C4-Alkylamination of C4-Halo-1H-1-tritylpyrazoles Using Pd(dba)2 or CuI von Usami, Yoshihide, Tatsui, Yuya, Yoneyama, Hiroki, Harusawa, Shinya

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Syntheses of cyclopentyl nucleoside (−)-neplanocin A through tetrazole-fragmentation from cyanophosphates von Yoneyama, Hiroki, Uemura, Kenji, Usami, Yoshihide, Harusawa, Shinya

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Synthesis of five-membered unsaturated compounds from ketones via cyanophosphates under neutral conditions: [1,5]-C H insertion of alkylidene carbenes generated by tetrazole fragme... von Yoneyama, Hiroki, Uemura, Kenji, Usami, Yoshihide, Harusawa, Shinya

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Histamine H3 receptor antagonist OUP-186 attenuates the proliferation of cultured human breast cancer cell lines von Tanaka, Satoshi, Sakaguchi, Minoru, Yoneyama, Hiroki, Usami, Yoshihide, Harusawa, Shinya

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Synthesis of Dihydrooxepino[3,2-c]Pyrazoles via Claisen Rearrangement and Ring-Closing Metathesis from 4-Allyloxy-1H-pyrazoles von Usami, Yoshihide, Kohno, Aoi, Yoneyama, Hiroki, Harusawa, Shinya

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Synthesis of 6-Halo-Substituted Pericosine A and an Evaluation of Their Antitumor and Antiglycosidase Activities von Usami, Yoshihide, Mizobuchi, Yoshino, Ijuin, Mai, Yamada, Takeshi, Morita, Mizuki, Mizuki, Koji, Yoneyama, Hiroki, Harusawa, Shinya

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Synthesis and structure–activity relationships of tetrazolato-bridged dinuclear platinum(II) complexes: A small modification at tetrazole C5 markedly influences the in vivo antitum... von Komeda, Seiji, Yoneyama, Hiroki, Uemura, Masako, Tsuchiya, Takahiro, Hoshiyama, Miyuu, Sakazaki, Tomoya, Hiramoto, Keiichi, Harusawa, Shinya

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Synthesis of Dihydropyrano[3,2- c ]pyrazoles via Double Bond Migration and Ring-Closing Metathesis von Usami, Yoshihide, Sumimoto, Kodai, Kishima, Azusa, Tatsui, Yuya, Yoneyama, Hiroki, Harusawa, Shinya

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Specific Conformational Change in Giant DNA Caused by Anticancer Tetrazolato-Bridged Dinuclear Platinum(II) Complexes: Middle-Length Alkyl Substituents Exhibit Minimum Effect von Komeda, Seiji, Yoneyama, Hiroki, Uemura, Masako, Muramatsu, Akira, Okamoto, Naoto, Konishi, Hiroaki, Takahashi, Hiroyuki, Takagi, Akimitsu, Fukuda, Wakao, Imanaka, Tadayuki, Kanbe, Toshio, Harusawa, Shinya, Yoshikawa, Yuko, Yoshikawa, Kenichi

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CuI-Catalyzed Coupling Reactions of 4-Iodopyrazoles and Alcohols: Application toward Withasomnine and Homologs von Usami, Yoshihide, Kubo, Yumika, Takagaki, Toshiki, Kuroiwa, Nao, Ono, Jun, Nishikawa, Kohei, Nakamizu, Ayaka, Tatsui, Yuya, Harusawa, Shinya, Hayama, Noboru, Yoneyama, Hiroki

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Syntheses and Glycosidase Inhibitory Activities, and in Silico Docking Studies of Pericosine E Analogs Methoxy-Substituted at C6 von Usami, Yoshihide, Higuchi, Megumi, Mizuki, Koji, Yamamoto, Mizuki, Kanki, Mao, Nakasone, Chika, Sugimoto, Yuya, Shibano, Makio, Uesawa, Yoshihiro, Nagai, Junko, Yoneyama, Hiroki, Harusawa, Shinya

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Synthesis of Marine Natural Product (−)-Pericosine E von Mizuki, Koji, Iwahashi, Kaoru, Murata, Naoko, Ikeda, Mayuko, Nakai, Yutaka, Yoneyama, Hiroki, Harusawa, Shinya, Usami, Yoshihide

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Synthesis of Natural O-Linked Carba-Disaccharides, (+)- and (-)-Pericosine E, and Their Analogues as α-Glucosidase Inhibitors von Usami, Yoshihide, Mizuki, Koji, Kawahata, Rikiya, Shibano, Makio, Sekine, Atsuko, Yoneyama, Hiroki, Harusawa, Shinya

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Data on synthesis and structure–activity relationships of tetrazolato-bridged dinuclear platinum(II) complexes von Komeda, Seiji, Yoneyama, Hiroki, Uemura, Masako, Tsuchiya, Takahiro, Hoshiyama, Miyuu, Sakazaki, Tomoya, Hiramoto, Keiichi, Harusawa, Shinya

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In Vitro Cytotoxicity and In Vivo Antitumor Efficacy of Tetrazolato-Bridged Dinuclear Platinum(II) Complexes with a Bulky Substituent at Tetrazole C5 von Komeda, Seiji, Uemura, Masako, Yoneyama, Hiroki, Harusawa, Shinya, Hiramoto, Keiichi

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Generation of Alkylidene Carbenes through Tetrazole Fragmentation: Recent Advances and Applications in Organic Synthesis von Harusawa, Shinya, Yoneyama, Hiroki, Usami, Yoshihide

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Synthesis of C4-Linked C0- and C2-Imidazole 2′-Deoxyribonucleoside Phos­phoramidites and Imidazole Base-Pairing Effects on DNA von Harusawa, Shinya, Yoneyama, Hiroki, Usami, Yoshihide, Yamamoto, Daisuke, Zhao, Zheng-yun

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Divergent Synthesis and Evaluation of Inhibitory Activities against Cyclooxygenases-1 and -2 of Natural Withasomnines and Analogues von Usami, Yoshihide, Watanabe, Ryo, Fujino, Yuiko, Shibano, Makio, Ishida, Chihiro, Yoneyama, Hiroki, Harusawa, Shinya, Ichikawa, Hayato

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Transformation of Benzaldehydes to Benzonitriles via Cyanophosphates without One-Carbon Homologation von Yoneyama, Hiroki, Okada, Ayami, Hayama, Noboru, Harusawa, Shinya, Usami, Yoshihide

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Introduction of Fluorine into Antitumor-Active Dinuclear Platinum(II) Complexes Leads to Modulation of In Vivo Antitumor Activity in Mice von Uemura, Masako, Hiramoto, Keiichi, Yoneyama, Hiroki, Harusawa, Shinya, Komeda, Seiji

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