Ligand‐Promoted Non‐Directed C−H Cyanation of Arenes von Liu, Luo‐Yan, Yeung, Kap‐Sun, Yu, Jin‐Quan

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A Survey of the Role of Noncovalent Sulfur Interactions in Drug Design von Beno, Brett R, Yeung, Kap-Sun, Bartberger, Michael D, Pennington, Lewis D, Meanwell, Nicholas A

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meta‐Selective C−H Arylation of Fluoroarenes and Simple Arenes von Liu, Luo‐Yan, Qiao, Jennifer X., Yeung, Kap‐Sun, Ewing, William R., Yu, Jin‐Quan

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Ligand‐Enabled β‐C(sp3)−H Lactamization of Tosyl‐Protected Aliphatic Amides Using a Practical Oxidant von Zhuang, Zhe, Liu, Shuang, Cheng, Jin‐Tang, Yeung, Kap‐Sun, Qiao, Jennifer X., Meanwell, Nicholas A., Yu, Jin‐Quan

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Ligand-accelerated non-directed C–H functionalization of arenes von Wang, Peng, Verma, Pritha, Xia, Guoqin, Shi, Jun, Qiao, Jennifer X., Tao, Shiwei, Cheng, Peter T. W., Poss, Michael A., Farmer, Marcus E., Yeung, Kap-Sun, Yu, Jin-Quan

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Diverse ortho-C(sp2)–H Functionalization of Benzaldehydes Using Transient Directing Groups von Liu, Xi-Hai, Park, Hojoon, Hu, Jun-Hao, Hu, Yan, Zhang, Qun-Liang, Wang, Bao-Long, Sun, Bing, Yeung, Kap-Sun, Zhang, Fang-Lin, Yu, Jin-Quan

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A General Amino Acid Synthesis Enabled by Innate Radical Cross‐Coupling von Ni, Shengyang, Garrido‐Castro, Alberto F., Merchant, Rohan R., de Gruyter, Justine N., Schmitt, Daniel C., Mousseau, James J., Gallego, Gary M., Yang, Shouliang, Collins, Michael R., Qiao, Jennifer X., Yeung, Kap‐Sun, Langley, David R., Poss, Michael A., Scola, Paul M., Qin, Tian, Baran, Phil S.

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Rational Development of Remote C−H Functionalization of Biphenyl: Experimental and Computational Studies von Fan, Zhoulong, Bay, Katherine L., Chen, Xiangyang, Zhuang, Zhe, Park, Han Seul, Yeung, Kap‐Sun, Houk, K. N., Yu, Jin‐Quan

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meta C–H Arylation of Electron-Rich Arenes: Reversing the Conventional Site Selectivity von Liu, Luo-Yan, Qiao, Jennifer X, Yeung, Kap-Sun, Ewing, William R, Yu, Jin-Quan

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Remote C−H Olefination of Heterocyclic Biaryls Enabled by Reversibly Bound Templates von Liu, Luo‐Yan, Fan, Zhoulong, Hoque, Md Emdadul, Qian, Shaoqun, Meng, Guangrong, Chekshin, Nikita, Tanaka, Keita, Qiao, Jennifer X., Yeung, Kap‐Sun, Yu, Jin‐Quan

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Advances in the Total Synthesis of Biologically Important Marine Macrolides von Yeung, Kap-Sun, Paterson, Ian

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Special issue of Medicinal Chemistry Research in honor of Dr. Nicholas A. Meanwell von Kadow, John F., Yeung, Kap-Sun, Murali Dhar, T. G.

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β‐Selective C−H Arylation of Electron‐Deficient Thiophenes, Pyrroles, and Furans von Liu, Luo‐Yan, Qiao, Jennifer X., Ewing, William R., Yeung, Kap‐Sun, Yu, Jin‐Quan

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Actin-Binding Marine Macrolides: Total Synthesis and Biological Importance von Yeung, Kap-Sun, Paterson, Ian

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PdII‐Catalyzed Enantioselective C(sp3)–H Arylation of Cyclobutyl Ketones Using a Chiral Transient Directing Group von Xiao, Li‐Jun, Hong, Kai, Luo, Fan, Hu, Liang, Ewing, William R., Yeung, Kap‐Sun, Yu, Jin‐Quan

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Discovery and Preclinical Characterization of the Cyclopropylindolobenzazepine BMS-791325, A Potent Allosteric Inhibitor of the Hepatitis C Virus NS5B Polymerase von Gentles, Robert G., Ding, Min, Bender, John A., Bergstrom, Carl P., Grant-Young, Katharine, Hewawasam, Piyasena, Hudyma, Thomas, Martin, Scott, Nickel, Andrew, Regueiro-Ren, Alicia, Tu, Yong, Yang, Zhong, Yeung, Kap-Sun, Zheng, Xiaofan, Chao, Sam, Sun, Jung-Hui, Beno, Brett R., Camac, Daniel M., Chang, Chong-Hwan, Gao, Mian, Morin, Paul E., Sheriff, Steven, Tredup, Jeff, Wan, John, Witmer, Mark R., Xie, Dianlin, Hanumegowda, Umesh, Knipe, Jay, Mosure, Kathy, Santone, Kenneth S., Parker, Dawn D., Zhuo, Xiaoliang, Lemm, Julie, Liu, Mengping, Pelosi, Lenore, Rigat, Karen, Voss, Stacey, Wang, Yi, Wang, Ying-Kai, Colonno, Richard J., Gao, Min, Roberts, Susan B., Gao, Qi, Ng, Alicia, Meanwell, Nicholas A, Kadow, John F.

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Discovery of a Hepatitis C Virus NS5B Replicase Palm Site Allosteric Inhibitor (BMS-929075) Advanced to Phase 1 Clinical Studies von Yeung, Kap-Sun, Beno, Brett R, Parcella, Kyle, Bender, John A, Grant-Young, Katherine A, Nickel, Andrew, Gunaga, Prashantha, Anjanappa, Prakash, Bora, Rajesh Onkardas, Selvakumar, Kumaravel, Rigat, Karen, Wang, Ying-Kai, Liu, Mengping, Lemm, Julie, Mosure, Kathy, Sheriff, Steven, Wan, Changhong, Witmer, Mark, Kish, Kevin, Hanumegowda, Umesh, Zhuo, Xiaoliang, Shu, Yue-Zhong, Parker, Dawn, Haskell, Roy, Ng, Alicia, Gao, Qi, Colston, Elizabeth, Raybon, Joseph, Grasela, Dennis M, Santone, Kenneth, Gao, Min, Meanwell, Nicholas A, Sinz, Michael, Soars, Matthew G, Knipe, Jay O, Roberts, Susan B, Kadow, John F

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Pd(II)-Catalyzed Enantioselective C(sp3)−H Arylation of Cyclobutyl Ketones Using a Chiral Transient Directing Group von Xiao, Li-Jun, Hong, Kai, Luo, Fan, Hu, Liang, Ewing, William R., Yeung, Kap-Sun, Yu, Jin-Quan

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A tautomeric ligand enables directed C‒H hydroxylation with molecular oxygen von Li, Zhen, Wang, Zhen, Chekshin, Nikita, Qian, Shaoqun, Qiao, Jennifer X., Cheng, Peter T., Yeung, Kap-Sun, Ewing, William R., Yu, Jin-Quan

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Pd II -Catalyzed Enantioselective C(sp 3 )-H Arylation of Cyclobutyl Ketones Using a Chiral Transient Directing Group von Xiao, Li-Jun, Hong, Kai, Luo, Fan, Hu, Liang, Ewing, William R, Yeung, Kap-Sun, Yu, Jin-Quan

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