Potent, orally absorbed glucagon receptor antagonists von de Laszlo, Stephen E., Hacker, Candice, Li, Bing, Kim, Dooseop, MacCoss, Malcolm, Mantlo, Nathan, Pivnichny, James V., Colwell, Larry, Koch, Gregory E., Cascieri, Margaret A., Hagmann, William K.

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Pyrroles and other heterocycles as inhibitors of P38 kinase von de Laszlo, Stephen E., Visco, Denise, Agarwal, Lily, Chang, Linda, Chin, Jayne, Croft, Gist, Forsyth, Amy, Fletcher, Daniel, Frantz, Betsy, Hacker, Candice, Hanlon, William, Harper, Coral, Kostura, Matthew, Li, Bing, Luell, Sylvie, MacCoss, Malcolm, Mantlo, Nathan, O'Neill, Edward A., Orevillo, Chad, Pang, Margaret, Parsons, Janey, Rolando, Anna, Sahly, Yousif, Sidler, Kelley, Widmer, W.Rick, O'Keefe, Stephen J.

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Substituted Imidazoles as Glucagon Receptor Antagonists von Chang, Linda L., Sidler, Kelly L., Cascieri, Margaret A., de Laszlo, Stephen, Koch, Greg, Li, Bing, MacCoss, Malcolm, Mantlo, Nathan, O'Keefe, Stephen, Pang, Margaret, Rolando, Anna, Hagmann, William K.

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Carbohydroxamido-oxazolidines: antibacterial agents that target lipid A biosynthesis von Chen, Meng-Hsin, Steiner, Mark G., de Laszlo, Stephen E., Patchett, Arthur A., Anderson, Matt S., Hyland, Sheryl A., Russell Onishi, H., Silyer, Lynn L., Raetz, Christian R.H.

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Synthesis and use of 3-amino-4-phenyl-2-piperidones and 4-amino-2-benzazepin-3-ones as conformationally restricted phenylalanine isosteres in renin inhibitors von De Laszlo, S. E, Bush, B. L, Doyle, J. J, Greenlee, W. J, Hangauer, D. G, Halgren, T. A, Lynch, R. J, Schorn, T. W, Siegl, P. K. S

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Characterization of a Novel, Non-peptidyl Antagonist of the Human Glucagon Receptor von Cascieri, M A, Koch, G E, Ber, E, Sadowski, S J, Louizides, D, de Laszlo, S E, Hacker, C, Hagmann, W K, MacCoss, M, Chicchi, G G, Vicario, P P

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The discovery of sulfonylated dipeptides as Potent VLA-4 antagonists von Hagmann, William K, Durette, Philippe L, Lanza, Thomas, Kevin, Nancy Jo, de Laszlo, Stephen E, Kopka, Ihor E, Young, David, Magriotis, Plato A, Li, Bing, Lin, Linus S, Yang, Ginger, Kamenecka, Theodore, Chang, Linda L, Wilson, Jonathan, MacCoss, Malcolm, Mills, Sander G, Van Riper, Gail, McCauley, Ermengilda, Egger, Linda A, Kidambi, Usha, Lyons, Kathryn, Vincent, Stella, Stearns, Ralph, Colletti, Adria, Teffera, Johannes, Tong, Sharon, Fenyk-Melody, Judy, Owens, Karen, Levorse, Dorothy, Kim, Philip, Schmidt, John A, Mumford, Richard A

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Deprotection of N- tert-butoxycarbonyl (Boc) groups in the presence of tert-butyl esters von Lin, Linus S, Lanza, Thomas, de Laszlo, Stephen E, Truong, Quang, Kamenecka, Theodore, Hagmann, William K

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Molecular Basis for p38 Protein Kinase Inhibitor Specificity von Lisnock, JeanMarie, Tebben, Andy, Frantz, Betsy, O'Neill, Edward A, Croft, Gist, O'Keefe, Stephen J, Li, Bing, Hacker, Candice, de Laszlo, Stephen, Smith, Anthony, Libby, Brian, Liverton, Nigel, Hermes, Jeffrey, LoGrasso, Philip

