Design, Synthesis and Biological Characterization of Histone Deacetylase 8 (HDAC8) Proteolysis Targeting Chimeras (PROTACs) with Anti-Neuroblastoma Activity von Darwish, Salma, Ghazy, Ehab, Heimburg, Tino, Herp, Daniel, Zeyen, Patrik, Salem-Altintas, Rabia, Ridinger, Johannes, Robaa, Dina, Schmidtkunz, Karin, Erdmann, Frank, Schmidt, Matthias, Romier, Christophe, Jung, Manfred, Oehme, Ina, Sippl, Wolfgang

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Binding Free Energy (BFE) Calculations and Quantitative Structure-Activity Relationship (QSAR) Analysis of Schistosoma mansoni Histone Deacetylase 8 (smHDAC8) Inhibitors von Simoben, Conrad V., Ghazy, Ehab, Zeyen, Patrik, Darwish, Salma, Schmidt, Matthias, Romier, Christophe, Robaa, Dina, Sippl, Wolfgang

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Synthesis, Molecular Docking and Biological Characterization of Pyrazine Linked 2-Aminobenzamides as New Class I Selective Histone Deacetylase (HDAC) Inhibitors with Anti-Leukemic... von Ibrahim, Hany S, Abdelsalam, Mohamed, Zeyn, Yanira, Zessin, Matthes, Mustafa, Al-Hassan M, Fischer, Marten A, Zeyen, Patrik, Sun, Ping, Bülbül, Emre F, Vecchio, Anita, Erdmann, Frank, Schmidt, Matthias, Robaa, Dina, Barinka, Cyril, Romier, Christophe, Schutkowski, Mike, Krämer, Oliver H, Sippl, Wolfgang

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The potential for histone deacetylase (HDAC) inhibitors as cestocidal drugs von Vaca, Hugo R., Celentano, Ana M., Agustina Toscanini, Maria, Heimburg, Tino, Ghazy, Ehab, Zeyen, Patrik, Hauser, Alexander-Thomas, Oliveira, Guilherme, Elissondo, Maria C., Jung, Manfred, Sippl, Wolfgang, Camicia, Federico, Cecilia Rosenzvit, Mara

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Structure-Based Design and Biological Characterization of Selective Histone Deacetylase 8 (HDAC8) Inhibitors with Anti-Neuroblastoma Activity von Heimburg, Tino, Kolbinger, Fiona R, Zeyen, Patrik, Ghazy, Ehab, Herp, Daniel, Schmidtkunz, Karin, Melesina, Jelena, Shaik, Tajith Baba, Erdmann, Frank, Schmidt, Matthias, Romier, Christophe, Robaa, Dina, Witt, Olaf, Oehme, Ina, Jung, Manfred, Sippl, Wolfgang

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Design, synthesis, and biological evaluation of dual targeting inhibitors of histone deacetylase 6/8 and bromodomain BRPF1 von Ghazy, Ehab, Zeyen, Patrik, Herp, Daniel, Hügle, Martin, Schmidtkunz, Karin, Erdmann, Frank, Robaa, Dina, Schmidt, Matthias, Morales, Elizabeth R., Romier, Christophe, Günther, Stefan, Jung, Manfred, Sippl, Wolfgang

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Identification of histone deacetylase 10 (HDAC10) inhibitors that modulate autophagy in transformed cells von Zeyen, Patrik, Zeyn, Yanira, Herp, Daniel, Mahmoudi, Fereshteh, Yesiloglu, Talha Z., Erdmann, Frank, Schmidt, Matthias, Robaa, Dina, Romier, Christophe, Ridinger, Johannes, Herbst-Gervasoni, Corey J., Christianson, David W., Oehme, Ina, Jung, Manfred, Krämer, Oliver H., Sippl, Wolfgang

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Synthesis, structure-activity relationships, cocrystallization and cellular characterization of novel smHDAC8 inhibitors for the treatment of schistosomiasis von Ghazy, Ehab, Heimburg, Tino, Lancelot, Julien, Zeyen, Patrik, Schmidtkunz, Karin, Truhn, Anne, Darwish, Salma, Simoben, Conrad V., Shaik, Tajith B., Erdmann, Frank, Schmidt, Matthias, Robaa, Dina, Romier, Christophe, Jung, Manfred, Pierce, Raymond, Sippl, Wolfgang

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The potential for histone deacetylase von Heimburg, Tino, Oliveira, Guilherme, Celentano, Ana María, Ghazy, Ehab, Zeyen, Patrik, Hauser, Alexander-Thomas, Camicia, Federico, Toscanini, María Agustina, Vaca, Hugo Rolando, Sippl, Wolfgang, Jung, Manfred, Elissondo, María Celina, Rosenzvit, Mara Cecilia

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