Discovery and optimization of a series of quinazolinone-derived antagonists of CXCR3 von Johnson, Michael, Li, An-Rong, Liu, Jiwen, Fu, Zice, Zhu, Liusheng, Miao, Shichang, Wang, Xuemei, Xu, Qingge, Huang, Alan, Marcus, Andrew, Xu, Feng, Ebsworth, Karen, Sablan, Emmanuel, Danao, Jay, Kumer, Jeff, Dairaghi, Dan, Lawrence, Chris, Sullivan, Tim, Tonn, George, Schall, Thomas, Collins, Tassie, Medina, Julio

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Potent and Orally Bioavailable GPR142 Agonists as Novel Insulin Secretagogues for the Treatment of Type 2 Diabetes von Toda, Narihiro, Hao, Xiaolin, Ogawa, Yasuyuki, Oda, Kozo, Yu, Ming, Fu, Zice, Chen, Yi, Kim, Yongjae, Lizarzaburu, Mike, Lively, Sarah, Lawlis, Shauna, Murakoshi, Michiko, Nara, Futoshi, Watanabe, Nobuaki, Reagan, Jeff D, Tian, Hui, Fu, Angela, Motani, Alykhan, Liu, Qingxiang, Lin, Yi-Jyun, Zhuang, Run, Xiong, Yumei, Fan, Peter, Medina, Julio, Li, Leping, Izumi, Masanori, Okuyama, Ryo, Shibuya, Satoshi

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Optimization of a series of quinazolinone-derived antagonists of CXCR3 von Liu, Jiwen, Fu, Zice, Li, An-Rong, Johnson, Michael, Zhu, Liusheng, Marcus, Andrew, Danao, Jay, Sullivan, Tim, Tonn, George, Collins, Tassie, Medina, Julio

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Discovery of potent and specific CXCR3 antagonists von Chen, Xiaoqi, Mihalic, Jeff, Deignan, Jeff, Gustin, Darin J., Duquette, Jason, Du, Xiaohui, Chan, Johann, Fu, Zice, Johnson, Michael, Li, An-Rong, Henne, Kirk, Sullivan, Tim, Lemon, Bryan, Ma, Ji, Miao, Shichang, Tonn, George, Collins, Tassie, Medina, Julio C.

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Discovery and optimization of CRTH2 and DP dual antagonists von Liu, Jiwen, Fu, Zice, Wang, Yingcai, Schmitt, Mike, Huang, Alan, Marshall, Derek, Tonn, George, Seitz, Lisa, Sullivan, Tim, Lucy Tang, H., Collins, Tassie, Medina, Julio

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Optimization of the heterocyclic core of the quinazolinone-derived CXCR3 antagonists von Li, An-Rong, Johnson, Michael G., Liu, Jiwen, Chen, Xiaoqi, Du, Xiaohui, Mihalic, Jeffrey T., Deignan, Jeffrey, Gustin, Darin J., Duquette, Jason, Fu, Zice, Zhu, Liusheng, Marcus, Andrew P., Bergeron, Phillipe, McGee, Lawrence R., Danao, Jay, Lemon, Bryan, Carabeo, Teresa, Sullivan, Timothy, Ma, Ji, Tang, Liang, Tonn, George, Collins, Tassie L., Medina, Julio C.

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Optimization of phenylacetic acid derivatives for CRTH2 and DP selective antagonism von Wang, Yingcai, Fu, Zice, Schmitt, Michael, Wang, Xuemei, Shen, Wang, Rickel, Erika, Martin, Tod, Budelsky, Alison, Marshall, Derek, Collins, Tassie, Tang, H. Lucy, Medina, Julio C., Liu, Jiwen (Jim)

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Discovery of AMG 853, a CRTH2 and DP Dual Antagonist von Liu, Jiwen, Li, An-Rong, Wang, Yingcai, Johnson, Mike G, Su, Yongli, Shen, Wang, Wang, Xuemei, Lively, Sarah, Brown, Matthew, Lai, SuJen, Gonzalez Lopez De Turiso, Felix, Xu, Qingge, Van Lengerich, Bettina, Schmitt, Mike, Fu, Zice, Sun, Ying, Lawlis, Shanna, Seitz, Lisa, Danao, Jay, Wait, Jill, Ye, Qiuping, Tang, Hua Lucy, Grillo, Mark, Collins, Tassie L, Sullivan, Timothy J, Medina, Julio C

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Structure-Guided Design, Synthesis, and Evaluation of Guanine-Derived Inhibitors of the eIF4E mRNA–Cap Interaction von Chen, Xiaoqi, Kopecky, David J, Mihalic, Jeff, Jeffries, Shawn, Min, Xiaoshan, Heath, Julie, Deignan, Jeff, Lai, SuJen, Fu, Zice, Guimaraes, Cristiano, Shen, Shanling, Li, Shyun, Johnstone, Sheree, Thibault, Stephen, Xu, Haoda, Cardozo, Mario, Shen, Wang, Walker, Nigel, Kayser, Frank, Wang, Zhulun

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Phenylalanine derivatives as GPR142 agonists for the treatment of Type II diabetes von Du, Xiaohui, Kim, Yong-Jae, Lai, SuJen, Chen, Xi, Lizarzaburu, Mike, Turcotte, Simon, Fu, Zice, Liu, Qingxiang, Zhang, Ying, Motani, Alykhan, Oda, Kozo, Okuyama, Ryo, Nara, Futoshi, Murakoshi, Michiko, Fu, Angela, Reagan, Jeff D., Fan, Peter, Xiong, Yumei, Shen, Wang, Li, Leping, Houze, Jonathan, Medina, Julio C.

