Effect of Ligand Structure on the Zinc-Catalyzed Henry Reaction. Asymmetric Syntheses of (−)-Denopamine and (−)-Arbutamine von Trost, Barry M, Yeh, Vince S. C, Ito, Hisanako, Bremeyer, Nadine

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Recent advances in the total syntheses of oxazole-containing natural products von Yeh, Vince S.C.

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A Dinuclear Zn Catalyst for the Asymmetric Nitroaldol (Henry) Reaction von Trost, Barry M., Yeh, Vince S. C.

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Total Synthesis of the Marine Alkaloid Halichlorine: Development and Use of a General Route to Chiral Piperidines von Liu, Dazhan, Acharya, Hukum P, Yu, Maolin, Wang, Jian, Yeh, Vince S. C, Kang, Shunzhen, Chiruta, Chandramouli, Jachak, Santosh M, Clive, Derrick L. J

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Stereocontrolled Synthesis of (+)-Boronolide von Trost, Barry M, Yeh, Vince S. C

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Synthetic Chemistry of Halichlorine and the Pinnaic Acids von Clive, Derrick L. J, Yu, Maolin, Wang, Jian, Yeh, Vince S. C, Kang, Shunzhen

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Utilizing Chemical Genomics to Identify Cytochrome b as a Novel Drug Target for Chagas Disease von Khare, Shilpi, Roach, Steven L, Barnes, S Whitney, Hoepfner, Dominic, Walker, John R, Chatterjee, Arnab K, Neitz, R Jeffrey, Arkin, Michelle R, McNamara, Case W, Ballard, Jaime, Lai, Yin, Fu, Yue, Molteni, Valentina, Yeh, Vince, McKerrow, James H, Glynne, Richard J, Supek, Frantisek

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Identification and Preliminary Characterization of a Potent, Safe, and Orally Efficacious Inhibitor of Acyl-CoA:Diacylglycerol Acyltransferase 1 von Yeh, Vince S. C, Beno, David W. A, Brodjian, Sevan, Brune, Michael E, Cullen, Steven C, Dayton, Brian D, Dhaon, Madhup K, Falls, Hugh D, Gao, Ju, Grihalde, Nelson, Hajduk, Philip, Hansen, T. Matthew, Judd, Andrew S, King, Andrew J, Klix, Russel C, Larson, Kelly J, Lau, Yau Y, Marsh, Kennan C, Mittelstadt, Scott W, Plata, Dan, Rozema, Michael J, Segreti, Jason A, Stoner, Eric J, Voorbach, Martin J, Wang, Xiaojun, Xin, Xili, Zhao, Gang, Collins, Christine A, Cox, Bryan F, Reilly, Regina M, Kym, Philip R, Souers, Andrew J

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Synthesis and structural activity relationship of 11β-HSD1 inhibitors with novel adamantane replacements von Yeh, Vince S.C., Kurukulasuriya, Ravi, Madar, David, Patel, Jyoti R., Fung, Steven, Monzon, Katina, Chiou, William, Wang, Jiahong, Jacobson, Peer, Sham, Hing L., Link, J.T.

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Practical Cu-catalyzed amination of functionalized heteroaryl halides von Yeh, Vince S.C., Wiedeman, Paul E.

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Synthesis and biological evaluation of heterocycle containing adamantane 11β-HSD1 inhibitors von Yeh, Vince S.C., Patel, Jyoti R., Yong, Hong, Kurukulasuriya, Ravi, Fung, Steven, Monzon, Katina, Chiou, William, Wang, Jiahong, Stolarik, Deanne, Imade, Hovis, Beno, David, Brune, Michael, Jacobson, Peer, Sham, Hing, Link, J.T.

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Discovery of orally active butyrolactam 11β-HSD1 inhibitors von Yeh, Vince S.C., Kurukulasuriya, Ravi, Fung, Steven, Monzon, Katina, Chiou, William, Wang, Jiahong, Stolarik, Deanne, Imade, Hovis, Shapiro, Robin, Knourek-Segel, Victoria, Bush, Eugene, Wilcox, Denise, Nguyen, Phong T., Brune, Michael, Jacobson, Peer, Link, J.T.

