Potentiation of rifampin activity in a mouse model of tuberculosis by activation of host transcription factor EB von Bryk, Ruslana, Mundhra, Shashirekha, Jiang, Xiuju, Wood, Madeleine, Pfau, Daniel, Weber, Elaina, Park, Suna, Zhang, Li, Wilson, Colin, Van der Westhuyzen, Renier, Street, Leslie J., Chibale, Kelly, Zimmerman, Matthew, Dartois, Veronique, Pastore, Nunzia, Ballabio, Andrea, Hawryluk, Natalie, Canan, Stacie, Khetani, Vikram, Camardo, Joseph, Nathan, Carl

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Overcoming synthetic challenges in targeting coenzyme A biosynthesis with the antimicrobial natural product CJ-15,801 von Domingo, Riyad, van der Westhuyzen, Renier, Hamann, Anton R, Mostert, Konrad J, Barnard, Leanne, Paquet, Tanya, Tjhin, Erick T, Saliba, Kevin J, van Otterlo, Willem A. L, Strauss, Erick

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Turnover-Dependent Covalent Inactivation of Staphylococcus aureus Coenzyme A‑Disulfide Reductase by Coenzyme A‑Mimetics: Mechanistic and Structural Insights von Wallace, Bret D, Edwards, Jonathan S, Wallen, Jamie R, Moolman, Wessel J. A, van der Westhuyzen, Renier, Strauss, Erick, Redinbo, Matthew R, Claiborne, Al

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Michael Acceptor-Containing Coenzyme A Analogues As Inhibitors of the Atypical Coenzyme A Disulfide Reductase from Staphylococcus aureus von van der Westhuyzen, Renier, Strauss, Erick

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Defining the Determinants of Specificity of Plasmodium Proteasome Inhibitors von Yoo, Euna, Stokes, Barbara H, de Jong, Hanna, Vanaerschot, Manu, Kumar, TRS, Lawrence, Nina, Njoroge, Mathew, Garcia, Arnold, Van der Westhuyzen, Renier, Momper, Jeremiah D, Ng, Caroline L, Fidock, David A, Bogyo, Matthew

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Pyrrolo[3,4‑c]pyridine-1,3(2H)‑diones: A Novel Antimycobacterial Class Targeting Mycobacterial Respiration von van der Westhuyzen, Renier, Winks, Susan, Wilson, Colin R, Boyle, Grant A, Gessner, Richard K, Soares de Melo, Candice, Taylor, Dale, de Kock, Carmen, Njoroge, Mathew, Brunschwig, Christel, Lawrence, Nina, Rao, Srinivasa P.S, Sirgel, Frederick, van Helden, Paul, Seldon, Ronnett, Moosa, Atica, Warner, Digby F, Arista, Luca, Manjunatha, Ujjini H, Smith, Paul W, Street, Leslie J, Chibale, Kelly

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Benzoheterocyclic Oxime Carbamates Active against Mycobacterium tuberculosis: Synthesis, Structure–Activity Relationship, Metabolism, and Biology Triaging von van der Westhuyzen, Renier, Mabhula, Amanda, Njaria, Paul M, Müller, Rudolf, Ngumbu Muhunga, Denis, Taylor, Dale, Lawrence, Nina, Njoroge, Mathew, Brunschwig, Christel, Moosa, Atica, Singh, Vinayak, Rao, Srinivasa P.S, Manjunatha, Ujjini H, Smith, Paul W, Warner, Digby F, Street, Leslie J, Chibale, Kelly

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Aminopyrazolo[1,5-a]pyrimidines as potential inhibitors of Mycobacterium tuberculosis: Structure activity relationships and ADME characterization von Soares de Melo, Candice, Feng, Tzu-Shean, van der Westhuyzen, Renier, Gessner, Richard K., Street, Leslie J., Morgans, Garreth L., Warner, Digby F., Moosa, Atica, Naran, Krupa, Lawrence, Nina, Boshoff, Helena I.M., Barry, Clifton E., Harris, C. John, Gordon, Richard, Chibale, Kelly

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The Antibiotic CJ-15,801 Is an Antimetabolite that Hijacks and Then Inhibits CoA Biosynthesis von van der Westhuyzen, Renier, Hammons, Justin C., Meier, Jordan L., Dahesh, Samira, Moolman, Wessel J.A., Pelly, Stephen C., Nizet, Victor, Burkart, Michael D., Strauss, Erick

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Overcoming synthetic challenges in targeting coenzyme A biosynthesis with the antimicrobial natural product CJ-15,801† †Electronic supplementary information (ESI) available: Additi... von Domingo, Riyad, van der Westhuyzen, Renier, Hamann, Anton R., Mostert, Konrad J., Barnard, Leanne, Paquet, Tanya, Tjhin, Erick T., Saliba, Kevin J., van Otterlo, Willem A. L., Strauss, Erick

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Corrigendum to “Aminopyrazolo[1,5-a]pyrimidines as potential inhibitors of Mycobacterium tuberculosis: Structure activity relationships and ADME characterization” [Bioorg. Med. Che... von Soares de Melo, Candice, Feng, Tzu-Shean, van der Westhuyzen, Renier, Gessner, Richard K., Street, Leslie J., Morgans, Garreth L., Warner, Digby F., Moosa, Atica, Naran, Krupa, Lawrence, Nina, Boshoff, Helena I.M., Barry, Clifton E., Harris, C. John, Gordon, Richard, Chibale, Kelly

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The Antibiotic CJ-15,801 is an Antimetabolite which Hijacks and then Inhibits CoA Biosynthesis von van der Westhuyzen, Renier, Hammons, Justin C., Meier, Jordan L., Dahesh, Samira, Moolman, Wessel J. A., Pelly, Stephen C., Nizet, Victor, Burkart, Michael D., Strauss, Erick

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