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A potent, orally active, balanced affinity angiotensin II AT1 antagonist and AT2 binding inhibitor von de Laszlo, Stephen E, Quagliato, Carol S, Greenlee, William J, Patchett, Arthur A, Chang, Raymond S. L, Lotti, Victor J, Chen, Tsing Bau, Scheck, Stacey A, Faust, Kristi A

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The selectivity of statine-based inhibitors against various human aspartic proteinases von Jupp, R A, Dunn, B M, Jacobs, J W, Vlasuk, G, Arcuri, K E, Veber, D F, Perlow, D S, Payne, L S, Boger, J, de Laszlo, S

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Molecular Basis for p38 Protein Kinase Inhibitor Specificity von Lisnock, JeanMarie, Tebben, Andy, Frantz, Betsy, O'Neill, Edward A, Croft, Gist, O'Keefe, Stephen J, Li, Bing, Hacker, Candice, de Laszlo, Stephen, Smith, Anthony, Libby, Brian, Liverton, Nigel, Hermes, Jeffrey, LoGrasso, Philip

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A nonpeptidic agonist ligand of the human C5a receptor: Synthesis, binding affinity optimization and functional characterization von de Laszlo, S.E., Allen, E.E., Li, B., Ondeyka, D., Rivero, R., Malkowitz, L., Molineaux, C., Siciliano, S.J., Springer, M.S., Greenlee, W.J., Mantlo, N.

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Amidines as amide bond replacements in VLA-4 antagonists von KAMENECKA, Theodore M, PARK, You-Jung, WEI TANG, COLLETTI, Adria, TEFFERA, Yohannes, STEARNS, Ralph, MACCOSS, Malcolm, SCHMIDT, John A, HAGMANN, William K, LIN, Linus S, DE LASZLO, Stephen, MCCAULEY, Ermengilda D, VAN RIPER, Gail, EGGER, Linda, KIDAMBI, Usha, MUMFORD, Richard A, TONG, Sharon

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AT1/AT2-BALANCED ANGIOTENSIN II ANTAGONISTS von Ashton, Wallace T., Chang, Linda L., Flanagan, Kelly L., Mantlo, Nathan B., Ondeyka, Debra L., Kim, Dooseop, de Laszlo, Stephen E., Glinka, Tomasz W., Rivero, Ralph A., Kevin, Nancy J., Chang, Raymond S.L., Siegl, Peter K.S., Kivlighn, Salah D., Greenlee, William J.

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Acute hypotensive responses to peptide inhibitors of renin in conscious monkeys: an effect on blood pressure independent of plasma renin inhibition von SCHAFFER, L. W, SCHORN, T. W, SIEGL, P. K. S, WINQUIST, R. J, STROUSE, J. F, PAYNE, L, CHAKRAVARTY, P. K, DE LASZLO, S. E, TENBROEKE, J, VEBER, D. F, GREENLEE, W. J

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N-Tetrahydrofuroyl-( l)-phenylalanine derivatives as potent VLA-4 antagonists von Yang, Ginger X., Chang, Linda L., Truong, Quang, Doherty, George A., Magriotis, Plato A., de Laszlo, Stephen E., Li, Bing, MacCoss, Malcolm, Kidambi, Usha, Egger, Linda A., McCauley, Ermengilda, Van Riper, Gail, Mumford, Richard A., Schmidt, John A., Hagmann, William K.

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N-(3-Phenylsulfonyl-3-piperidinoyl)-phenylalanine derivatives as potent, selective VLA-4 antagonists von Gutteridge, Clare E, de Laszlo, Stephen E, Kamenecka, Theodore M, McCauley, Ermengilda, van Riper, Gail, Mumford, Richard A, Kidambi, Usha, Egger, Linda A, Tong, Sharon, Hagmann, William K

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Identification of Unique VLA-4 Antagonists from a Combinatorial Library von de Laszlo, Stephen E., Li, Bing, McCauley, Ermengilda, Van Riper, Gail, Hagmann, William K.

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N-Aryl-prolyl-dipeptides as potent antagonists of VLA-4 von Kamenecka, Theodore M., Lanza, Jr, Thomas, de Laszlo, Stephen E., Li, Bing, McCauley, Ermengilda D., Van Riper, Gail, Egger, Linda A., Kidambi, Usha, Mumford, Richard A., Tong, Sharon, MacCoss, Malcolm, Schmidt, John A., Hagmann, William K.

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