In silico, in vitro, X-ray crystallography, and integrated strategies for discovering spermidine synthase inhibitors for Chagas disease von Yoshino, Ryunosuke, Yasuo, Nobuaki, Hagiwara, Yohsuke, Ishida, Takashi, Inaoka, Daniel Ken, Amano, Yasushi, Tateishi, Yukihiro, Ohno, Kazuki, Namatame, Ichiji, Niimi, Tatsuya, Orita, Masaya, Kita, Kiyoshi, Akiyama, Yutaka, Sekijima, Masakazu

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NMR Biochemical Assay for Oxidosqualene Cyclase: Evaluation of Inhibitor Activities on Trypanosoma cruzi and Human Enzymes von Tani, Osamu, Akutsu, Yukie, Ito, Shinji, Suzuki, Takayuki, Tateishi, Yukihiro, Yamaguchi, Tomohiko, Niimi, Tatsuya, Namatame, Ichiji, Chiba, Yasunori, Sakashita, Hitoshi, Kubota, Tomomi, Yanagi, Tetsuo, Mizukami, Shusaku, Hirayama, Kenji, Furukawa, Koji, Yamasaki, Kazuhiko

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Correction to NMR Biochemical Assay for Oxidosqualene Cyclase: Evaluation of Inhibitor Activities on Trypanosoma cruzi and Human Enzymes von Tani, Osamu, Akutsu, Yukie, Ito, Shinji, Suzuki, Takayuki, Tateishi, Yukihiro, Yamaguchi, Tomohiko, Niimi, Tatsuya, Namatame, Ichiji, Chiba, Yasunori, Sakashita, Hitoshi, Kubota, Tomomi, Yanagi, Tetsuo, Mizukami, Shusaku, Hirayama, Kenji, Furukawa, Koji, Yamasaki, Kazuhiko

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Molecular Basis for SUMOylation-dependent Regulation of DNA Binding Activity of Heat Shock Factor 2 von Tateishi, Yukihiro, Ariyoshi, Mariko, Igarashi, Ryuji, Hara, Hideyuki, Mizuguchi, Kenji, Seto, Azusa, Nakai, Akira, Kokubo, Tetsuro, Tochio, Hidehito, Shirakawa, Masahiro

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The structure of the third intracellular loop of the muscarinic acetylcholine receptor M2 subtype von Ichiyama, Susumu, Oka, Yoshiaki, Haga, Kazuko, Kojima, Shuichi, Tateishi, Yukihiro, Shirakawa, Masahiro, Haga, Tatsuya

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Structural analysis of pituitary adenylate cyclase-activating polypeptides bound to phospholipid membranes by magic angle spinning solid-state NMR von Komi, Nobuyasu, Okawa, Kayo, Tateishi, Yukihiro, Shirakawa, Masahiro, Fujiwara, Toshimichi, Akutsu, Hideo

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Structure-based drug design of 1,3,5-triazine and pyrimidine derivatives as novel FGFR3 inhibitors with high selectivity over VEGFR2 von Kuriwaki, Ikumi, Kameda, Minoru, Hisamichi, Hiroyuki, Kikuchi, Shigetoshi, Iikubo, Kazuhiko, Kawamoto, Yuichiro, Moritomo, Hiroyuki, Kondoh, Yutaka, Amano, Yasushi, Tateishi, Yukihiro, Echizen, Yuka, Iwai, Yoshinori, Noda, Atsushi, Tomiyama, Hiroshi, Suzuki, Tomoyuki, Hirano, Masaaki

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Structural insights into the novel inhibition mechanism of Trypanosoma cruzi spermidine synthase von Amano, Yasushi, Namatame, Ichiji, Tateishi, Yukihiro, Honboh, Kazuya, Tanabe, Eiki, Niimi, Tatsuya, Sakashita, Hitoshi

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Synthesis and structure-activity relationships of pyrimidine derivatives as potent and orally active FGFR3 inhibitors with both increased systemic exposure and enhanced in vitro po... von Kuriwaki, Ikumi, Kameda, Minoru, Iikubo, Kazuhiko, Hisamichi, Hiroyuki, Kawamoto, Yuichiro, Kikuchi, Shigetoshi, Moritomo, Hiroyuki, Kondoh, Yutaka, Terasaka, Tadashi, Amano, Yasushi, Tateishi, Yukihiro, Echizen, Yuka, Iwai, Yoshinori, Noda, Atsushi, Tomiyama, Hiroshi, Nakazawa, Taisuke, Hirano, Masaaki

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An NMR Biochemical Assay for Fragment-Based Drug Discovery: Evaluation of an Inhibitor Activity on Spermidine Synthase of Trypanosoma cruzi von Yamasaki, Kazuhiko, Tani, Osamu, Tateishi, Yukihiro, Tanabe, Eiki, Namatame, Ichiji, Niimi, Tatsuya, Furukawa, Koji, Sakashita, Hitoshi

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High-throughput construction method for expression vector of peptides for NMR study suited for isotopic labeling von Tenno, Takeshi, Goda, Natsuko, Tateishi, Yukihiro, Tochio, Hidehito, Mishima, Masaki, Hayashi, Hidenori, Shirakawa, Masahiro, Hiroaki, Hidekazu