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Synthesis of medium-sized rings using the intramolecular Pauson–Khand reaction von Krafft, Marie E, Fu, Zice, Boñaga, Llorente Vicente R

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Synthesis of benzimidazoles from 1,1-dibromoethenes von Shen, Wang, Kohn, Todd, Fu, Zice, Jiao, XianYun, Lai, Sujen, Schmitt, Michael

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Chiral P,N-Ligands Based on Ketopinic Acid in the Asymmetric Heck Reaction von Gilbertson, Scott R, Fu, Zice

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5‑Alkyl-2-urea-Substituted Pyridines: Identification of Efficacious Glucokinase Activators with Improved Properties von Kohn, Todd J, Du, Xiaohui, Lai, SuJen, Xiong, YuMei, Komorowski, Renee, Veniant, Murielle, Fu, Zice, Jiao, Xianyun, Pattaropong, Vatee, Chow, David, Cardozo, Mario, Jin, Lixia, Conn, Marion, DeWolf, Walter E, Kraser, Christopher F, Hinklin, Ronald J, Boys, Mark L, Medina, Julio C, Houze, Jonathan, Dransfield, Paul, Coward, Peter

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Novel Series of Potent Glucokinase Activators Leading to the Discovery of AM-2394 von Dransfield, Paul J, Pattaropong, Vatee, Lai, Sujen, Fu, Zice, Kohn, Todd J, Du, Xiaohui, Cheng, Alan, Xiong, Yumei, Komorowski, Renee, Jin, Lixia, Conn, Marion, Tien, Eric, DeWolf, Walter E, Hinklin, Ronald J, Aicher, Thomas D, Kraser, Christopher F, Boyd, Steven A, Voegtli, Walter C, Condroski, Kevin R, Veniant-Ellison, Murielle, Medina, Julio C, Houze, Jonathan, Coward, Peter

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C5-Alkyl-2-methylurea-Substituted Pyridines as a New Class of Glucokinase Activators von Du, Xiaohui, Hinklin, Ronald J, Xiong, Yumei, Dransfield, Paul, Park, Jaehyeon, Kohn, Todd J, Pattaropong, Vatee, Lai, SuJen, Fu, Zice, Jiao, Xianyun, Chow, David, Jin, Lixia, Davda, Jasmine, Veniant, Murielle M, Anderson, Deborah A, Baer, Brian R, Bencsik, Josef R, Boyd, Steven A, Chicarelli, Mark Joseph, Mohr, Peter J, Wang, Bin, Condroski, Kevin R, DeWolf, Walter E, Conn, Marion, Tran, Thanhvien, Yang, Jerry, Aicher, Thomas D, Medina, Julio C, Coward, Peter, Houze, Jonathan B

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Aminopyrazole–Phenylalanine Based GPR142 Agonists: Discovery of Tool Compound and in Vivo Efficacy Studies von Yu, Ming, Lizarzaburu, Mike, Motani, Alykhan, Fu, Zice, Du, Xiaohui, Liu, Jiwen (Jim), Jiao, Xianyun, Lai, SuJen, Fan, Peter, Fu, Angela, Liu, Qingxiang, Murakoshi, Michiko, Nara, Futoshi, Oda, Kozo, Okuyama, Ryo, Reagan, Jeff D, Watanabe, Nobuaki, Yamazaki, Mami, Xiong, Yumei, Zhang, Ying, Zhuang, Run, Lin, Daniel C.-H, Houze, Jonathan B, Medina, Julio C, Li, Leping

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Corrigendum to “Phenylalanine derivatives as GPR142 agonists for the treatment of Type II diabetes” [Bioorg. Med. Chem. Lett. 22 (2012) 6218–6223] von Du, Xiaohui, Kim, Yong-Jae, Lai, SuJen, Chen, Xi, Lizarzaburu, Mike, Turcotte, Simon, Fu, Zice, Liu, Qingxiang, Zhang, Ying, Motani, Alykhan, Oda, Kozo, Okuyama, Ryo, Nara, Futoshi, Murakoshi, Michiko, Fu, Angela, Reagan, Jeff D., Fan, Peter, Xiong, Yumei, Shen, Wang, Li, Leping, Houze, Jonathan, Medina, Julio C.

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Proline-Based P, N Ligands in Asymmetric Allylation and the Heck Reaction von Gilbertson, Scott R, Xie, Dejian, Fu, Zice

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Palladium-catalyzed synthesis of vinyl phosphines from ketones von Gilbertson, Scott R., Fu, Zice, Starkey, Gale W.

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