Opioids activate brain analgesic circuits through cytochrome P450/epoxygenase signaling von Ding, Xinxin, Hough, Lindsay B, Conroy, Jennie L, Fang, Cheng, Gu, Jun, Zeitlin, Scott O, Yang, Weizhu, Yang, Jun, VanAlstine, Melissa A, Nalwalk, Julia W, Albrecht, Phillip J, Mazurkiewicz, Joseph E, Snyder-Keller, Abigail, Shan, Zhixing, Zhang, Shao-Zhong, Wentland, Mark P, Behr, Melissa, Knapp, Brian I, Bidlack, Jean M, Zuiderveld, Obbe P, Leurs, Rob

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Non-imidazole histamine H 3 ligands. Part III. New 4- n-propylpiperazines as non-imidazole histamine H 3-antagonists von Walczyński, Krzysztof, Zuiderveld, Obbe P., Timmerman, Henk

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N -Substituted Piperidinyl Alkyl Imidazoles:  Discovery of Methimepip as a Potent and Selective Histamine H 3 Receptor Agonist von Kitbunnadaj, Ruengwit, Hashimoto, Takeshi, Poli, Enzo, Zuiderveld, Obbe P., Menozzi, Alessandro, Hidaka, Ryoko, de Esch, Iwan J. P., Bakker, Remko A., Menge, Wiro M. P. B., Yamatodani, Atsushi, Coruzzi, Gabriella, Timmerman, Henk, Leurs, Rob

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Identification of 4-(1 H -Imidazol-4(5)-ylmethyl)pyridine (Immethridine) as a Novel, Potent, and Highly Selective Histamine H 3 Receptor Agonist von Kitbunnadaj, Ruengwit, Zuiderveld, Obbe P., Christophe, Bernard, Hulscher, Saskia, Menge, Wiro M. P. B., Gelens, Edith, Snip, Erwin, Bakker, Remko A., Celanire, Sylvain, Gillard, Michel, Talaga, Patrice, Timmerman, Henk, Leurs, Rob

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A Selective Human H 4 -Receptor Agonist:  (−)-2-Cyano-1-methyl-3-{(2 R ,5 R )-5- [1 H -imidazol-4(5)-yl]tetrahydrofuran-2-yl}methylguanidine von Hashimoto, Takeshi, Harusawa, Shinya, Araki, Lisa, Zuiderveld, Obbe P., Smit, Martine J., Imazu, Tomonari, Takashima, Seiichiroh, Yamamoto, Yumiko, Sakamoto, Yasuhiko, Kurihara, Takushi, Leurs, Rob, Bakker, Remko A., Yamatodani, Atsushi

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8R-Lisuride Is a Potent Stereospecific Histamine H1-Receptor Partial Agonist von Bakker, R.A., Weiner, D.M., ter Laak, T., Beuming, T., Zuiderveld, O.P., Edelbroek, M., Hacksell, U., Timmerman, H., Brann, M.R., Leurs, R.

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Synthesis and Structure−Activity Relationships of Conformationally Constrained Histamine H 3 Receptor Agonists von Kitbunnadaj, Ruengwit, Zuiderveld, Obbe P., De Esch, Iwan J. P., Vollinga, Roeland C., Bakker, Remko, Lutz, Martin, Spek, Anthony L., Cavoy, Emile, Deltent, Marie-France, Menge, Wiro M. P. B., Timmerman, Henk, Leurs, Rob

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Characterization of the Binding Site of the Histamine H 3 Receptor. 1. Various Approaches to the Synthesis of 2-(1 H -Imidazol-4-yl)cyclopropylamine and Histaminergic Activity of (... von De Esch, Iwan J. P., Vollinga, Roeland C., Goubitz, Kees, Schenk, Henk, Appelberg, Ulf, Hacksell, Uli, Lemstra, Sylvia, Zuiderveld, Obbe P., Hoffmann, Marcel, Leurs, Rob, Menge, Wiro M. P. B., Timmerman, Henk

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Pharmacological characterisation of the histamine H 3 receptor in the rat hippocampus von Alves-Rodrigues, Alexandra, Timmerman, Henk, Willems, Edwin, Lemstra, Sylvia, Zuiderveld, Obbe P, Leurs, Rob

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Synthesis and pharmacological evaluation of some amino-acid-containing cyproheptadine derivatives as dual antagonists of histamine H 1- and leukotriene D 4-receptors von Zhang, MQ, van de Stolpe, A, Zuiderveld, OP, Timmerman, H

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Synthesis and pharmacological evaluation of some amino-acid-containing cyproheptadine derivatives as dual antagonists of histamine H1- and leukotriene D4-receptors von Zhang, MQ, van de Stolpe, A, Zuiderveld, OP, Timmerman, H

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Screening of cattle urine samples for the presence of beta-agonists with a functional test : some preliminary results von SCHILT, R, HOOIJERINK, H, HUF, F. A, ZUIDERVELD, O. P, BAST, A

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Histamine H 1 receptor ligands : Part I. Novel thiazol-4-ylethanamine derivatives: synthesis and in vitro pharmacology von Walczyński, K., Timmerman, H., Zuiderveld, O.P., Zhang, M.Q., Glinka, R.

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Histamine H 1 receptor ligands : Part II. Synthesis and in vitro pharmacology of 2-[2-(phenylamino)thiazol-4-yl]ethanamine and 2-(2-benzhydrylthiazol-4-yl)ethanamine derivatives von Walczyński, Krzysztof, Guryn, Roman, Zuiderveld, Obbe P, Zhang, Ming-Qiang, Timmerman, Henk

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Effect of inhibitors of enkephalin degradation in the isolated guinea-pig ileum von van Amsterdam, Jan G.C., van Buuren, Karel J.H., Krielaart, Marco J., Zuiderveld, Obbe P., Tijms, Rob P.J.H.

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Non-imidazole histamine H 3 ligands. Part I. Synthesis of 2-(1-piperazinyl)- and 2-(hexahydro-1 H-1,4-diazepin-1-yl)benzothiazole derivatives as H 3-antagonists with H 1 blocking a... von Walczyński, Krzysztof, Guryn, Roman, Zuiderveld, Obbe P., Timmerman, Henk

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