Discovery of Cycloalkyl[c]thiophenes as Novel Scaffolds for Hypoxia-Inducible Factor-2α Inhibitors von Buchstaller, Hans-Peter, Sala-Hojman, Ada, Leiendecker, Matthias, Albers, Joachim, Anlauf, Uwe, Berges, Nina, Dong, Liming, Fuchß, Thomas, Germann, Martina, Knehans, Tim, Krier, Mireille, Lecomte, Marc, Müller, Daniel, Müller, Sandra R., Leuthner, Birgitta, Lindemann, Ralph, Musil, Djordje, Nowak, Mateusz, Reither, Vivian, Rettig, Corinna, Schindler, Christina E. M., Pakulska, Urszula, Spuck, Dieter, Wegener, Ansgar, Zarębski, Adrian

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Novel method of measurement of in vitro drug uptake in OATP1B3 overexpressing cells in the presence of dextran von Kowal-Chwast, Anna, Gabor-Worwa, Ewelina, Gaud, Nilesh, Gogola, Dawid, Piątek, Agnieszka, Zarębski, Adrian, Littlewood, Peter, Smoluch, Marek, Brzózka, Krzysztof, Kuś, Kamil

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Synthesis of amide and sulfonamide substituted N-aryl 6-aminoquinoxalines as PFKFB3 inhibitors with improved physicochemical properties von Boutard, Nicolas, Białas, Arkadiusz, Sabiniarz, Aleksandra, Guzik, Paweł, Banaszak, Katarzyna, Biela, Artur, Bień, Marcin, Buda, Anna, Bugaj, Barbara, Cieluch, Ewelina, Cierpich, Anna, Dudek, Łukasz, Eggenweiler, Hans-Michael, Fogt, Joanna, Gaik, Monika, Gondela, Andrzej, Jakubiec, Krzysztof, Jurzak, Mirek, Kitlińska, Agata, Kowalczyk, Piotr, Kujawa, Maciej, Kwiecińska, Katarzyna, Leś, Marcin, Lindemann, Ralph, Maciuszek, Monika, Mikulski, Maciej, Niedziejko, Paulina, Obara, Alicja, Pawlik, Henryk, Rzymski, Tomasz, Sieprawska-Lupa, Magdalena, Sowińska, Marta, Szeremeta-Spisak, Joanna, Stachowicz, Agata, Tomczyk, Mateusz M., Wiklik, Katarzyna, Włoszczak, Łukasz, Ziemiańska, Sylwia, Zarębski, Adrian, Brzózka, Krzysztof, Nowak, Mateusz, Fabritius, Charles-Henry

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5-Keto-3-cyano-2,4-diaminothiophenes as selective maternal embryonic leucine zipper kinase inhibitors von Boutard, Nicolas, Sabiniarz, Aleksandra, Czerwińska, Klaudia, Jarosz, Małgorzata, Cierpich, Anna, Kolasińska, Ewa, Wiklik, Katarzyna, Gluza, Karolina, Commandeur, Claude, Buda, Anna, Stasiowska, Agata, Bobowska, Aneta, Galek, Mariusz, Fabritius, Charles-Henry, Bugaj, Marta, Palacz, Edyta, Mazan, Andrzej, Zarębski, Adrian, Krawczyńska, Karolina, Żurawska, Małgorzata, Zawadzki, Przemysław, Milik, Mariusz, Węgrzyn, Paulina, Dobrzańska, Monika, Brzózka, Krzysztof, Kowalczyk, Piotr

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Identification of changes in the transcriptome profile of human hepatoma HepG2 cells stimulated with interleukin-1 beta von Jura, Jolanta, Węgrzyn, Paulina, Zarębski, Adrian, Władyka, Benedykt, Koj, Aleksander

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Gene transfer of CuZn superoxide dismutase enhances the synthesis of vascular endothelial growth factor von Grzenkowicz-Wydra, Jolanta, Cisowski, Jarosław, Nakonieczna, Joanna, Zarebski, Adrian, Udilova, Natalia, Nohl, Hans, Józkowicz, Alicja, Podhajska, Anna, Dulak, Józef

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A search for genes modulated by interleukin-6 alone or with interleukin-1β in HepG2 cells using differential display analysis von Węgrzyn, Paulina, Jura, Jolanta, Kupiec, Tomasz, Piekoszewski, Wojciech, Władyka, Benedykt, Zarębski, Adrian, Koj, Aleksander

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Discovery and Structure–Activity Relationships of N‐Aryl 6‐Aminoquinoxalines as Potent PFKFB3 Kinase Inhibitors von Boutard, Nicolas, Białas, Arkadiusz, Sabiniarz, Aleksandra, Guzik, Paweł, Banaszak, Katarzyna, Biela, Artur, Bień, Marcin, Buda, Anna, Bugaj, Barbara, Cieluch, Ewelina, Cierpich, Anna, Dudek, Łukasz, Eggenweiler, Hans‐Michael, Fogt, Joanna, Gaik, Monika, Gondela, Andrzej, Jakubiec, Krzysztof, Jurzak, Mirek, Kitlińska, Agata, Kowalczyk, Piotr, Kujawa, Maciej, Kwiecińska, Katarzyna, Leś, Marcin, Lindemann, Ralph, Maciuszek, Monika, Mikulski, Maciej, Niedziejko, Paulina, Obara, Alicja, Pawlik, Henryk, Rzymski, Tomasz, Sieprawska‐Lupa, Magdalena, Sowińska, Marta, Szeremeta‐Spisak, Joanna, Stachowicz, Agata, Tomczyk, Mateusz M., Wiklik, Katarzyna, Włoszczak, Łukasz, Ziemiańska, Sylwia, Zarębski, Adrian, Brzózka, Krzysztof, Nowak, Mateusz, Fabritius, Charles‐Henry

