Structure-Activity Studies on the Corticotropin Releasing Factor Antagonist Astressin, leading to a Minimal Sequence necessary for Antagonistic Activity von Rijkers, Dirk T.S, Kruijtzer, John A.W, van Oostenbrugge, Marja, Ronken, Eric, den Hartog, Jack A.J, Liskamp, Rob M.J

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A straightforward synthesis of 1,3-dichloro-5,8-dihydroisoquinoline by consecutive Stille cross-coupling and metathesis reactions von van den Hoogenband, Adri, den Hartog, Jack A.J., Faber-Hilhorst, Nancy, Lange, Jos H.M., Terpstra, Jan Willem

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An efficient synthesis of 4-bromo-N-substituted oxindoles by an intramolecular copper-catalyzed amidation reaction von van den Hoogenband, Adri, Lange, Jos H.M., den Hartog, Jack A.J., Henzen, Remco, Terpstra, Jan Willem

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An optimized solid phase synthesis strategy- including on-resin lactamization-of astressin, its retro-, inverso-, and retro-inverso isomers as corticotropin releasing factor antago... von Rijkers, Dirk T. S., den Hartog, Jack A. J., Liskamp, Rob M. J.

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Synthesis and biological activity of N-terminal lipidated and/or fluorescently labeled conjugates of astressin as corticotropin releasing factor antagonists von Rijkers, Dirk T.S., den Hartog, Jack A.J., Liskamp, Rob M.J.

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An efficient one-pot synthesis of novel 4-aryl-1-methyloxindoles von van den Hoogenband, Adri, Lange, Jos H.M., Iwema-Bakker, Wouter I., den Hartog, Jack A.J., van Schaik, Jord, Feenstra, Rolf W., Terpstra, Jan Willem

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High Target Homology Does Not Guarantee Inhibition: Aminothiazoles Emerge as Inhibitors of Plasmodium falciparum von Johannsen, Sandra, Gierse, Robin M., Krüger, Arne, Edwards, Rachel L., Nanna, Vittoria, Fontana, Anna, Zhu, Di, Masini, Tiziana, de Carvalho, Lais Pessanha, Poizat, Mael, Kieftenbelt, Bart, Hodge, Dana M., Alvarez, Sophie, Bunt, Daan, Lacour, Antoine, Shams, Atanaz, Meissner, Kamila Anna, de Souza, Edmarcia Elisa, Dröge, Melloney, van Vliet, Bernard, den Hartog, Jack, Hutter, Michael C., Held, Jana, Odom John, Audrey R., Wrenger, Carsten, Hirsch, Anna K. H.

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Solid-phase synthesis of peptidosulfonamide containing peptides derived from Leu-enkephalin von de Bont, Dries B.A, Dijkstra, Gerard D.H, den Hartog, Jack A.J, Liskamp, Rob M.J

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Design and Synthesis of an orally active GPIIb/IIIa antagonist based on a phenylpiperazine scaffold von van Maarseveen, Jan H, den Hartog, Jack A.J, Tipker, Koos, Reinders, Jan-Hendrik, Brakkee, Joost, Schön, Uwe, Kehrbach, Wolfgang, Kruse, Chris G

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A novel synthesis of N-(piperidin-4-yl)-1,3-dihydroindol-2-one via an intramolecular Pd-catalyzed amination von van den Hoogenband, Adri, den Hartog, Jack A.J., Lange, Jos H.M., Terpstra, Jan Willem

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Solid phase ring-closing metathesis: Cyclization/cleavage approach towards a seven membered cycloolefin von van Maarseveen, Jan H., den Hartog, Jack A.J., Engelen, Victor, Finner, Emil, Visser, Geb, Kruse, Chris G.

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Chemical synthesis of a messenger RNA fragment: AUGUUCUUCUUCUUCUUC von Den Hartog, Jack A. J, Wille, Gerry, Scheublin, Rolf A, Van Boom, Jacques H

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Chemical synthesis of pppA2'p5'A2'p5'A, an interferon-induced inhibitor of protein synthesis, and some functional analogs von Den Hartog, Jack A. J, Wijnands, Robert A, Van Boom, Jacques H, Crea, Roberto

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Two novel syntheses of the histamine H3 antagonist thioperamide von Lange, Jos H.M., Wals, Henri C., den Hoogenband, Adri van, de Kuilen, Aalt van, den Hartog, Jack A.J.

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Two novel syntheses of the histamine H 3 antagonist thioperamide von Lange, Jos H.M., Wals, Henri C., den Hoogenband, Adri van, de Kuilen, Aalt van, den Hartog, Jack A.J.

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An Efficient Synthesis of 4-Bromo-N-substituted Oxindoles by an Intramolecular Copper-Catalyzed Amidation Reaction von van den Hoogenband, Adri, Lange, Jos H. M., den Hartog, Jack A. J., Henzen, Remco, Terpstra, Jan Willem

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Piperazinophenyl- and piperazinophenyloxy-carboxylic acid derivatives as well as processes and intermediates for their preparation and medicaments containing these compounds von ANTEL, JOCHEN, KRUSE, C.G, BIELENBERG, GERHARD-WILHELM, ZIEGLER, DIETER, KEHRBACH, WOLFGANG, VAN MAARSEVEEN, J.H, REINDERS, JAN-HENDRIK, DEN HARTOG, JACK A.J, SCHOEN, UWE

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An Efficient One-Pot Synthesis of Novel 4-Aryl-1-methyloxindoles von van den Hoogenband, Adri, Lange, Jos H. M., Iwema-Bakker, Wouter I., den Hartog, Jack A. J., van Schaik, Jord, Feenstra, Rolf W., Terpstra, Jan Willem

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Conformational Analysis of the Nucleotides A2′‐5′A, A2′‐5′A2′‐5′A and A2′‐5′U from Nuclear Magnetic Resonance and Circular Dichroism Studies von DOORNBOS, Johannes, HARTOG, Jack A. J., BOOM, Jacques H. v., ALTONA, Cornelis

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Chemical synthesis of a messenger ribonucleic acid fragment: AUGUUCUUCUUCUUCUUC von den Hartog, J A, Wille, G, Scheublin, R A, van Boom, J H

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