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A Highly Efficient Synthesis of Potent and Selective Butyrolactam Inhibitors of 11β-Hsd1 von Yeh, Vince S. C, Kurukulasuriya, Ravi, Kerdesky, Francis A

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Proteasome inhibition for treatment of leishmaniasis, Chagas disease and sleeping sickness von Khare, Shilpi, Nagle, Advait S., Biggart, Agnes, Lai, Yin H., Liang, Fang, Davis, Lauren C., Barnes, S. Whitney, Mathison, Casey J. N., Myburgh, Elmarie, Gao, Mu-Yun, Gillespie, J. Robert, Liu, Xianzhong, Tan, Jocelyn L., Stinson, Monique, Rivera, Ianne C., Ballard, Jaime, Yeh, Vince, Groessl, Todd, Federe, Glenn, Koh, Hazel X. Y., Venable, John D., Bursulaya, Badry, Shapiro, Michael, Mishra, Pranab K., Spraggon, Glen, Brock, Ansgar, Mottram, Jeremy C., Buckner, Frederick S., Rao, Srinivasa P. S., Wen, Ben G., Walker, John R., Tuntland, Tove, Molteni, Valentina, Glynne, Richard J., Supek, Frantisek

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Antitrypanosomal Treatment with Benznidazole Is Superior to Posaconazole Regimens in Mouse Models of Chagas Disease von Khare, Shilpi, Liu, Xianzhong, Stinson, Monique, Rivera, Ianne, Groessl, Todd, Tuntland, Tove, Yeh, Vince, Wen, Ben, Molteni, Valentina, Glynne, Richard, Supek, Frantisek

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Discovery and Characterization of Clinical Candidate LXE408 as a Kinetoplastid-Selective Proteasome Inhibitor for the Treatment of Leishmaniases von Nagle, Advait, Biggart, Agnes, Be, Celine, Srinivas, Honnappa, Hein, Andreas, Caridha, Diana, Sciotti, Richard J, Pybus, Brandon, Kreishman-Deitrick, Mara, Bursulaya, Badry, Lai, Yin H, Gao, Mu-Yun, Liang, Fang, Mathison, Casey J. N, Liu, Xiaodong, Yeh, Vince, Smith, Jeffrey, Lerario, Isabelle, Xie, Yongping, Chianelli, Donatella, Gibney, Michael, Berman, Ashley, Chen, Yen-Liang, Jiricek, Jan, Davis, Lauren C, Liu, Xianzhong, Ballard, Jaime, Khare, Shilpi, Eggimann, Fabian Kurt, Luneau, Alexandre, Groessl, Todd, Shapiro, Michael, Richmond, Wendy, Johnson, Kevin, Rudewicz, Patrick J, Rao, Srinivasa P. S, Thompson, Christopher, Tuntland, Tove, Spraggon, Glen, Glynne, Richard J, Supek, Frantisek, Wiesmann, Christian, Molteni, Valentina

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Synthesis of a 6-azaspiro[4.5]decane related to halichlorine and the pinnaic acids von Clive, Derrick L.J., Yeh, Vince S.C.

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Optimization of Platelet-Derived Growth Factor Receptor (PDGFR) Inhibitors for Duration of Action, as an Inhaled Therapy for Lung Remodeling in Pulmonary Arterial Hypertension von Shaw, Duncan E, Baig, Ferheen, Bruce, Ian, Chamoin, Sylvie, Collingwood, Stephen P, Cross, Sarah, Dayal, Satish, Drückes, Peter, Furet, Pascal, Furminger, Vikki, Haggart, Deborah, Hussey, Martin, Konstantinova, Irena, Loren, Jon C, Molteni, Valentina, Roberts, Sonia, Reilly, John, Saunders, Alex M, Stringer, Rowan, Sviridenko, Lilya, Thomas, Matthew, Thomson, Christopher G, Tomlins, Christine, Wen, Ben, Yeh, Vince, Pearce, Andrew C

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Lead Identification to Clinical Candidate Selection: Drugs for Chagas Disease von Neitz, R. Jeffrey, Chen, Steven, Supek, Frantisek, Yeh, Vince, Kellar, Danielle, Gut, Jiri, Bryant, Clifford, Gallardo-Godoy, Alejandra, Molteni, Valentina, Roach, Steven L., Chatterjee, Arnab K., Robertson, Stephanie, Renslo, Adam R., Arkin, Michelle, Glynne, Richard, McKerrow, James, Siqueira-Neto, Jair L.

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Utilizing Chemical Genomics to Identify Cytochrome b as a Novel Drug Target for Chagas Disease: e1005058 von Khare, Shilpi, Roach, Steven L, Barnes, S Whitney, Hoepfner, Dominic, Walker, John R, Chatterjee, Arnab K, Neitz, R Jeffrey, Arkin, Michelle R, McNamara, Case W, Ballard, Jaime, Lai, Yin, Fu, Yue, Molteni, Valentina, Yeh, Vince, McKerrow, James H, Glynne, Richard J, Supek, Frantisek

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