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Regulatory feedback loop between NF-κB and MCP-1-induced protein 1 RNase von Skalniak, Lukasz, Mizgalska, Danuta, Zarebski, Adrian, Wyrzykowska, Paulina, Koj, Aleksander, Jura, Jolanta

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Gfi1 Coordinates Epigenetic Repression of p21Cip/WAF1 by Recruitment of Histone Lysine Methyltransferase G9a and Histone Deacetylase 1 von Duan, Zhijun, Zarebski, Adrian, Montoya-Durango, Diego, Grimes, H Leighton, Horwitz, Marshall

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Abstract A49: Repression of tumor survival pathways by novel, selective inhibitors of MNK1 and MNK2 kinases von Rzymski, Tomasz, Dreas, Agnieszka, Milik, Mariusz, Kucwaj, Katarzyna, Zarebski, Adrian, Skuta, Malgorzata Szajewska, Cierpich, Anna, Fabritius, Charles, Brzozka, Krzysztof

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Mutations in Growth Factor Independent-1 Associated with Human Neutropenia Block Murine Granulopoiesis through Colony Stimulating Factor-1 von Zarebski, Adrian, Velu, Chinavenmeni S., Baktula, Avinash M., Bourdeau, Tristan, Horman, Shane R., Basu, Sudeep, Bertolone, Salvatore J., Horwitz, Marshal, Hildeman, David A., Trent, John O., Grimes, H. Leighton

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Abstract 2160: Development of selective MELK kinase inhibitors for cancer treatments von Kowalczyk, Piotr, Wegrzyn, Paulina, Zawadzki, Przemyslaw, Palacz, Edyta, Trebacz, Ewa, Wiklik, Katarzyna, Milik, Mariusz, Zarebski, Adrian, Krawczynska, Karolina, Brzózka, Krzysztof

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Abstract 755: Repression of tumor survival pathways by novel and selective inhibitors of MNK1 and MNK2 kinases in glioblastoma and colorectal cancer von Rzymski, Tomasz, Szajewska-Skuta, Malgorzata, Zarebski, Adrian, Sitarz, Kamil, Sapala, Lukasz, Zurawska, Malgorzata, Salwinska, Magdalena, Windak, Renata, Trebacz, Ewa, Daniel-Wojcik, Joanna, Obuchowicz, Radoslaw, Winnik, Bozena, Wincza, Ewelina, Kulesza, Urszula, Kucwaj-Borysz, Katarzyna, Milik, Mariusz, Dreas, Agnieszka, Brzozka, Krzysztof

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Targeting kinases hyperphosphorylating tau protein: Elucidation of kinase inhibition profile most efficient in restoring physiological tau phosphorylation von Nowak, Mateusz, Fabritius, Charles-Henry, Zarebski, Adrian, Guratowska, Monika, Windak, Renata

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P4–424: Targeting kinases hyperphosphorylating tau protein: Elucidation of kinase inhibition profile most efficient in restoring physiological tau phosphorylation von Nowak, Mateusz, Fabritius, Charles‐Henry, Zarebski, Adrian, Guratowska, Monika, Windak, Renata

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Abstract 3845: Antitumor activity of SEL120: An orally available dual inhibitors of Haspin/CDK9, for standalone and combination therapy with AuroraB inhibitors in solid tumors and... von Rzymski, Tomasz, Zarebski, Adrian, Windak, Renata, Sibinska, Zaneta, Klosowska-Wardega, Agnieszka, Trebacz, Ewa, Cholody, Marek, Szamborska-Gbur, Agnieszka, Milik, Mariusz, Prymula, Katarzyna, Brzozka, Krzysztof, Beuzen, Nicolas

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Abstract 4499: In vitro and in vivo evaluation of novel Pim kinase inhibitors with potent anticancer activity von Brzozka, Krzysztof, Zarebski, Adrian, Trebacz, Ewa, Czardybon, Wojciech, Chołody, Marek, Beuzen, Nicolas

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Regulatory feedback loop between NF-[kappa]B and MCP-1-induced protein 1 RNase von Skalniak, Lukasz, Mizgalska, Danuta, Zarebski, Adrian, Wyrzykowska, Paulina, Koj, Aleksander, Jura, Jolanta

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Abstract A242: Identification of novel and specific Pim-1 kinase inhibitors with potent anticancer activity in hematological and solid tumor malignancies von Brzozka, Krzysztof, Czardybon, Wojciech, Kaczorowska, Katarzyna, Zarebski, Adrian, Smagur, Jan, Beuzen, Nicolas

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