Structural evidence for the roles of divalent cations in actin polymerization and activation of ATP hydrolysis von Scipion, Clement P. M., Ghoshdastider, Umesh, Ferrer, Fernando J., Yuen, Tsz-Ying, Wongsantichon, Jantana, Robinson, Robert C.

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Total Synthesis of 7′,8′-Dihydroaigialospirol von Yuen, Tsz-Ying, Brimble, Margaret A

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Total Synthesis of Paecilospirone von Yuen, Tsz-Ying, Yang, Sung-Hyun, Brimble, Margaret A.

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A Maillard Approach to 2-Formylpyrroles: Synthesis of Magnolamide, Lobechine and Funebral von Yuen, Tsz-Ying, Eaton, Samantha E., Woods, Tom M., Furkert, Daniel P., Choi, Ka Wai, Brimble, Margaret A.

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Synthetic approaches to [5,6]-benzannulated spiroketal natural products von McLeod, Michael C., Brimble, Margaret A., Rathwell, Dominea C. K., Wilson, Zoe E., Yuen, Tsz-Ying

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Stapled β‑Hairpin Antimicrobial Peptides with Improved Stability and Activity against Drug-Resistant Gram-Negative Bacteria von Selvarajan, Vanitha, Tram, Nhan D. T., Xu, Jian, Ngen, Sarah T. Y., Koh, Jun-Jie, Teo, Jeanette W. P., Yuen, Tsz-Ying, Ee, Pui Lai Rachel

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Design-rules for stapled peptides with in vivo activity and their application to Mdm2/X antagonists von Chandramohan, Arun, Josien, Hubert, Yuen, Tsz Ying, Duggal, Ruchia, Spiegelberg, Diana, Yan, Lin, Juang, Yu-Chi Angela, Ge, Lan, Aronica, Pietro G., Kaan, Hung Yi Kristal, Lim, Yee Hwee, Peier, Andrea, Sherborne, Brad, Hochman, Jerome, Lin, Songnian, Biswas, Kaustav, Nestor, Marika, Verma, Chandra S., Lane, David P., Sawyer, Tomi K., Garbaccio, Robert, Henry, Brian, Kannan, Srinivasaraghavan, Brown, Christopher J., Johannes, Charles W., Partridge, Anthony W.

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Incorporation of Putative Helix-Breaking Amino Acids in the Design of Novel Stapled Peptides: Exploring Biophysical and Cellular Permeability Properties von Partridge, Anthony W, Kaan, Hung Yi Kristal, Juang, Yu-Chi, Sadruddin, Ahmad, Lim, Shuhui, Brown, Christopher J, Ng, Simon, Thean, Dawn, Ferrer, Fernando, Johannes, Charles, Yuen, Tsz Ying, Kannan, Srinivasaraghavan, Aronica, Pietro, Tan, Yaw Sing, Pradhan, Mohan R, Verma, Chandra S, Hochman, Jerome, Chen, Shiying, Wan, Hui, Ha, Sookhee, Sherborne, Brad, Lane, David P, Sawyer, Tomi K

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Receptor Activity-modifying Proteins 2 and 3 Generate Adrenomedullin Receptor Subtypes with Distinct Molecular Properties von Watkins, Harriet A., Chakravarthy, Madhuri, Abhayawardana, Rekhati S., Gingell, Joseph J., Garelja, Michael, Pardamwar, Meenakshi, McElhinney, James M.W.R., Lathbridge, Alex, Constantine, Arran, Harris, Paul W.R., Yuen, Tsz-Ying, Brimble, Margaret A., Barwell, James, Poyner, David R., Woolley, Michael J., Conner, Alex C., Pioszak, Augen A., Reynolds, Christopher A., Hay, Debbie L.

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Stereoisomerism of stapled peptide inhibitors of the p53-Mdm2 interaction: an assessment of synthetic strategies and activity profiles von Yuen, Tsz Ying, Brown, Christopher J, Xue, Yuezhen, Tan, Yaw Sing, Ferrer Gago, Fernando J, Lee, Xue Er, Neo, Jin Yong, Thean, Dawn, Kaan, Hung Yi Kristal, Partridge, Anthony W, Verma, Chandra S, Lane, David P, Johannes, Charles W

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De-risking Drug Discovery of Intracellular Targeting Peptides: Screening Strategies to Eliminate False-Positive Hits von Ng, Simon, Juang, Yu-Chi, Chandramohan, Arun, Kaan, Hung Yi Kristal, Sadruddin, Ahmad, Yuen, Tsz Ying, Ferrer-Gago, Fernando J, Lee, Xue’Er Cheryl, Liew, Xi, Johannes, Charles W, Brown, Christopher J, Kannan, Srinivasaraghavan, Aronica, Pietro G, Berglund, Nils A, Verma, Chandra S, Liu, Lijuan, Stoeck, Alexander, Sawyer, Tomi K, Partridge, Anthony W, Lane, David P

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De Novo Sequencing of Synthetic Bis-cysteine Peptide Macrocycles Enabled by “Chemical Linearization” of Compound Mixtures von Chen, Zhi’ang, Lim, Yi Wee, Neo, Jin Yong, Ting Chan, Rachel Shu, Koh, Li Quan, Yuen, Tsz Ying, Lim, Yee Hwee, Johannes, Charles W., Gates, Zachary P.

