Synthesis of Acrylamides via the Doebner–Knoevenagel Condensation von Zacuto, Michael J

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Nickel/Photoredox-Catalyzed Methylation of (Hetero)aryl Chlorides Using Trimethyl Orthoformate as a Methyl Radical Source von Kariofillis, Stavros K, Shields, Benjamin J, Tekle-Smith, Makeda A, Zacuto, Michael J, Doyle, Abigail G

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Mild, Redox‐Neutral Formylation of Aryl Chlorides through the Photocatalytic Generation of Chlorine Radicals von Nielsen, Matthew K., Shields, Benjamin J., Liu, Junyi, Williams, Michael J., Zacuto, Michael J., Doyle, Abigail G.

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A Quantitative Assay of Sodium Triacetoxyborohydride von Zacuto, Michael J, Perona, Joseph, Dunn, Robert

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Asymmetric Synthesis of Highly Functionalized Tetrahydropyran DPP‑4 Inhibitor von Xu, Feng, Zacuto, Michael J, Kohmura, Yoshinori, Rosen, Jon, Gibb, Andrew, Alam, Mahbub, Scott, Jeremy, Tschaen, David

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One-Step RhCl3-Catalyzed Deprotection of Acyclic N-Allyl Amides von Zacuto, Michael J, Xu, Feng

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Synthesis of the HCV Protease Inhibitor Vaniprevir (MK-7009) Using Ring-Closing Metathesis Strategy von Kong, Jongrock, Chen, Cheng-yi, Balsells-Padros, Jaume, Cao, Yang, Dunn, Robert F, Dolman, Sarah J, Janey, Jacob, Li, Hongmei, Zacuto, Michael J

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Evolution of a Manufacturing Route to Omarigliptin, A Long-Acting DPP‑4 Inhibitor for the Treatment of Type 2 Diabetes von Chung, John Y. L, Scott, Jeremy P, Anderson, Camille, Bishop, Brian, Bremeyer, Nadine, Cao, Yang, Chen, Qinghao, Dunn, Robert, Kassim, Amude, Lieberman, David, Moment, Aaron J, Sheen, Faye, Zacuto, Michael

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One-Step Synthesis of 1‑Chloro-3-arylacetone Derivatives from Arylacetic Acids von Zacuto, Michael J, Dunn, Robert F, Figus, Margaret

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Chemoselectivity of the Ru-Catalyzed Cycloisomerization Reaction for the Synthesis of Dihydropyrans; Application to the Synthesis of l-Forosamine von Zacuto, Michael J, Tomita, Daisuke, Pirzada, Zainab, Xu, Feng

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Asymmetric Synthesis of Telcagepant, a CGRP Receptor Antagonist for the Treatment of Migraine von Xu, Feng, Zacuto, Michael, Yoshikawa, Naoki, Desmond, Richard, Hoerrner, Scott, Itoh, Tetsuji, Journet, Michel, Humphrey, Guy R, Cowden, Cameron, Strotman, Neil, Devine, Paul

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Two Approaches to the Chemical Development and Large-Scale Preparation of a Pyrimidyl Tetrazole Intermediate von Mullens, Peter, Cleator, Ed, McLaughlin, Mark, Bishop, Brian, Edwards, John, Goodyear, Adrian, Andreani, Teresa, Jin, Yan, Kong, Jongrock, Li, Hongmei, Williams, Michael, Zacuto, Michael

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Preparation of 4-Allylisoindoline via a Kumada Coupling with Allylmagnesium Chloride von Zacuto, Michael J, Shultz, C. Scott, Journet, Michel

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Tandem Silylformylation−Crotylsilylation/Tamao Oxidation of Internal Alkynes: A Remarkable Example of Generating Complexity from Simplicity von Spletstoser, Jared T, Zacuto, Michael J, Leighton, James L

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Divergent Synthesis of Complex Polyketide-Like Macrolides from a Simple Polyol Fragment von Zacuto, Michael J, Leighton, James L

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Tandem Intramolecular Silylformylation−Crotylsilylation:  Highly Efficient Synthesis of Polyketide Fragments von Zacuto, Michael J, O'Malle, Steven J, Leighton, James L

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Chirality Control in the Kilogram-Scale Manufacture of Single-Enantiomer CELMoDs: Synthesis of Iberdomide·BSA, Part 2 von Zacuto, Michael J., Traverse, John F., Geherty, Maryll E., Bostwick, Kirsten F., Jordan, Christopher, Zhang, Chengmin

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Mild, Redox‐Neutral Formylation of Aryl Chlorides through the Photocatalytic Generation of Chlorine Radicals von Nielsen, Matthew K., Shields, Benjamin J., Liu, Junyi, Williams, Michael J., Zacuto, Michael J., Doyle, Abigail G.

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Copper-Catalyzed Addition of Alcohols to Carbodiimides: Oxygen as an Accelerant von Wells, Lucille A., Gau, Michael R., Peddicord, Michael B., Bostwick, Kirsten F., Kozlowski, Marisa C., Zacuto, Michael J.

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Process Development and Kilogram-Scale Manufacture of Key Intermediates toward Single-Enantiomer CELMoDs: Synthesis of Iberdomide·BSA, Part 1 von Zacuto, Michael J., Traverse, John F., Bostwick, Kirsten F., Geherty, Maryll E., Primer, David N., Zhang, Weihong, Zhang, Chengmin, Janes, Rachel D., Marton, Christopher

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