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Discovery of a Hidden Trypanosoma cruzi Spermidine Synthase Binding Site and Inhibitors through In Silico, In Vitro, and X‑ray Crystallography von Yoshino, Ryunosuke, Yasuo, Nobuaki, Hagiwara, Yohsuke, Ishida, Takashi, Inaoka, Daniel Ken, Amano, Yasushi, Tateishi, Yukihiro, Ohno, Kazuki, Namatame, Ichiji, Niimi, Tatsuya, Orita, Masaya, Kita, Kiyoshi, Akiyama, Yutaka, Sekijima, Masakazu

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The structure of the third intracellular loop of the muscarinic acetylcholine receptor M 2 subtype von Ichiyama, Susumu, Oka, Yoshiaki, Haga, Kazuko, Kojima, Shuichi, Tateishi, Yukihiro, Shirakawa, Masahiro, Haga, Tatsuya

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3P-091 Molecular basis for SUMOylation-dependent regulation of DNA binding activity of Heat Shock Factor 2(Nucleic acid binding proteins,The 47th Annual Meeting of the Biophysical... von Ariyoshi, Mariko, Tateishi, yukihiro, Igarashi, Ryuji, Hara, Hideyuki, Mizuguchi, Kenji, Tochio, Hidehito, Shirakawa, Masahiro

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3P-091 SUMO化による転写調節因子heat shock factor 2のDNA結合阻害の分子機構(核酸結合蛋白質,第47回日本生物物理学会年会)

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P-05-04 Fragment Evolution identified novel inhibitors of Trypanosoma cruzi Spermidine synthase von YASUSHI AMANO, Ichiji Namatame, Yukihiro Tateishi, Kazuya Honbou, Eiki Tanabe, Yohsuke Hagiwara, Shinji Ito, Masashi Imanishi, Tatsuya Niimi, Hitoshi Sakashita, Kazuhiko Yamasaki, Tomomi Kubota, Osamu Tani, Koji Furukawa

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Pathological prognostic factors predicting lymph node metastasis in submucosal invasive (T1) colorectal carcinoma von Tateishi, Yoko, Nakanishi, Yukihiro, Taniguchi, Hirokazu, Shimoda, Tadakazu, Umemura, Satoshi

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Sensory neurons that respond to sex and aggregation pheromones in the nymphal cockroach von Tateishi, Kosuke, Nishimura, Yukihiro, Sakuma, Masayuki, Yokohari, Fumio, Watanabe, Hidehiro

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A Case of Varicella Zoster Virus Encephalitis with Advanced Human Immunodeficiency Virus Disease Diagnosed by Brain Biopsy von Yoshimura, Yukihiro, Nakase, Dai, So, Yuna, Miyata, Nobuyuki, Takahashi, Kenta, Katano, Harutaka, Chiba, Sawako, Tateishi, Yoko

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DOCK2 is involved in the host genetics and biology of severe COVID-19 von Namkoong, Ho, Shirai, Yuya, Okuzaki, Daisuke, Wang, Qingbo S., Ishihara, Rino, Hamamoto, Junko, Shimizu, Eigo, Morita, Takayoshi, Naito, Toshio, Okamori, Satoshi, Takano, Kenji, Takaku, Yotaro, Tada, Ai, Miyawaki, Masayoshi, Kawana, Masatoshi, Honda, Takayuki, Tateishi, Tomoya, Saito, Ryuichi, Sado, Toshikatsu, Kimura, Tomoki, Yoshiyama, Takashi, Arakawa, Kenichi, Yoshida, Shuichi, Mitamura, Keiko, Uchida, Tomoyuki, Konishi, Shunichiro, Nakachi, Ichiro, Murakami, Koji, Sano, Hirohito, Baba, Hiroaki, Namba, Shinichi, Kawamura, Yusuke, Kuge, Tomoki, Matsumoto, Kinnosuke, Takemoto, Norihiko, Eguchi, Hirotaka, Fukusumi, Takahito, Inohara, Hidenori, Takeda, Yoshito, Shinozuka, Keisuke, Shoko, Tomohisa, Kojima, Mitsuaki, Adachi, Tomohiro, Miyazawa, Naoki, Sado, Reiko, Kawashima, Hidetoshi, Sekikawa, Yoshiyuki, Nishi, Koichi, Tani, Mayuko, Suzuki, Junya, Nakatsumi, Hiroki, Ogura, Takashi, Fukui, Yasutaka, Makino, Yasushi, Yagi, Kazuma, Fuke, Satoshi, Saito, Hiroshi, Tsuchida, Tomoya, Morikawa, Daiki, Takata, Tohru, Odani, Toshio, Shichinohe, Yasuo, Koshida, Kiyoshi, Hayashi, Kentaro, Hiranuma, Hisato, Nagata, Kaoru, Ueda, Ken, Hanada, Satoko, Kawamura, Kodai, Nishiyama, Kenta, Hashimoto, Naozumi, Maeda, Shunsuke, Ono, Hiroshi, Shibusawa, Takayuki, Masuda, Makoto, Ohba, Takehiko, Eriguchi, Yoshihiro, Yonekawa, Akiko, Kan-o, Keiko, Kanaoka, Kensuke, Inoue, Yoshiaki, Kai, Hirayasu, Hida, Naoya, Takada, Minoru, Ogura, Shinji, Togashi, Yuki, Ogata, Tomouki, Nishiyama, Kei, Ooshima, Nobuharu, Watanabe, Masafumi, Tanaka, Akihiko, Tanino, Yoshinori, Minemura, Hiroyuki, Tominaga, Yoshiteru, Utsugi, Mitsuyoshi, Saito, Yoshinobu, Kumanogoh, Atsushi, Hasegawa, Naoki, Kanai, Takanori, Fukunaga, Koichi

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