The Role of Water Networks in Phosphodiesterase Inhibitor Dissociation and Kinetic Selectivity von Blaazer, Antoni R., Singh, Abhimanyu K., Zara, Lorena, Boronat, Pierre, Bautista, Lady J., Irving, Steve, Majewski, Maciej, Barril, Xavier, Wijtmans, Maikel, Danielson, U. Helena, Sterk, Geert Jan, Leurs, Rob, Muijlwijk‐Koezen, Jacqueline E., Brown, David G., Esch, Iwan J. P.

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Online Versus Offline Peer Feedback in Higher Education: A Meta-Analysis von Jongsma, Mirella V., Scholten, Danny J., van Muijlwijk-Koezen, Jacqueline E., Meeter, Martijn

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From Insight to Modulation of CXCR4 and ACKR3 (CXCR7) Function von Smit, Martine J., van Muijlwijk-Koezen, Jacqueline E.

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Activating Students’ Interest and Participation in Lectures and Practical Courses Using Their Electronic Devices von Wijtmans, Maikel, van Rens, Lisette, van Muijlwijk-Koezen, Jacqueline E

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From recipe to research: introducing undergraduate students to the nature of science using a hybrid practical course centred on drug discovery for neglected diseases von Wijtmans, Maikel, Edink, Ewald, van Linden, Oscar PJ, Zheng, Yang, Blaazer, Antoni R, Siderius, Marco, van Muijlwijk-Koezen, Jacqueline E

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Progress in Free Energy Perturbation: Options for Evolving Fragments von Zara, Lorena, Efrém, Nina-Louisa, van Muijlwijk-Koezen, Jacqueline E., de Esch, Iwan J.P., Zarzycka, Barbara

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Discovery of fragments inducing conformational effects in dynamic proteins using a second-harmonic generation biosensor von FitzGerald, Edward A, Butko, Margaret T, Boronat, Pierre, Cederfelt, Daniela, Abramsson, Mia, Ludviksdottir, Hildur, van Muijlwijk-Koezen, Jacqueline E, de Esch, Iwan J. P, Dobritzsch, Doreen, Young, Tracy, Danielson, U. Helena

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Practical Guidelines to Redesign Introductory Chemistry Courses Using a Flexible and Adaptive Blended Format von Scholten, Danny J, Wijtmans, Maikel, Dekker, Stefan J, Vuuregge, Anna H, Boon, Erik J. J, Vos, J. Chris, Siderius, Marco, Westbroek, Hanna, van Muijlwijk-Koezen, Jacqueline E

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Exploring the Activity Profile of TbrPDEB1 and hPDE4 Inhibitors Using Free Energy Perturbation von Zara, Lorena, Moraca, Francesca, Van Muijlwijk-Koezen, Jacqueline E., Zarzycka, Barbara, Abel, Robert, de Esch, Iwan J. P.

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Enhancing trust, safety and quality: exploring the role of dialogue in peer feedback on professional competencies von Jongsma, Mirella V., Scholten, Danny J., Houtkamp, Jorick, Meeter, Martijn, van Muijlwijk-Koezen, Jacqueline E.

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Structure-Activity Relationships of Quinoxaline-Based 5-HT3A and 5-HT3AB Receptor-Selective Ligands von Thompson, Andrew J., Verheij, Mark H. P., van Muijlwijk-Koezen, Jacqueline E., Lummis, Sarah C. R., Leurs, Rob, de Esch, Iwan J. P.

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Design, Synthesis, and Structure–Activity Relationships of Highly Potent 5‑HT3 Receptor Ligands von Verheij, Mark H. P, Thompson, Andrew J, van Muijlwijk-Koezen, Jacqueline E, Lummis, Sarah C. R, Leurs, Rob, de Esch, Iwan J. P

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Small and colorful stones make beautiful mosaics: fragment-based chemogenomics von de Graaf, Chris, Vischer, Henry F., de Kloe, Gerdien E., Kooistra, Albert J., Nijmeijer, Saskia, Kuijer, Martien, Verheij, Mark H.P., England, Paul J., van Muijlwijk-Koezen, Jacqueline E., Leurs, Rob, de Esch, Iwan J.P.

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Exploration of the molecular architecture of the orthosteric binding site in the α4β2 nicotinic acetylcholine receptor with analogs of 3-(dimethylamino)butyl dimethylcarbamate (DMA... von Bach, Tinna B., Jensen, Anders A., Petersen, Jette G., Sørensen, Troels E., Della Volpe, Serena, Liu, Jun, Blaazer, Antoni R., van Muijlwijk-Koezen, Jacqueline E., Balle, Thomas, Frølund, Bente

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Thiazole and Thiadiazole Analogues as a Novel Class of Adenosine Receptor Antagonists von van Muijlwijk-Koezen, Jacqueline E, Timmerman, Hendrik, Vollinga, Roeland C, Frijtag von Drabbe Künzel, Jacobien, de Groote, Miriam, Visser, Sven, IJzerman, Adriaan P

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Surface Plasmon Resonance Biosensor Based Fragment Screening Using Acetylcholine Binding Protein Identifies Ligand Efficiency Hot Spots (LE Hot Spots) by Deconstruction of Nicotini... von de Kloe, Gerdien E, Retra, Kim, Geitmann, Matthis, Källblad, Per, Nahar, Tariq, van Elk, René, Smit, August B, van Muijlwijk-Koezen, Jacqueline E, Leurs, Rob, Irth, Hubertus, Danielson, U. Helena, de Esch, Iwan J. P

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A Novel Class of Adenosine A3 Receptor Ligands. 2. Structure Affinity Profile of a Series of Isoquinoline and Quinazoline Compounds von van Muijlwijk-Koezen, Jacqueline E, Timmerman, Henk, Link, Regina, van der Goot, Henk, IJzerman, Adriaan P

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Isoquinoline and Quinazoline Urea Analogues as Antagonists for the Human Adenosine A3 Receptor von van Muijlwijk-Koezen, Jacqueline E, Timmerman, Henk, van der Goot, Henk, Menge, Wiro M. P. B, Frijtag von Drabbe Künzel, Jacobien, de Groote, Miriam, IJzerman, Adriaan P

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Structure-based design, synthesis and structure–activity relationships of dibenzosuberyl- and benzoate-substituted tropines as ligands for acetylcholine-binding protein von Edink, Ewald, Akdemir, Atilla, Jansen, Chimed, Elk, René van, Zuiderveld, Obbe, de Kanter, Frans J.J., van Muijlwijk-Koezen, Jacqueline E., Smit, August B., Leurs, Rob, de Esch, Iwan J.P.

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A Novel Class of Adenosine A3 Receptor Ligands. 1. 3-(2-Pyridinyl)isoquinoline Derivatives von van Muijlwijk-Koezen, Jacqueline E, Timmerman, Henk, Link, Regina, van der Goot, Henk, IJzerman, Adriaan P

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