Discovery of Conformationally Constrained ALK2 Inhibitors von González-Álvarez, Héctor, Ensan, Deeba, Xin, Tao, Wong, Jong Fu, Zepeda-Velázquez, Carlos A., Cros, Julien, Sweeney, Melissa N., Hoffer, Laurent, Kiyota, Taira, Wilson, Brian J., Aman, Ahmed, Roberts, Owen, Isaac, Methvin B., Bullock, Alex N., Smil, David, Al-awar, Rima

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Discovery of Small-Molecule Antagonists of the PWWP Domain of NSD2 von Ferreira de Freitas, Renato, Liu, Yanli, Szewczyk, Magdalena M, Mehta, Naimee, Li, Fengling, McLeod, David, Zepeda-Velázquez, Carlos, Dilworth, David, Hanley, Ronan P, Gibson, Elisa, Brown, Peter J, Al-Awar, Rima, James, Lindsey I, Arrowsmith, Cheryl H, Barsyte-Lovejoy, Dalia, Min, Jinrong, Vedadi, Masoud, Schapira, Matthieu, Allali-Hassani, Abdellah

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Targeting ALK2: An Open Science Approach to Developing Therapeutics for the Treatment of Diffuse Intrinsic Pontine Glioma von Ensan, Deeba, Smil, David, Zepeda-Velázquez, Carlos A, Panagopoulos, Dimitrios, Wong, Jong Fu, Williams, Eleanor P, Adamson, Roslin, Bullock, Alex N, Kiyota, Taira, Aman, Ahmed, Roberts, Owen G, Edwards, Aled M, O’Meara, Jeff A, Isaac, Methvin B, Al-awar, Rima

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Structure-Based Optimization of a Small Molecule Antagonist of the Interaction Between WD Repeat-Containing Protein 5 (WDR5) and Mixed-Lineage Leukemia 1 (MLL1) von Getlik, Matthäus, Smil, David, Zepeda-Velázquez, Carlos, Bolshan, Yuri, Poda, Gennady, Wu, Hong, Dong, Aiping, Kuznetsova, Ekaterina, Marcellus, Richard, Senisterra, Guillermo, Dombrovski, Ludmila, Hajian, Taraneh, Kiyota, Taira, Schapira, Matthieu, Arrowsmith, Cheryl H, Brown, Peter J, Vedadi, Masoud, Al-awar, Rima

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A First-in-Class, Highly Selective and Cell-Active Allosteric Inhibitor of Protein Arginine Methyltransferase 6 von Shen, Yudao, Li, Fengling, Szewczyk, Magdalena M, Halabelian, Levon, Chau, Irene, Eram, Mohammad S, Dela Seña, Carlo, Park, Kwang-Su, Meng, Fanye, Chen, He, Zeng, Hong, McLeod, David, Zepeda-Velázquez, Carlos A, Campbell, Robert M, Mader, Mary M, Watson, Brian M, Schapira, Matthieu, Arrowsmith, Cheryl H, Al-Awar, Rima, Barsyte-Lovejoy, Dalia, Kaniskan, H. Ümit, Brown, Peter J, Vedadi, Masoud, Jin, Jian

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Enantioselective Organocatalytic Michael/Aldol Sequence: Anticancer Natural Product (+)-trans-Dihydrolycoricidine von McNulty, James, Zepeda-Velázquez, Carlos

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Correction to "Structure-Activity Relationship of USP5 Inhibitors" von Mann, Mandeep K, Zepeda-Velázquez, Carlos A, González-Álvarez, Héctor, Dong, Aiping, Kiyota, Taira, Aman, Ahmed M, Loppnau, Peter, Li, Yanjun, Wilson, Brian, Arrowsmith, Cheryl H, Al-Awar, Rima, Harding, Rachel J, Schapira, Matthieu

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Structure–Activity Relationship of USP5 Inhibitors von Mann, Mandeep K, Zepeda-Velázquez, Carlos A, González-Álvarez, Héctor, Dong, Aiping, Kiyota, Taira, Aman, Ahmed M, Loppnau, Peter, Li, Yanjun, Wilson, Brian, Arrowsmith, Cheryl H, Al-Awar, Rima, Harding, Rachel J, Schapira, Matthieu

