tetrahydropyrano[4,3- b]indoles and their antibacterial and antifungal activity von Leboho, Tlabo C., Michael, Joseph P., van Otterlo, Willem A.L., van Vuuren, Sandy F., de Koning, Charles B.

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In search of a cytostatic agent derived from the alkaloid lycorine: Synthesis and growth inhibitory properties of lycorine derivatives von Evdokimov, Nikolai M., Lamoral-Theys, Delphine, Mathieu, Véronique, Andolfi, Anna, Frolova, Liliya V., Pelly, Stephen C., van Otterlo, Willem A.L., Magedov, Igor V., Kiss, Robert, Evidente, Antonio, Kornienko, Alexander

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Microtubule‐Targeting 7‐Deazahypoxanthines Derived from Marine Alkaloid Rigidins: Exploration of the N3 and N9 Positions and Interaction with Multidrug‐Resistance Proteins von Dasari, Ramesh, Błauż, Andrzej, Medellin, Derek C., Kassim, Roaa M., Viera, Carlos, Santarosa, Maximo, van der Westhuyzen, Alet E., van Otterlo, Willem A. L., Olivas, Taryn, Yildiz, Tugba, Betancourt, Tania, Shuster, Charles B., Rogelj, Snezna, Rychlik, Błażej, Hudnall, Todd, Frolova, Liliya V., Kornienko, Alexander

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Overcoming synthetic challenges in targeting coenzyme A biosynthesis with the antimicrobial natural product CJ-15,801 von Domingo, Riyad, van der Westhuyzen, Renier, Hamann, Anton R, Mostert, Konrad J, Barnard, Leanne, Paquet, Tanya, Tjhin, Erick T, Saliba, Kevin J, van Otterlo, Willem A. L, Strauss, Erick

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Stealth lipoplex decorated with triazole-tethered galactosyl moieties: a strong hepatotropic gene vector von Govender, Dhineshree, Islam, Rafique Ul, De Koning, Charles B, van Otterlo, Willem A. L, Arbuthnot, Patrick, Ariatti, Mario, Singh, Moganavelli

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Sphaeropsidin A C15–C16 Cross‐Metathesis Analogues with Potent Anticancer Activity von Wagh, Sachin B., Berthold, Dino, Majeed, Iram, Lewis, L. Kevin, Schilter, David, Mertens, Birgit, Evidente, Antonio, Otterlo, Willem A. L., Mathieu, Véronique, Kornienko, Alexander

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Targeting Her2-insYVMA with Covalent InhibitorsA Focused Compound Screening and Structure-Based Design Approach von Lategahn, Jonas, Hardick, Julia, Grabe, Tobias, Niggenaber, Janina, Jeyakumar, Kirujan, Keul, Marina, Tumbrink, Hannah L, Becker, Christian, Hodson, Luke, Kirschner, Tonia, Klövekorn, Philip, Ketzer, Julia, Baumann, Matthias, Terheyden, Susanne, Unger, Anke, Weisner, Jörn, Müller, Matthias P, van Otterlo, Willem A. L, Bauer, Sebastian, Rauh, Daniel

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Metathesis Reactions for the Synthesis of Ring-Fused Carbazoles von Pelly, Stephen C, Parkinson, Christopher J, van Otterlo, Willem A. L, de Koning, Charles B

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Alkaloids with Activity against the Zika Virus Vector Aedes aegypti (L.)-Crinsarnine and Sarniensinol, Two New Crinine and Mesembrine Type Alkaloids Isolated from the South African... von Masi, Marco, Cala, Antonio, Tabanca, Nurhayat, Cimmino, Alessio, Green, Ivan R, Bloomquist, Jeffrey R, van Otterlo, Willem A L, Macias, Francisco A, Evidente, Antonio

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