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Total Synthesis of Paecilospirone von Yuen, Tsz-Ying, Yang, Sung-Hyun, Brimble, Margaret A.

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Synthesis of Chiral Alkenyl Cyclopropane Amino Acids for Incorporation into Stapled Peptides von Yuen, Tsz Ying, Brown, Christopher J, Tan, Yaw Sing, Johannes, Charles W

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Design-Rules for Stapled Alpha-Helical Peptides with On-Target In Vivo Activity: Application to Mdm2/X dual antagonists von Chandramohan, Arun, Josien, Hubert, Yuen, Tsz Ying, Duggal, Ruchia, Spiegelberg, Diana, Yan, Lin, Angela Juang, Yu-Chi, Ge, Lan, Aronica, Pietro, Kaan, Kristal, Lim, Yee Hwee, Peier, Andrea, Sherborne, Brad, Hochman, Jerome, Lin, Songnian, Biswas, Kaustav, Henry, Brian, Nestor, Marika, Verma, Chandra S, Lane, David, Sawyer, Tomi, Garbaccio, Robert, Kannan, Srinivasaraghavan, Brown, Christopher J., Johannes, Charles W, Partridge, Anthony William

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Macrocyclic α helical peptide therapeutic modality: A perspective of learnings and challenges von Sawyer, Tomi K., Partridge, Anthony W., Kaan, Hung Yi Kristal, Juang, Yu-Chi, Lim, Shuhui, Johannes, Charles, Yuen, Tsz Ying, Verma, Chandra, Kannan, Srinivasaraghavan, Aronica, Pietro, Tan, Yaw Sing, Sherborne, Brad, Ha, Sookhee, Hochman, Jerome, Chen, Shiying, Surdi, Laura, Peier, Andrea, Sauvagnat, Berengere, Dandliker, Peter J., Brown, Christopher J., Ng, Simon, Ferrer, Fernando, Lane, David P.

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NanoClick: A High Throughput, Target-Agnostic Peptide Cell Permeability Assay von Peier, Andrea, Ge, Lan, Boyer, Nicolas, Frost, John, Duggal, Ruchia, Biswas, Kaustav, Edmondson, Scott, Hermes, Jeffrey D, Yan, Lin, Zimprich, Chad, Sadruddin, Ahmad, Kristal Kaan, Hung Yi, Chandramohan, Arun, Brown, Christopher J, Thean, Dawn, Lee, Xue Er, Yuen, Tsz Ying, Ferrer-Gago, Fernando J, Johannes, Charles W, Lane, David P, Sherborne, Brad, Corona, Cesear, Robers, Matthew B, Sawyer, Tomi K, Partridge, Anthony W

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Liposome Click Membrane Permeability Assay for Identifying Permeable Peptides von Desai, Tanvi J., Habulihaz, Bahanu, Cannon, Joe R., Chandramohan, Arun, Kaan, Hung Yi Kristal, Sadruddin, Ahmad, Yuen, Tsz Ying, Johannes, Charles, Thean, Dawn, Brown, Chris J., Lane, David P., Partridge, Anthony W., Evers, Raymond, Sawyer, Tomi K., Hochman, Jerome

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Macrocyclization of an all- d linear α-helical peptide imparts cellular permeability von Kannan, Srinivasaraghavan, Aronica, Pietro G. A., Ng, Simon, Gek Lian, Dawn Thean, Frosi, Yuri, Chee, Sharon, Shimin, Jiang, Yuen, Tsz Ying, Sadruddin, Ahmad, Kaan, Hung Yi Kristal, Chandramohan, Arun, Wong, Jin Huei, Tan, Yaw Sing, Chang, Zi Wei, Ferrer-Gago, Fernando J., Arumugam, Prakash, Han, Yi, Chen, Shiying, Rénia, Laurent, Brown, Christopher J., Johannes, Charles W., Henry, Brian, Lane, David P., Sawyer, Tomi K., Verma, Chandra S., Partridge, Anthony W.

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Granzyme B PET Imaging of Combined Chemotherapy and Immune Checkpoint Inhibitor Therapy in Colon Cancer von Goggi, Julian L, Hartimath, Siddesh V, Xuan, Tan Yun, Khanapur, Shivashankar, Jieu, Beverly, Chin, Hui Xian, Ramasamy, Boominathan, Cheng, Peter, Rong, Tang Jun, Fong, Yong Fui, Yuen, Tsz Ying, Msallam, Rasha, Chacko, Ann-Marie, Renia, Laurent, Johannes, Charles, Hwang, You Yi, Robins, Edward G

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