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A chemical biology toolbox to study protein methyltransferases and epigenetic signaling von Scheer, Sebastian, Ackloo, Suzanne, Medina, Tiago S., Schapira, Matthieu, Li, Fengling, Ward, Jennifer A., Lewis, Andrew M., Northrop, Jeffrey P., Richardson, Paul L., Kaniskan, H. Ümit, Shen, Yudao, Liu, Jing, Smil, David, McLeod, David, Zepeda-Velazquez, Carlos A., Luo, Minkui, Jin, Jian, Barsyte-Lovejoy, Dalia, Huber, Kilian V. M., De Carvalho, Daniel D., Vedadi, Masoud, Zaph, Colby, Brown, Peter J., Arrowsmith, Cheryl H.

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iPSC Neuronal Assay Identifies Amaryllidaceae Pharmacophore with Multiple Effects against Herpesvirus Infections von McNulty, James, D’Aiuto, Leonardo, Zhi, Yun, McClain, Lora, Zepeda-Velázquez, Carlos, Ler, Spencer, Jenkins, Hilary A, Yee, Michael B, Piazza, Paolo, Yolken, Robert H, Kinchington, Paul R, Nimgaonkar, Vishwajit L

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Total Synthesis of the Natural Product (+)‐trans‐Dihydronarciclasine via an Asymmetric Organocatalytic [3+3]‐Cycloaddition and discovery of its potent anti‐Zika Virus (ZIKV) Activi... von Revu, Omkar, Zepeda‐Velázquez, Carlos, Nielsen, Alex J., McNulty, James, Yolken, Robert H., Jones‐Brando, Lorraine

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A non-traditional crystal-based compound screening method targeting the ATP binding site of Plasmodium falciparum GRP78 for identification of novel nucleoside analogues von Mrozek, Alexander, Antoshchenko, Tetyana, Chen, Yun, Zepeda-Velázquez, Carlos, Smil, David, Kumar, Nirbhay, Lu, Hua, Park, Hee-Won

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Development of a robust reagent for the two-carbon homologation of aldehydes to (E)-α,β-unsaturated aldehydes in water von MCNULTY, James, ZEPEDA-VELAZQUEZ, Carlos, MCLEOD, David

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Enantioselective Organocatalytic Michael/Aldol Sequence: Anticancer Natural Product (+)-trans-Dihydrolycoricidine von McNulty, James, Zepeda-Velázquez, Carlos

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Truncated ring-A amaryllidaceae alkaloid modulates the host cell integrated stress response, exhibiting antiviral activity to HSV-1 and SARSCoV-2 von McNulty, James, Babu-Dokuburra, Chanti, Scattolon, Jon, Zepeda-Velazquez, Carlos, Wesesky, Maribeth A., Caldwell, Jill K., Zheng, Wenxiao, Milosevic, Jadranka, Kinchington, Paul R., Bloom, David C., Nimgaonkar, Vishwajit L., D’Aiuto, Leonardo

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Development of a robust reagent for the two-carbon homologation of aldehydes to (E)-α,β-unsaturated aldehydes in waterElectronic supplementary information (ESI) available: Full exp... von McNulty, James, Zepeda-Velázquez, Carlos, McLeod, David

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The synthesis of densely functionalised α-acyloxy enaminals and enaminones via a novel homogeneous silver(i) catalysed rearrangement von Keskar, Kunal, Zepeda-Velazquez, Carlos, Dokuburra, Chanti Babu, Jenkins, Hilary A, McNulty, James

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ChemInform Abstract: Enantioselective Organocatalytic Michael/Aldol Sequence: Anticancer Natural Product (+)-trans-Dihydrolycoricidine von McNulty, James, Zepeda-Velazquez, Carlos

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ChemInform Abstract: Development of a Robust Reagent for the Two-Carbon Homologation of Aldehydes to (E)-α,β-Unsaturated Aldehydes in Water von McNulty, James, Zepeda-Velazquez, Carlos, McLeod, David

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ChemInform Abstract: Wittig Reactions of Trialkylphosphine-Derived Ylides: New Directions and Applications in Organic Synthesis von McNulty, James, McLeod, David, Das, Priyabrata, Zepeda-Velazquez, Carlos

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